MedPath

Azithromycin for Acute Exacerbations Requiring Hospitalization

Phase 3
Terminated
Conditions
Chronic Obstructive Pulmonary Disease
Interventions
Drug: Placebo
Registration Number
NCT02135354
Lead Sponsor
Wim Janssens
Brief Summary

This project (funded by the IWT-TBM program) will organize a randomized placebo-controlled multicenter intervention trial in 500 COPD patients to study the effectiveness and safety of azithromycin therapy in the acute setting of COPD exacerbations requiring hospital admission. Although long-term use of azithromycin is proven effective to prevent exacerbations, inherent risks outweigh the benefits. By reducing the dose and duration of the azithromycin treatment and by restricting the treatment to acute periods with highest risk for treatment failure, benefits may counterbalance potential side effects, which may result in a new treatment strategy for these acute events.

The present study is designed by the services of respiratory medicine of the Leuven and Ghent University hospitals but will run in total in 17 different large hospitals in Belgium, of which 12 are located in Flanders.

Detailed Description

In this 9 month, randomized, placebo-controlled, parallel-group, multicenter intervention trial, 500 patients will be randomly assigned (1:1 ratio) to receive either azithromycin or placebo on top of standard therapy in the acute treatment of COPD exacerbations requiring hospitalization. The study drug (azithromycin or placebo) will be initiated and uploaded within 48 hours after hospital admission (500mg once a day for 3 days) and subsequently administered for a prolonged period of 3 months at a lower maintenance dose (250mg every 2 days). An additional follow-up period of 6 months without study drug will be foreseen to study relapse after study drug withdrawal.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
301
Inclusion Criteria
  • Established diagnosis of COPD by medical doctor (based on clinical history OR pulmonary function test)
  • Smoking history of at least 10 pack-years (10 pack-years are defined as 20 cigarettes a day for 10 years, or 10 cigarettes a day for 20 years, etc.)
  • Current hospitalization for potential infectious AECOPD treated with standard therapy
  • History of at least one exacerbation during the last year (prior to the current hospital admission) for which systemic steroids and/or antibiotics were taken
  • ECG at admission
Exclusion Criteria
  • Mechanical or non-invasive ventilation at moment of randomization (D1)
  • Long QT interval on ECG (QTc > 450msec for males or > 470msec for females)
  • History of life-threatening arrhythmias
  • Myocardial infarction (NSTEMI or STEMI) less than 6 weeks before start of study drug
  • Unstable angina pectoris or acute myocardial infarction (NSTEMI or STEMI) at admission
  • Drugs with high risk for long QT interval and torsade de pointes (amiodarone, flecainide, procainamide, sotalol, droperidol, haldol, citalopram, other macrolides)
  • Documented uncorrected severe hypokalemia (K+ < 3.0 mmol/L) or hypomagnesemia (Mg2+ < 0.5 mmol/L)
  • Chronic systemic steroids (> 4 mg methylprednisolone /day for ≥ 2 months)
  • Actual use of macrolides for at least 2 weeks
  • Allergy to macrolides
  • Active cancer treatment
  • Life expectancy < 3 months
  • Pregnant or breast-feeding subjects. Woman of childbearing potential must have a pregnancy test performed and a negative result must be documented before start of treatment

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PlaceboPlaceboN = 250 * From day 1 up to and including day 3: 500 mg placebo PO once a day * From day 4 up to and including day 90: 250 mg placebo PO once every 2 days
AzithromycinAzithromycinN = 250 * From day 1 up to and including day 3: 500 mg azithromycin PO once a day * From day 4 up to and including day 90: 250 mg azithromycin PO once every 2 days
Primary Outcome Measures
NameTimeMethod
Time to clinical failureWill be assessed between day 1 (from 1 hour after first drug intake) till day 90 (24 hours after last study drug intake)

Clinical failure is a composite endpoint as multiple clinical interventions may indicate that an initiated therapy is failing. Clinical failure is defined as the composite of death, treatment intensification (additional dose of systemic steroids, switch antibiotics for respiratory reasons or new course of systemic steroids and/or antibiotics) and step up in hospital care for respiratory reasons (from ward to ICU during index event, or from home to ward or ICU (new admission) after discharge).

