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Study to Evaluate Safety and Efficacy of UB-421 Antibody in HIV-1 Infected Adults

Phase 2
Completed
Conditions
HIV-1 Infection in Adults
Interventions
Drug: Antibody UB-421
Registration Number
NCT01668043
Lead Sponsor
United Biomedical
Brief Summary

The purpose of this Phase IIa study is to determine whether the antibody (UB-421), targeting the HIV-1 receptor on the CD4 molecule of T-lymphocytes and monocytes, is safe and effective when multiple doses are administered by intravenous infusion to asymptomatic HIV-1 infected adults and to assess pharmacokinetic parameters of the antibody in blood and on cells. The neutralizing activity of UB-421 blocks HIV-1 from binding to its receptor on CD4-positive cells; thus, UB-421 functions as an immunotherapeutic intervention to prevent HIV-1 infection.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
29
Inclusion Criteria
  • Asymptomatic, treatment-naive, HIV-1 seropositive
  • CD4+ T cell count >350 cells/cubic millimeter
  • HIV-1 viral load >5,000 copies/mL
  • Other inclusion criteria apply
Exclusion Criteria
  • Active infection requiring immediate therapy (except HIV-1)
  • Previous exposure to monoclonal antibody (including UB-421)
  • Prior participation in any HIV vaccine trial
  • Use of immunomodulating drugs or systemic chemotherapy
  • Other exclusion criteria apply

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Antibody UB-421 Cohort 2Antibody UB-42125 mg/kg BW, 4 biweekly doses for 8-week treatment period
Antibody UB-421 Cohort 1Antibody UB-42110 mg/kg BW, 8 weekly doses for 8-week treatment period
Primary Outcome Measures
NameTimeMethod
To evaluate safety and tolerability of multiple intravenous infusions of two dose cohorts of UB-42116-week study period

Safety evaluations include physical examination, measurement of vital signs, clinical chemistry and hematology tests at each visit (to assess changes from normal range), incidence of adverse event (AE) and serious AE (SAE) of two dose cohorts and are followed for 16 weeks (end of study).

Overall treatment tolerability of UB-421 for each cohort is defined as the percentage of the number of actual infusion doses divided by number of actual infusion doses plus number of missed doses of subject(s) who drops out due to drug-related AE(s); calculation follows specific formula.

To evaluate efficacy by measurement of individual maximal viral load reduction and mean maximal viral load reduction of two dose cohorts of UB-421.16-week study period

Efficacy measurements include virologic responses and determination of the proportion of subjects with viral load \<50 copies/mL or \<200 copies/mL; viral load reduction \>0.5 log10 copies/mL or \>1.0 log10 copies/mL; viral rebound over 0.5 log10 increase in viral load from the nadir value during 8-week treatment period, suggesting presence of study drug resistance mutants. HIV-1 viral load is determined at each blood collection during 16-week study period.

Secondary Outcome Measures
NameTimeMethod
To determine pharmacokinetic parameters of two dose cohorts of UB-421.16-week study period

Pharmacokinetic analyses are calculated at each visit during 8-week treatment period to determine the serum concentration before and after each infusion of UB-421 and during the 8-week follow-up period to determine the clearance of study drug in circulation.

To determine the anti-UB-421 antibody concentration in serum of two dose cohorts of UB-42116-week study period

Immunogenicity of the study drug is measured by analytical ELISA test at each visit to determine if the anti-UB-421 antibody concentration is increased above the pre-treatment baseline level.

Trial Locations

Locations (2)

Taipei Veterans General Hospital (TVGH)

🇨🇳

Taipei City, Beitou District, Taiwan

Kaohsiung Veterans General Hospital (KVGH)

🇨🇳

Kaohsiung City, Zuoying District, Taiwan

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