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SOLUTION: Study of Oral Liprotamase Unit-Matched Therapy Of Non-Porcine Origin in Patients With Cystic Fibrosis

Phase 3
Completed
Conditions
Exocrine Pancreatic Insufficiency
Cystic Fibrosis
Interventions
Drug: Liprotamase
Drug: porcine (pig) PERT
Registration Number
NCT02279498
Lead Sponsor
Anthera Pharmaceuticals
Brief Summary

Liprotamase powder is a non-porcine, soluble and stable mixture of three digestive enzymes including lipase, protease, and amylase. The purpose of the present study is to provide additional efficacy and safety data compared to approved, porcine-derived, enterically-coated and encapsulated pancreatic enzyme replacement therapy. The primary efficacy endpoint of the study will be comparative efficacy measured as the change in the coefficient of fat absorption (CFA) in Cystic Fibrosis patients with exocrine pancreatic insufficiency (EPI).

Liprotamase is stable in stomach and digestive fluids allowing administration in a variety of convenient formulations and with a number of foods without enteric coating.

Detailed Description

Porcine derived enzymes are used for pancreatic enzyme replacement therapy in patients with cystic fibrosis (CF). Liprotamase is a biotechnology-derived enzyme replacement without enteric coating. This is an open-label, assessor blind, parallel group, multicenter, international trial to evaluate the noninferiority of liprotamase and pancrelipase in CF patients aged ≥7 years with pancreatic insufficiency. Subjects were randomized to liprotamase or pancrelipase, dose-matched to pre-study lipase doses. The lower bound of the 95% confidence interval (CI) for noninferiority was -15% for treatment difference in change from baseline coefficient of fat absorption (CFA).

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
128
Inclusion Criteria
  • Diagnosis of Cystic Fibrosis based on presentation, genotype and/or sweat chloride
  • Fecal elastase <100 mcg/g stool
  • Minimum Coefficient of Fat (CFA) at screening while on stable PERT therapy
  • Good nutritional status
Read More
Exclusion Criteria
  • History or diagnosis of fibrosing colonopathy
  • Distal intestinal obstruction syndrome in 6 months prior to screening
  • Receiving enteral tube feedings
  • Chronic diarrheal illness unrelated to pancreatic insufficiency
  • Liver abnormalities, or liver or lung transplant, or significant bowel resection
  • Forced expiratory volume in 1 second (FEV1) <30%
Read More

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
LiprotamaseLiprotamaseIndividually-optimized dose to be administered orally
porcine (pig) PERTporcine (pig) PERTIndividually-optimized dose to be administered orally
Primary Outcome Measures
NameTimeMethod
Treatment Difference in Coefficient of Fat Absorption (CFA) Change From BaselineBaseline, 7 weeks

The primary endpoint evaluates the difference between treatment arms in change from baseline in coefficient of fat absorption (CFA). As such, descriptive statistics for individual treatment arms are not provided in this measure, but are reported in the secondary endpoints

Secondary Outcome Measures
NameTimeMethod
Coefficient of Nitrogen Absorption (CNA)Baseline, 7 weeks

Change from baseline in coefficient of nitrogen absorption

Coefficient of Fat Absorption (CFA)Baseline, 7 weeks

Change from baseline in coefficient of fat absorption

Trial Locations

Locations (54)

Investigator Site 132

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Portland, Maine, United States

Investigator Site 115

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Pittsburgh, Pennsylvania, United States

Investigator Site 120

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Gainesville, Florida, United States

Investigator Site 102

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Jacksonville, Florida, United States

Investigator Site 134

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Jackson, Mississippi, United States

Investigator Site 133

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Edmonton, Alberta, Canada

Investigator Site 121

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Burlington, Vermont, United States

Investigator Site 110

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Atlanta, Georgia, United States

Investigator Site 123

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Long Beach, California, United States

Investigator Site 209

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Rzeszow, Poland

Investigator Site 107

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Los Angeles, California, United States

Investigator Site 127

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Chicago, Illinois, United States

Investigator Site 401

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Madrid, Spain

Investigator Site 103

🇺🇸

Cleveland, Ohio, United States

Investigator Site 501

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Brno, Czechia

Investigator Site 106

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Hershey, Pennsylvania, United States

Investigator Site 113

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Toledo, Ohio, United States

Investigator Site 502

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Plzen, Czechia

Investigator Site 303

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Debrecen, Hajdu-Bihar, Hungary

Investigator Site 206

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Lodz, Poland

Investigator Site 104

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Indianapolis, Indiana, United States

Investigator Site 130

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Miami, Florida, United States

Investigator Site 135

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Las Vegas, Nevada, United States

Investigator Site 116

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Houston, Texas, United States

Investigator Site 111

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Dallas, Texas, United States

Investigator Site 304

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Mosdos, Somogy County, Hungary

Investigator Site 105

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Wichita, Kansas, United States

Investigator Site 109

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Glenview, Illinois, United States

Investigator Site 128

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Lexington, Kentucky, United States

Investigator Site 126

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East Lansing, Michigan, United States

Investigator Site 125

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Fort Worth, Texas, United States

Investigator Site 129

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Morgantown, West Virginia, United States

Investigator Site 301

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Ajka, Veszprem County, Hungary

Investigator Site 305

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Szeged, Csongrad County, Hungary

Investigator Site 302

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Torokbalint, Pest County, Hungary

Investigator Site 601

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Jerusalem, Israel

Investigator Site 203

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Karpacz, Poland

Investigator Site 208

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Bialystok, Poland

Investigator Site 201

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Lublin, Poland

Investigator Site 205

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Lublin, Poland

Investigator Site 202

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Rabka Zdroj, Poland

Investigator Site 204

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Sopot, Poland

Investigator Site 207

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Warszawa, Poland

Investigator Site 403

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Madrid, Spain

Investigator Site 402

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Malaga, Spain

Investigator Site 404

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Valencia, Spain

Investigator Site 122

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Louisville, Kentucky, United States

Investigator Site 124

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Ann Arbor, Michigan, United States

Investigator Site 101

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Oklahoma City, Oklahoma, United States

Investigator Site 114

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Aurora, Colorado, United States

Investigator Site 117

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Orlando, Florida, United States

Investigator Site 136

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Oklahoma City, Oklahoma, United States

Investigator Site 119

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Portland, Oregon, United States

Investigator Site 112

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Richmond, Virginia, United States

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