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A Study of VX-445 Combination Therapy in CF Subjects Homozygous for F508del (F/F)

Phase 3
Completed
Conditions
Cystic Fibrosis
Interventions
Drug: TEZ/IVA
Drug: VX-445/TEZ/IVA
Drug: IVA
Drug: Placebo
Registration Number
NCT03525548
Lead Sponsor
Vertex Pharmaceuticals Incorporated
Brief Summary

This study will evaluate the efficacy of VX-445 in triple combination (TC) with tezacaftor (TEZ) and ivacaftor (IVA) in subjects with cystic fibrosis (CF) who are homozygous for the F508del mutation (F/F)

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
113
Inclusion Criteria
  • Homozygous for the F508del mutation (F/F)
  • Forced expiratory volume in 1 second (FEV1) value ≥40% and ≤90% of predicted mean for age, sex, and height

Key

Exclusion Criteria
  • Clinically significant cirrhosis with or without portal hypertension
  • Lung infection with organisms associated with a more rapid decline in pulmonary status
  • Solid organ or hematological transplantation

Other protocol defined Inclusion/Exclusion criteria may apply

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
TEZ/IVATEZ/IVAFollowing a run-in period of 4 weeks with Tezacaftor (TEZ)/Ivacaftor (IVA), participants received TEZ 100 milligram (mg)/IVA 150 mg as fixed-dose combination (FDC) tablet in the morning and IVA 150 mg as mono tablet in the evening for 4 weeks in the triple combination (TC) treatment period.
TEZ/IVAPlaceboFollowing a run-in period of 4 weeks with Tezacaftor (TEZ)/Ivacaftor (IVA), participants received TEZ 100 milligram (mg)/IVA 150 mg as fixed-dose combination (FDC) tablet in the morning and IVA 150 mg as mono tablet in the evening for 4 weeks in the triple combination (TC) treatment period.
VX-445/TEZ/IVA TCPlaceboFollowing a run-in period of 4 weeks with TEZ/IVA, participants received VX-445 200 mg/TEZ 100 mg/IVA 150 mg as FDC tablets in the morning and IVA 150 mg as mono tablet in the evening for 4 weeks in the TC treatment period.
TEZ/IVAIVAFollowing a run-in period of 4 weeks with Tezacaftor (TEZ)/Ivacaftor (IVA), participants received TEZ 100 milligram (mg)/IVA 150 mg as fixed-dose combination (FDC) tablet in the morning and IVA 150 mg as mono tablet in the evening for 4 weeks in the triple combination (TC) treatment period.
VX-445/TEZ/IVA TCVX-445/TEZ/IVAFollowing a run-in period of 4 weeks with TEZ/IVA, participants received VX-445 200 mg/TEZ 100 mg/IVA 150 mg as FDC tablets in the morning and IVA 150 mg as mono tablet in the evening for 4 weeks in the TC treatment period.
VX-445/TEZ/IVA TCIVAFollowing a run-in period of 4 weeks with TEZ/IVA, participants received VX-445 200 mg/TEZ 100 mg/IVA 150 mg as FDC tablets in the morning and IVA 150 mg as mono tablet in the evening for 4 weeks in the TC treatment period.
Primary Outcome Measures
NameTimeMethod
Absolute Change in Percent Predicted Forced Expiratory Volume in 1 Second (ppFEV1)From Baseline at Week 4

FEV1 is the volume of air that can forcibly be blown out in one second, after full inspiration.

Secondary Outcome Measures
NameTimeMethod
Observed Pre-Dose Concentration (Ctrough) of VX-445, TEZ, TEZ Metabolite (M1-TEZ), and IVADay 1 and Week 4
Safety and Tolerability as Assessed by Number of Participants With Treatment-Emergent Adverse Events (AEs) and Serious Adverse Events (SAEs)From first dose of study drug in TC treatment period up to 28 days after last dose of study drug or to the completion of study participation date, whichever occurs first (up to Week 8)
Absolute Change in Sweat Chloride (SwCl)From Baseline at Week 4

Sweat samples were collected using an approved collection device.

Absolute Change in Cystic Fibrosis Questionnaire-Revised (CFQ-R) Respiratory Domain ScoreFrom Baseline at Week 4

The CFQ-R is a validated participant-reported outcome measuring health-related quality of life for participants with cystic fibrosis. Respiratory domain assessed respiratory symptoms, score range: 0-100; higher scores indicate fewer symptoms and better health-related quality of life.

