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Long-Acting Cabotegravir Plus VRC-HIVMAB075-00-AB (VRC07-523LS) for Viral Suppression in Adults Living With HIV-1

Phase 2
Completed
Conditions
HIV Infections
Interventions
Drug: Oral Cabotegravir (CAB)
Drug: Nucleoside Reverse Transcriptase Inhibitors (NRTIs)
Drug: Long-Acting Injectable Cabotegravir (CAB LA)
Biological: VRC07-523LS
Drug: Standard of Care (SOC) Oral ART
Registration Number
NCT03739996
Lead Sponsor
National Institute of Allergy and Infectious Diseases (NIAID)
Brief Summary

The purpose of this study is to assess the safety, tolerability, pharmacokinetics, and antiviral activity of long-acting cabotegravir (CAB LA) plus the broadly neutralizing monoclonal antibody,VRC-HIVMAB075-00-AB (VRC07-523LS), in adults living with HIV-1 with suppressed plasma viremia.

Detailed Description

This study will assess the safety, tolerability, pharmacokinetics, and antiviral activity of long-acting cabotegravir (CAB LA) plus the broadly neutralizing monoclonal antibody, VRC-HIVMAB075-00-AB (VRC07-523LS), in adults living with HIV-1 with suppressed plasma viremia.

The study will be conducted in three steps. At Step 1 entry, all participants will discontinue their current antiretroviral therapy (ART) regimen except for nucleoside reverse transcriptase inhibitors (NRTIs), and initiate oral CAB.

During Step 1, participants tolerating oral CAB plus their current two NRTIs, and displaying viral suppression (HIV-1 RNA \<50 copies/mL), will register to Step 2. At entry into Step 2, eligible participants will stop their oral CAB and NRTIs and will receive a VRC07-523LS infusion plus CAB LA injection. After entry in Step 2, participants will receive CAB LA every 4 weeks through Week R2+44 plus VRC07-523LS every 8 weeks through Week R2+40.

At the last visit in Step 2 (Week R2+48), or at premature study treatment discontinuation, all participants who received any CAB LA or VRC07-523LS will enter Step 3 and switch to standard of care (SOC) oral ART for approximately 48 weeks.

Participants will attend a number of study visits throughout the study. Study visits may include a physical examination, clinical assessment, pregnancy testing, and blood and urine collection. Participants will remain in the study for up to 101 weeks, including approximately 5 weeks in Step 1, 48 weeks in Step 2, followed by 48 weeks in Step 3.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
75
Inclusion Criteria

Not provided

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Exclusion Criteria

Not provided

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Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
CAB LA + VRC07-523LSStandard of Care (SOC) Oral ARTStep 1: CAB administered orally as one 30 mg tablet once daily, plus two NRTIs, for 5 weeks. Step 2: CAB LA loading dose (600 mg) administered as one IM injection at Step 2 entry study visit, and maintenance dose (400 mg), starting at 4 weeks after CAB LA loading dose, and then every 4 weeks through Week R2+44. VRC07-523LS (40 mg/kg) administered as an IV infusion starting at Step 2 entry and then every 8 weeks through Week R2+40. Step 3: SOC oral ART regimen for approximately 48 weeks.
CAB LA + VRC07-523LSOral Cabotegravir (CAB)Step 1: CAB administered orally as one 30 mg tablet once daily, plus two NRTIs, for 5 weeks. Step 2: CAB LA loading dose (600 mg) administered as one IM injection at Step 2 entry study visit, and maintenance dose (400 mg), starting at 4 weeks after CAB LA loading dose, and then every 4 weeks through Week R2+44. VRC07-523LS (40 mg/kg) administered as an IV infusion starting at Step 2 entry and then every 8 weeks through Week R2+40. Step 3: SOC oral ART regimen for approximately 48 weeks.
CAB LA + VRC07-523LSNucleoside Reverse Transcriptase Inhibitors (NRTIs)Step 1: CAB administered orally as one 30 mg tablet once daily, plus two NRTIs, for 5 weeks. Step 2: CAB LA loading dose (600 mg) administered as one IM injection at Step 2 entry study visit, and maintenance dose (400 mg), starting at 4 weeks after CAB LA loading dose, and then every 4 weeks through Week R2+44. VRC07-523LS (40 mg/kg) administered as an IV infusion starting at Step 2 entry and then every 8 weeks through Week R2+40. Step 3: SOC oral ART regimen for approximately 48 weeks.
CAB LA + VRC07-523LSVRC07-523LSStep 1: CAB administered orally as one 30 mg tablet once daily, plus two NRTIs, for 5 weeks. Step 2: CAB LA loading dose (600 mg) administered as one IM injection at Step 2 entry study visit, and maintenance dose (400 mg), starting at 4 weeks after CAB LA loading dose, and then every 4 weeks through Week R2+44. VRC07-523LS (40 mg/kg) administered as an IV infusion starting at Step 2 entry and then every 8 weeks through Week R2+40. Step 3: SOC oral ART regimen for approximately 48 weeks.
CAB LA + VRC07-523LSLong-Acting Injectable Cabotegravir (CAB LA)Step 1: CAB administered orally as one 30 mg tablet once daily, plus two NRTIs, for 5 weeks. Step 2: CAB LA loading dose (600 mg) administered as one IM injection at Step 2 entry study visit, and maintenance dose (400 mg), starting at 4 weeks after CAB LA loading dose, and then every 4 weeks through Week R2+44. VRC07-523LS (40 mg/kg) administered as an IV infusion starting at Step 2 entry and then every 8 weeks through Week R2+40. Step 3: SOC oral ART regimen for approximately 48 weeks.
Primary Outcome Measures
NameTimeMethod
Frequency of either 1) the occurrence of a Grade 3 or higher adverse event (AE); or 2) premature study treatment discontinuation due to an AE (regardless of grade)Measured through Week R3+48 of Step 3

