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ANAVEX2-73 Study in Parkinson's Disease Dementia

Phase 2
Completed
Conditions
Parkinsons Disease With Dementia
Interventions
Registration Number
NCT03774459
Lead Sponsor
Anavex Life Sciences Corp.
Brief Summary

A Phase 2, Double-Blind, Randomized, Placebo-Controlled Study to Evaluate the Safety, Tolerability, and Efficacy of ANAVEX2-73 for Cognitive Impairment in Patients with Parkinson's Disease with Dementia (PDD)

Detailed Description

This is a Phase 2, multicenter, randomized, double-blind, placebo-controlled, parallel-group, three-arm, 14-week study in PD patients with dementia. The study includes a 2 week Screening / Baseline Observation Period and a 14-week Treatment Period (including a 2 week Titration Period), and a 2-week Safety Follow-Up Period

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
132
Inclusion Criteria
  • Diagnosis of idiopathic Parkinson's disease (PD) consistent with the UK Parkinson's Disease Society Brain Bank diagnostic criteria.

  • Diagnosis of probable PD dementia (PDD) according to the Movement Disorder Society Task Force clinical diagnostic criteria.

  • Montreal Cognitive Assessment (MoCA) score of 13 to 23, inclusive, at Screening.

  • Male or female and aged ≥ 50 years.

  • Caregivers and subjects (or legal representative) must understand and have signed approved informed consent.

  • Caregivers and subjects (or legal representative) must be able to understand study requirements and be willing to follow instructions.

  • Stable regimen of anti-Parkinson's disease medications (including levodopa, dopamine agonists, MAO-B inhibitors, or the COMT inhibitor entacapone), which has been stable for at least 4 weeks prior to Baseline.

  • Treatment with cholinesterase inhibitor (rivastigmine, donepezil and galantamine (Exelon®, Aricept®, or Reminyl®) will be permitted, provided the dose has been stable for a minimum of 8 weeks prior to randomization.

  • Subjects with history of depression on antidepressant medications will be allowed if depression is controlled and they have been on a stable daily dose of the antidepressant for ≥8 weeks before Baseline.

  • Contraception:

    • Women of childbearing potential must use an acceptable method of contraception starting 4 weeks prior to study drug administration and for a minimum of 4 weeks after study completion. Otherwise, women must be postmenopausal (at least one year absence of vaginal bleeding or spotting) as confirmed by FSH greater than or equal to 40 mIU/mL or 40 IU/L or be surgically sterile.
    • Men with a potentially fertile partner must have had a vasectomy or be willing to use an acceptable method of contraception for the duration of the study and for 3 months after study drug discontinuation.
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Exclusion Criteria
  • History of any significant neurologic or psychiatric disorder other than PD that can contribute to cognitive impairment.

  • Any other condition or clinically significant abnormal findings like severe co-morbidities e.g. history of stroke, poor kidney or liver function on the physical or neurological examination, medical and psychiatric history, at screening or at baseline that, in the opinion of the Investigator, would make the subject unsuitable for the study.

  • Potential symptomatic causes of cognitive impairment including but not limited to

    1. abnormal thyroid function test at screening (TSH)
    2. abnormal B12 level at screening
    3. MRI findings (by history) pointing to a potential symptomatic cause of cognitive dysfunction, including significant vascular changes, or communicating hydrocephalus.
  • Treatment with memantine or amantadine. If appropriate the drugs can be discontinued for a minimum of 4 weeks prior to randomization.

  • Use of over the counter (OTC) or prescription medication for sleep on 2 or more occasions per week (less than that is allowed).

  • History of depression as measured by Beck Depression Inventory score >17 at screening.

  • Treatment with any other investigational drug or device within 4 weeks prior to screening.

  • Smoking > 1 pack of cigarettes per day (as assessed for the 4 weeks prior to screening).

  • Women who are pregnant or lactating.

  • Known allergy or sensitivity to ANAVEX2-73 or any of its components.