Trial Locations

Locations (44)

Universitair Ziekenhuis Brussel - Campus Jette

🇧🇪

Brussels, Belgium

UZ Antwerpen

🇧🇪

Edegem, Belgium

Universitair Ziekenhuis Gent

🇧🇪

Gent, Belgium

HagaZiekenhuis van den Haag

🇳🇱

Den Haag, Netherlands

University of Virginia Primary Care Center

🇺🇸

Charlottesville, Virginia, United States

Universitaire Ziekenhuizen Leuven - Campus Gasthuisberg

🇧🇪

Leuven, Belgium

Heart of England NHS Foundation Trust, Birmingham Heartlands Hospital

🇬🇧

Birmingham, United Kingdom

Academic Medical Center

🇳🇱

Amsterdam, Netherlands

The Royal Belfast Hospital for Sick Children

🇬🇧

Belfast, United Kingdom

Cliniques Universitaires de Bruxelles Hopital Erasme

🇧🇪

Brussels, Belgium

University of Arkansas for Medical Sciences

🇺🇸

Little Rock, Arkansas, United States

Banner University of Arizona Medical Center

🇺🇸

Tucson, Arizona, United States

University Medical Center, Utrecht, Department of Pulmonology and Tuberculosis

🇳🇱

Heidelberglaan, Netherlands

Southampton General Hospital

🇬🇧

Southampton, United Kingdom

Leeds General Infirmary

🇬🇧

Leeds, United Kingdom

UMC St. Radboud

🇳🇱

Nijmegen, Netherlands

Erasmus Medical Center

🇳🇱

Rotterdam, Netherlands

Tulane Medical Center

🇺🇸

New Orleans, Louisiana, United States

ProMedica Toledo Hospital/ Toledo Children's Hospital/ Pediatric Pulmonary & Cystic Fibrosis Center

🇺🇸

Toledo, Ohio, United States

Royal Devon and Exeter NHS Foundation Trust, Royal Devon and Exeter Hospital

🇬🇧

Exeter, United Kingdom

King's College Hospital

🇬🇧

London, United Kingdom

Saint Francis Medical Center/ Children's Hospital of Illinoise/OSF

🇺🇸

Peoria, Illinois, United States

Miller Children's Hospital/ Long Beach Memorial

🇺🇸

Long Beach, California, United States

Children's Hospital Los Angeles

🇺🇸

Los Angeles, California, United States

Valley Children's Hospital

🇺🇸

Madera, California, United States

Northwestern Memorial Hospital

🇺🇸

Chicago, Illinois, United States

Harper University Hospital

🇺🇸

Detroit, Michigan, United States

UNC Marisco Clinical Research Center

🇺🇸

Chapel Hill, North Carolina, United States

Nationwide Children's Hospital

🇺🇸

Columbus, Ohio, United States

National Jewish Health

🇺🇸

Denver, Colorado, United States

Tampa General Hospital Cardiac and Lung Transplant Clinic

🇺🇸

Tampa, Florida, United States

Joe DiMaggio Cystic Fibrosis & Pulmonary Center/ Joe DiMaggio Children's Hospital/ Memorial Regional Hospital

🇺🇸

Hollywood, Florida, United States

Rainbow Babies and Children's Hospital/University Hospitals Cleveland Medical Center

🇺🇸

Cleveland, Ohio, United States

Central Florida Pulmonary Group, PA

🇺🇸

Orlando, Florida, United States

Massachusetts General Hospital Cystic Fibrosis Center Clinical Research Center

🇺🇸

Boston, Massachusetts, United States

The University of Texas Southwestern Medical Center

🇺🇸

Dallas, Texas, United States

Nemours Children's Hospital

🇺🇸

Orlando, Florida, United States

New York Medical College

🇺🇸

Valhalla, New York, United States

Children's Hospital of Philadelphia

🇺🇸

Philadelphia, Pennsylvania, United States

Medical University of South Carolina

🇺🇸

Charleston, South Carolina, United States

West Virginia University

🇺🇸

Morgantown, West Virginia, United States

University of Oklahoma Health Sciences Center

🇺🇸

Oklahoma City, Oklahoma, United States

Vermont Lung Center

🇺🇸

Colchester, Vermont, United States

Dayton Children's Hospital

🇺🇸

Dayton, Ohio, United States

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