Primary outcome measure will also be analysed in following subgroups as an exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Secondary Outcome Measures
NameTimeMethod
Total days of additional/prolonged systemic steroid use at Day 90 (key secondary #3)Will be assessed on day 90 (last day of treatment phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Total days of hospital days within 90 and within 270 daysWill be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Total days in intensive care within 90 and within 270 daysWill be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

COPD Assessment Test (CAT) score at Day 90 (key secondary #2)Will be assessed on day 90 (last day of treatment phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Time to first step up in hospital care for respiratory reasons within 90 and within 270 daysWill be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Number of clinical failures up to Day 90 (key secondary #1)Will be assessed on day 90 (last day of treatment phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III

* ICS use vs no ICS use

Quality of Life - 5 Dimensions (EQ5D) score at Day 90 and at Day 270Will be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Speech, Spatial and Qualities of Hearing (SSQ5) score at Day 90 and Day 270Will be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Pre-bronchodilator forced expiratory volume in 1 second (FEV1) at Day 90 and Day 270Will be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Number of clinical failures up to Day 270Will be assessed on day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III

* ICS use vs no ICS use

Time to clinical failure up to Day 90 and up to Day 270Will be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Time to new exacerbation within 90 and within 270 daysWill be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

A new exacerbation is defined as the composite of new course of systemic steroids and/or antibiotics, and hospitalization for respiratory reasons, all after the index event.

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Number of new exacerbations up to 90 days and up to 270 daysWill be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

COPD Assessment Test (CAT) score at Day 270Will be assessed on day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Modified Medical Research Council (mMRC) score at Day 90 and Day 270Will be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Total dose of additional/prolonged systemic steroids at Day 270Will be assessed on day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Total days of additional/prolonged systemic steroid use at Day 270Will be assessed on day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Total days of non-study antibiotic use at Day 90 and Day 270Will be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Number of home physician contacts at Day 90 and Day 270Will be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Average cost of hospitalization at Day 90 and Day 270 including the index hospitalizationWill be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Time to death within 90 and within 270 daysWill be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Time to first treatment intensification within 90 and within 270 daysWill be assessed on day 90 (last day of treatment phase) and day 270 (last day of follow-up phase)

Secondary outcome measure will also be analysed in following subgroups as exploratory analysis:

* Male vs female

* Smoker vs ex-smoker (stopped smoking \> 6 months)

* GOLD A, B vs GOLD C vs GOLD D

* former GOLD I, II vs III vs IV

* High CRP (\> 50 mg/dL) vs low CRP (\< 50 mg/dL)

* Age \> 65 years vs ≤ 65 years

* Anthonissen I vs Anthonissen II vs Anthonissen III at admission

* ICS use vs no ICS use

Trial Locations

Locations (20)

Jessa Ziekenhuis

🇧🇪

Hasselt, Vlaanderen, Belgium

Grand Hôpital de Charleroi

🇧🇪

Gilly, Wallonië, Belgium

St. Augustinus Ziekenhuis

🇧🇪

Antwerpen, Vlaanderen, Belgium

Onze-Lieve-Vrouwziekenhuis

🇧🇪

Aalst, Belgium

AZ Groeninge Ziekenhuis

🇧🇪

Kortrijk, Vlaanderen, Belgium

Heilig Hart Ziekenhuis

🇧🇪

Roeselare, Vlaanderen, Belgium

UZ Gent

🇧🇪

Gent, Vlaanderen, Belgium

UZ Gasthuisberg

🇧🇪

Leuven, Vlaanderen, Belgium

Clinique Reine Astrid

🇧🇪

Malmedy, Belgium

CHU Charleroi

🇧🇪

Charleroi, Wallonië, Belgium

ZNA Middelheim

🇧🇪

Antwerpen, Vlaanderen, Belgium

St. Jan Brugge Ziekenhuis

🇧🇪

Brugge, Vlaanderen, Belgium

Imelda Ziekenhuis

🇧🇪

Bonheiden, Vlaanderen, Belgium

St. Andriesziekenhuis

🇧🇪

Tielt, Vlaanderen, Belgium

UZ Brussel

🇧🇪

Brussel, Brussel Hoofdstedelijk Gewest, Belgium

St. Pieterziekenhuis

🇧🇪

Brussel, Brussels Hoofdstedelijk Gewest, Belgium

Maria Middelaresziekenhuis

🇧🇪

Gent, Vlaanderen, Belgium

CHU Liège

🇧🇪

Liège, Wallonië, Belgium

CHU Mont-Godinne

🇧🇪

Yvoir, Wallonië, Belgium

Clinique Sainte-Elisabeth

🇧🇪

Namur, Belgium

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