  • Suicidal ideation on the Columbia Suicide Severity Rating Scale (C-SSRS) of type 4 or type 5, or any suicidal behavior, in the past 6 months. Type 4 indicates active suicidal ideation with some intent to act, without a specific plan. Type 5 indicates active suicidal ideation with a specific plan and intent.

  • Use of centrally acting anticholinergic drugs during the 4 weeks before randomization.

  • Medications used for overactive bladder will be allowed provided that the regimen has been stable 4 weeks prior to randomization.

  • Treatment with any dopamine receptor blocking medications with the exception of low dose quetiapine (≤50 mg/day). Pimavanserin (≤34 mg/day) will be allowed.

  • History of neurosurgical intervention (e.g., deep brain stimulation) for PD.

  • Unpredictable motor fluctuations that would interfere with administering cognitive assessments in the ON state.

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Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Mid dose ANAVEX2-73Mid dose ANAVEX2-73Mid dose ANAVEX2-73
High dose ANAVEX2-73High dose ANAVEX2-73High dose ANAVEX2-73
Placebo oral capsulePlacebo oral capsulePlacebo oral capsule
Primary Outcome Measures
NameTimeMethod
Number of participants with treatment-related adverse events as assessed by CTCAE v4.014 weeks

Assess the safety and tolerability of ANAVEX2-73 compared to placebo

Cognitive Drug Research (CDR) Computerized Assessment System Continuity of Attention14 weeks

Change from Baseline to End of Treatment in Continuity of Attention as measured by Cognitive Drug Research (CDR) Computerized Assessment System Continuity of Attention test

Secondary Outcome Measures
NameTimeMethod
SDS-CL-2514 weeks

Incidence of sleep disorders symptoms (SDS-CL-25)

MDS-UPDRS Part III Total Score (Motor Scores)14 weeks

Change from baseline to End of Treatment as measured by MDS-UPDRS Part III Total Score (Motor Scores)

Trial Locations

Locations (25)

KaRa MINDS

🇦🇺

Macquarie Park, Australia

Hospital Santa Caterina

🇪🇸

Girona, Spain

Clinica Ruber Internacional

🇪🇸

Madrid, Spain

Hospital Mutua Terrasa

🇪🇸

Barcelona, Spain

Hammond Health

🇦🇺

Malvern, Australia

Hospital Cruces Bilbao

🇪🇸

Barakaldo, Spain

Hospital del Henares

🇪🇸

Coslada, Spain

Hospital General Universitario de Elche

🇪🇸

Elche, Spain

Hospital Universitario Vall d'Hebron

🇪🇸

Barcelona, Spain

Hospital Universitario de Burgos

🇪🇸

Burgos, Spain

Hospital Clínico San Carlos

🇪🇸

Madrid, Spain

Hospital de La Princesa

🇪🇸

Madrid, Spain

Hospital General Universitario Gregorio Marañón

🇪🇸

Madrid, Spain

Hospital Universitario Puerta de Hierro

🇪🇸

Madrid, Spain

Hospital Infanta Leónor

🇪🇸

Madrid, Spain

Hospital Universitario Ramón y Cajal

🇪🇸

Madrid, Spain

Hospital HM Puerta del Sur

🇪🇸

Móstoles, Spain

Hospital Universitario Central de Asturias (HUCA)

🇪🇸

Oviedo, Spain

Clínica Universidad de Navarra (CUN)

🇪🇸

Pamplona, Spain

Hospital de Santiago de Compostela

🇪🇸

Santiago de Compostela, Spain

Hospital Universitario Virgen del Rocío

🇪🇸

Sevilla, Spain

Clínica Universidad de Navarra (CUN) - Sede Madrid- Servicio de Neurología -

🇪🇸

Madrid, Spain

Hospital Universitario Puerta del Mar

🇪🇸

Cadiz, Spain

Hospital Arquitecto Marcide

🇪🇸

Ferrol, Spain

Hospital de la Santa Creu i Sant Pau

🇪🇸

Barcelona, Spain

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