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Evaluation of TRC101 in Subjects With Chronic Kidney Disease and Metabolic Acidosis

Phase 1
Completed
Conditions
Acidosis
Interventions
Drug: Placebo
Registration Number
NCT02809183
Lead Sponsor
Tricida, Inc.
Brief Summary

This was a double-blind, placebo-controlled, parallel-design, 6-arm, fixed dose study. The study enrolled 135 adult male and female subjects with Stage 3 or 4 chronic kidney disease and low serum bicarbonate levels. The study was conducted in two parts. In Part 1 study drug dosing (TRC101 or placebo) continued for 14 days twice daily (BID). In Part 2 study drug dosing (TRC101 or placebo) continued for 14 days once daily (QD).

The maximum study duration per subject was anticipated to be up to 42 days.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
135
Inclusion Criteria
  • Estimated glomerular filtration rate (eGFR) of 20 to <60 mL/min/1.73m2
  • Serum bicarbonate level of 12 to 20 mEq/L
Exclusion Criteria
  • Any level of low serum bicarbonate that, in the opinion of the Investigator, requires emergency intervention.
  • Severe comorbid conditions other than chronic kidney disease.
  • Chronic obstructive pulmonary disease.
  • Anticipated changes in doses of any of the following drugs or drug classes: diuretics, non-ophthalmic carbonic anhydrase inhibitors, oral diabetes drugs, antihypertensive drugs, antacids, H2-blockers, or proton pump inhibitors.
  • Excluded drugs or drug classes: insulin, non-daily or "as needed" diuretics, herbal products, dietary supplements, multivitamins, naturopathic remedies, sodium bicarbonate, potassium citrate, sodium citrate or other alkali therapy, non-steroidal anti-inflammatory drugs (NSAIDs), fiber supplements, laxatives, calcium and magnesium supplements, or electrolyte binders and other binder drugs.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Placebo-BIDPlaceboAdministered twice daily (BID) for 14 days
TRC101 (1.5g BID)TRC101Administered twice daily (BID) for 14 days
TRC101 (3g BID)TRC101Administered twice daily (BID) for 14 days
TRC101 (4.5g BID)TRC101Administered twice daily (BID) for 14 days
TRC101 (6g QD)TRC101Administered once daily (QD) for 14 days
Placebo-QDPlaceboAdministered once daily (QD) for 14 days
Primary Outcome Measures
NameTimeMethod
Number of Subjects With Treatment Emergent Adverse Events (TEAEs) and Number of Subjects Who Discontinued Study Drug Due to a TEAEThrough treatment period completion (Day 15)

The number and percentage of subjects who reported treatment-emergent adverse events (TEAEs) summarized by system organ class and preferred term (see Reported Adverse Events) as well as by severity, causality, seriousness, and action taken with regard to study drug. All analyses were descriptive.

Change From Baseline to the End of Treatment (Day 15) in Serum Bicarbonate Within Each Individual TRC101 Dose GroupBaseline and Day 15

Serum bicarbonate at Day 15 minus serum bicarbonate at Baseline

Secondary Outcome Measures
NameTimeMethod
Change From Baseline in Serum Bicarbonate at Day 15 Within the Combined TRC101 Treatment GroupBaseline and Day 15

Serum bicarbonate at Day 15 minus serum bicarbonate at Baseline

Comparison of Change From Baseline in Serum Bicarbonate at Day 15 Between the Combined TRC101 Treatment Group Versus PlaceboBaseline and Day 15

Serum bicarbonate at Day 15 minus serum bicarbonate at Baseline for the Combined TRC101 Treatment Group versus that for Placebo

Change From Baseline in Serum Bicarbonate at Day 15 Within the TRC101 6g QD Dose GroupBaseline and Day 15

Serum bicarbonate at Day 15 minus serum bicarbonate at Baseline

Change From Baseline in Serum Bicarbonate at Day 15 Comparison Between the TRC101 6g QD Dose Group Versus PlaceboBaseline and Day 15

Serum bicarbonate at Day 15 minus serum bicarbonate at Baseline for the TRC101 6g dose group versus that for Placebo

Change From Baseline in Serum Bicarbonate at Day 15 Comparison Between the TRC101 6g QD Dose Group Versus the TRC101 3g BID Dose GroupBaseline and Day 15

Serum bicarbonate at Day 15 minus serum bicarbonate at Baseline for the TRC101 6g QD dose group versus that for the TRC101 3g BID dose group

Comparison of Change From Baseline in Serum Bicarbonate at Day 15 Between Each TRC101 Dose Group Versus PlaceboBaseline and Day 15

Serum bicarbonate at Day 15 minus serum bicarbonate at Baseline for each TRC101 dose group versus that for Placebo

Comparison of the Proportion of Subjects Whose Serum Bicarbonate Values Increased From Baseline to Day 15 by Greater Than or Equal to 2, 3, or 4 mEq/L Between Each TRC101 Dose Group Versus PlaceboBaseline and Day 15

Comparison of the proportion of subjects whose serum bicarbonate values increased from Baseline to Day 15 by greater than or equal to 2, 3, or 4 mEq/L between each TRC101 BID Dose Group versus Placebo

Comparison of the Proportion of Subjects in the TRC101 6g QD Dose Group Whose Serum Bicarbonate Values Increased From Baseline to Day 15 by Greater Than or Equal to 2, 3, or 4 mEq/L Versus PlaceboBaseline and Day 15

Comparison of the proportion of subjects whose serum bicarbonate values increased from Baseline to Day 15 by greater than or equal to 2, 3, or 4 mEq/L between the 6g TRC101 QD Dose Group versus Placebo

Trial Locations

Locations (5)

Investigative Site 3

🇬🇪

Tbilisi, Georgia

Investigative Site 6

🇬🇪

Tbilisi, Georgia

Investigative Site 1

🇧🇬

Sofia, Bulgaria

Investigative Site 5

🇬🇪

Tbilisi, Georgia

Investigative Site 4

🇬🇪

Tbilisi, Georgia

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