MedPath

Nortriptyline for the Treatment of Functional Dyspepsia

Phase 3
Conditions
Functional Dyspepsia
Interventions
Drug: Placebo
Registration Number
NCT03652571
Lead Sponsor
Maastricht University Medical Center
Brief Summary

Functional dyspepsia (FD) is a common functional gastrointestinal disorder characterized by upper abdominal discomfort/pain and/or symptoms of meal-related fullness/satiety. There is currently no definitive therapy that is beneficial for all FD patients. Accumulating evidence suggests efficacy of tricyclic antidepressants (TCAs) in FD. However, no firm conclusion can be drawn currently due to the relatively small amount of studies and large heterogeneity between studies. In addition, TCAs are often associated with side effects, which occur early after initiation of therapy preceding the therapeutic effect and often result in discontinuation of the therapy. These side effects are related to drug metabolism, which depend on polymorphisms of the cytochrome P (CYP) enzyme system. It is therefore hypothesized that pre-treatment assessment of CYP genotype and subsequent exclusion of abnormal metabolizers limits the occurrence of side-effects and as such improves compliance and efficacy.

Detailed Description

Not available

Recruitment & Eligibility

Status
UNKNOWN
Sex
All
Target Recruitment
154
Inclusion Criteria
  • Age 18-65 years;
  • A diagnosis of FD according to the Rome IV criteria;
  • Predicted CYP2D6 extensive metabolizer phenotype on the basis of CYP genotyping
  • Insufficient effect of first line treatment with proton pump inhibitors (twice daily) or prokinetics;
  • In the presence of alarm symptoms, patients are required to have undergone an upper gastrointestinal endoscopy (without evidence of organic disease), and have tested negative for Helicobacter pylori 2 years prior to inclusion;
  • Women in their fertile age (<55 years old) must use contraception or be postmenopausal for at least two years.
Exclusion Criteria
  • Predicted CYP2D6 poor, intermediate or ultrarapid metabolizer phenotype on the basis of CYP genotyping

  • Evidence of current anxiety and/or depression disorder as defined by a score ≥ 10 on the GAD-7 and/or PHQ-9 questionnaire;

  • Current use or any previous use of psychotropic medication in the last 3 months prior to inclusion;

  • Inability to discontinue prokinetics, NSAIDs or opioids;

  • Using drugs of abuse;

  • Using more than 2 or 3 units of alcohol per day (females and males respectively)

  • Previous major abdominal surgery or radiotherapy interfering with gastrointestinal function:

    1. Uncomplicated appendectomy, cholecystectomy and hysterectomy allowed unless within the past 6 months;
    2. Other surgery upon judgment of the principle investigator;
  • History of gastric ulcer;

  • History of liver disease, cholangitis, achlorhydria, gallstones or other diseases of the gallbladder/biliary system;

  • History of epilepsy

  • History of glaucoma

  • Pregnancy or lactation.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PlaceboPlaceboPlacebo
NortriptylineNortriptylineNortriptyline in an escalating dose regimen: Week 1-2: 10mg daily Week 3-4: 25mg daily Week 5-12: 50mg daily
Primary Outcome Measures
NameTimeMethod
Symptom response12 weeks

Response to therapy, as defined by a 30% reduction from baseline (i.e. the run-in period) in the weekly average of daily symptom scores, during at least 50% of weeks 3-12 of treatment. Symptoms will be assessed daily using a digital diary (mobile phone application). Recorded symptoms include the five core symptoms of FD: epigastric pain, epigastric burning, postprandial fullness, early satiety and upper abdominal bloating.

Secondary Outcome Measures
NameTimeMethod
Adequate relief12 weeks

Self-reported adequate relief. Adequate relief is defined as a 'yes' response in at least 50% of weeks 3-12 of the treatment. Reported via digital diary (mobile phone application)

General quality of life12 weeks, 3 & 6 months

Assessed with the use of the Euro-Qol-5D (EQ-5D; change from baseline).

Dyspepsia-specific quality of life12 weeks, 3 & 6 months

Dyspepsia-specific quality of life, assessed with the use of the Nepean Dyspepsia Index (NDI; change from baseline).

Cost-utility12 weeks, 3 & 6 months

Cost-utility, as determined by calculations incorporating total treatment costs and changes in EQ-5D-5L (QALYs gained), and results from the Medical Consumption Questionnaire (MCQ) and Productivity Cost Questionnaire (PCQ) \[savings from reduced medical resource use and increased work productivity respectively\].

Use of rescue medication.12 weeks

As reported via digital diary (mobile phone application)

Number and severity of side effects.12 weeks

As reported via digital diary (mobile phone application)

Responder rates following discontinuation6 months

Responder rates following discontinuation of treatment at 6 months follow-up, as defined by a "Yes" to the query regarding adequate relief from baseline symptoms.

Negative mood - anxiety12 weeks, 3 & 6 months

Assessed with the use of the Generalized Anxiety Disorder-7 (GAD-7; change from baseline)

Negative mood - depression12 weeks, 3 & 6 months

Assessed with the use of the Patient Health Questionnaire-9 (PHQ-9; change from baseline)

Trial Locations

Locations (14)

Medisch Spectrum Twente

🇳🇱

Enschede, Netherlands

Tergooi Hilversum

🇳🇱

Hilversum, Netherlands

Alrijne ziekenhuis

🇳🇱

Leiden, Netherlands

AMC

🇳🇱

Amsterdam, Netherlands

VUmc

🇳🇱

Amsterdam, Netherlands

Jeroen Bosch ziekenhuis

🇳🇱

Den Bosch, Netherlands

Rijnstate

🇳🇱

Arnhem, Netherlands

Gelderse Vallei

🇳🇱

Ede, Netherlands

Martini Ziekenhuis

🇳🇱

Groningen, Netherlands

Maastrich University Medical Center

🇳🇱

Maastricht, Netherlands

Medisch Centrum Leeuwarden

🇳🇱

Leeuwarden, Netherlands

Bernhoven

🇳🇱

Uden, Netherlands

Diakonessenhuis

🇳🇱

Utrecht, Netherlands

MMC

🇳🇱

Veldhoven, Netherlands

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