Both of which are possibly, probably, or definitely related (as judged by the core team) to the CAB LA plus VRC07-523LS combination.

Number of participants who experience virologic failureMeasured through Week R2+44 of Step 2

Defined as confirmed HIV-1 RNA greater than or equal to 200 copies/mL

Secondary Outcome Measures
NameTimeMethod
Frequency of viral resistance of breakthrough isolatesMeasured through Week R2+44 of Step 2

Based on laboratory evaluations

Trough levels of the concentration of CAB LAMeasured through Week R2+48 of Step 2

Based on PK sampling

Number of participants who experience virologic failureMeasured through Week R2+44 of Step 2

Defined by the U.S. Food and Drug Administration (FDA) snapshot algorithm

Frequency of either 1) virologic failure (confirmed HIV-1 RNA greater than or equal to 200 copies/mL); or 2) premature discontinuation of the CAB LA plus VRC07-523LS combinationMeasured through Week R2+44 of Step 2

Based on laboratory evaluations

Number of participants with confirmed HIV-1 RNA greater than or equal to 50 copies/mLMeasured through Week R2+24 of Step 2

Based on laboratory evaluations

Number of participants with either 1) confirmed HIV-1 RNA greater than or equal to 50 copies/mL; or 2) premature discontinuation of the CAB LA plus VRC07-523LS combinationMeasured through Week R2+44 of Step 2

Based on laboratory evaluations

Frequency of anti-idiotype antibodies against VRC07-523LS in samples collected from representative time points throughout the studyMeasured through Week R2+48 of Step 2

Based on laboratory evaluations

Frequency of either 1) the occurrence of a Grade 3 or higher AE; or 2) premature oral CAB discontinuation due to an AE (regardless of grade)Measured through Week 5 of Step 1

Both of which are possibly, probably, or definitely related (as judged by the core team) to oral CAB.

Number of participants who prematurely discontinue oral CAB or the CAB LA plus VRC07-523LS combinationMeasured through Week R2+44 of Step 2

Based on self report

Frequency of the occurrence of a Grade 3 or higher AE that is possibly, probably, or definitely related (as judged by the core team) to oral CAB or the CAB LA plus VRC07-523LS combinationMeasured through Week R3+48 of Step 3

Frequency of the occurrence of a Grade 3 or higher AE that is possibly, probably, or definitely related (as judged by the core team) to oral CAB or the CAB LA plus VRC07-523LS combination

Trough levels of the concentration of VRC07-523LSMeasured through Week R2+48 of Step 2

Based on PK sampling

Trial Locations

Locations (19)

Johns Hopkins University CRS

🇺🇸

Baltimore, Maryland, United States

Puerto Rico AIDS Clinical Trials Unit CRS

🇵🇷

San Juan, Puerto Rico

UCSD Antiviral Research Center CRS

🇺🇸

San Diego, California, United States

University of Washington AIDS CRS

🇺🇸

Seattle, Washington, United States

University of Colorado Hospital CRS

🇺🇸

Aurora, Colorado, United States

Weill Cornell Chelsea CRS

🇺🇸

New York, New York, United States

Penn Therapeutics, CRS

🇺🇸

Philadelphia, Pennsylvania, United States

Ohio State University CRS

🇺🇸

Columbus, Ohio, United States

Chapel Hill CRS

🇺🇸

Chapel Hill, North Carolina, United States

Cincinnati Clinical Research Site

🇺🇸

Cincinnati, Ohio, United States

Alabama CRS

🇺🇸

Birmingham, Alabama, United States

Washington University Therapeutics (WT) CRS

🇺🇸

Saint Louis, Missouri, United States

Northwestern University CRS

🇺🇸

Chicago, Illinois, United States

Ucsf Hiv/Aids Crs

🇺🇸

San Francisco, California, United States

Rush University CRS

🇺🇸

Chicago, Illinois, United States

Columbia P&S CRS

🇺🇸

New York, New York, United States

New Jersey Medical School Clinical Research Center CRS

🇺🇸

Newark, New Jersey, United States

Weill Cornell Uptown CRS

🇺🇸

New York, New York, United States

University of Rochester Adult HIV Therapeutic Strategies Network CRS

🇺🇸

Rochester, New York, United States

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