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Phase 1 Study of Ibrutinib and Immuno-Chemotherapy Using Temozolomide, Etoposide, Doxil, Dexamethasone, Ibrutinib,Rituximab (TEDDI-R) in Primary CNS Lymphoma

Registration Number
NCT02203526
Lead Sponsor
National Cancer Institute (NCI)
Brief Summary

BACKGROUND:

* Primary CNS lymphoma (PCNSL) is a rare subtype of diffuse large B-cell lymphoma.

* The outcome for patients with this diagnosis is significantly worse than for that of systemic DLBCL. Most treatment approaches in the past have included high dose methotrexate and radiation treatment.

* Most PCNSLs appear to be of activated B-cell (ABC) origin.

* Ibrutinib is an inhibitor of Bruton s tyrosine kinase (BTK) and effective for systemic DLBCL of ABC origin.

* We propose doing a study in which ibrutinib is combined with a novel chemotherapy platform called dose adjusted temozolomide, etoposide, doxil, dexamethasone, ibrutinib, rituximab (TEDDI-R).

OBJECTIVE:

- Identify the maximum tolerated dose (MTD) of ibrutinib or the dose that achieves adequate CSF concentrations, whichever comes first, when ibrutinib is given with TEDDI-R.

ELIGIBILITY:

* Relapsed/refractory PCNSL.

* Age greater than or equal to 18 years.

* No pregnant or breast-feeding women.

* Adequate organ function (defined in protocol).

STUDY DESIGN:

* This is a phase 1 study of 40 patients.

* The study will have two components.

1. Phase 1: MTD of ibrutinib will be identified or the dose at which ibrutinib achieves a concentration of less than or equal to 100 nM in the CSF, when given in combination with TEDDI-R immuno-chemotherapy, whichever comes first.

2. Expansion cohort: Safety and tolerability of the regimen in relapsed/refractory or previously untreated PCNSL (DLBCL type) will be assessed at the final ibrutinib dose with TEDDI-R in 10 patients. Secondary objectives will be PFS and OS.

Detailed Description

Background:

* Primary CNS lymphoma (PCNSL) is a rare subtype of diffuse large B-cell lymphoma

* The outcome for patients with this diagnosis is significantly worse than for that of systemic DLBCL.

Most treatment approaches in the past have included high dose methotrexate and radiation treatment.

* Most PCNSLs appear to be of activated B-cell (ABC) origin

* Ibrutinib is an inhibitor of Bruton s tyrosine kinase (BTK) and effective for systemic DLBCL of ABC origin.

* We propose doing a study in which ibrutinib is combined with a novel chemotherapy platform called temozolomide, etoposide, doxil, dexamethasone, ibrutinib, rituximab (TEDDI-R).

Objective:

* To identify the dose of ibrutinib with anti-fungal prophylaxis that can be safely administered to achieve an ibrutinib median CSF CMAX of 1.98 nM (Range 0.69 to 11.1)

* Revised in Amendment M (version date: 11/03/2020): To assess the safety, feasibility, and complete response (CR) rate of the TEDDI-R in untreated PCNSL (DLBCL type) patients.

Eligibility:

* Relapsed/refractory or untreated PCNSL

* Age \>= 18 years.

* No pregnant or breast-feeding women.

* Adequate organ function (defined in protocol).

Study Design:

* This is a phase 1 study of 93 patients.

* The study will have three components.

* Phase 1: MTD of ibrutinib will be identified or the dose at which ibrutinib achieves a concentration of \>= 100 nM in the CSF, when given in combination with TEDDI-R immuno-chemotherapy, whichever comes first.

* Expansion cohort: Safety and tolerability of the regimen in relapsed/refractory PCNSL (DLBCL type) will be assessed at the final ibrutinib dose with TEDDI-R in 10 patients. Secondary objectives will be PFS and OS.

* Revised Study Design: Effective with Amendment G (version date: 7/31/2017), new ibrutinib dose levels are being added together with anti-fungal prophylaxis to determine the dose of ibrutinib that may be safely given with the chemotherapy platform.

* Effective with Amendment M (version date: 11/03/2020), a second expansion cohort of untreated PCNSL (DLBCL type) will be added: Safety, feasibility, and complete response rate of the regimen in untreated PCNSL (DLBCL type) will be assessed at the final ibrutinib dose with TEDDI-R in 15 patients. Secondary objectives will be PFS and OS.

* Effective with Amendment 06/04/2021, a new dosing schedule will be tested in up to 10 relapsed or refractory patients and 15 patients with untreated PCNSL. Secondary objectives will be PFS and OS.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
93
Inclusion Criteria

Not provided

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Exclusion Criteria

Not provided

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Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Arm 1-A (original study design - prior to Amendment G)Ibrutinib (Arm 4)TEDD-R (cycle 1) with ibrutinib; TEDDI-R with cytarabine (cycles 2-6)
Arm 1-A (original study design - prior to Amendment G)Ibrutinib (Arms 2, 3 and 4)TEDD-R (cycle 1) with ibrutinib; TEDDI-R with cytarabine (cycles 2-6)
Arm 1-A (original study design - prior to Amendment G)Ibrutinib (Arm 1 - Closed with Amendment G)TEDD-R (cycle 1) with ibrutinib; TEDDI-R with cytarabine (cycles 2-6)
Arm 4 (Dose Expansion; Amendment 06/04/21)MethotrexateTEDDI-R, cytarabine or methotrexate, isavuconazole, ibrutinib for 10 days
Arm 1-A (original study design - prior to Amendment G)CytarabineTEDD-R (cycle 1) with ibrutinib; TEDDI-R with cytarabine (cycles 2-6)
Arm 1-A (original study design - prior to Amendment G)TEDDTEDD-R (cycle 1) with ibrutinib; TEDDI-R with cytarabine (cycles 2-6)
Arm 4 (Dose Expansion; Amendment 06/04/21)TEDDITEDDI-R, cytarabine or methotrexate, isavuconazole, ibrutinib for 10 days
Arm 1-A (original study design - prior to Amendment G)TEDDITEDD-R (cycle 1) with ibrutinib; TEDDI-R with cytarabine (cycles 2-6)
Arm 1-B (original study design-prior to Amendment G)TEDDITEDDI-R with cytarabine
Arm 3 (Dose Expansion; prior to Amendment 06/04/2021)TEDDITEDDI-R with cytarabine and isavuconazole
Arm 4 (Dose Expansion; Amendment 06/04/21)Ibrutinib (Arm 4)TEDDI-R, cytarabine or methotrexate, isavuconazole, ibrutinib for 10 days
Arm 2 (Dose Escalation; prior to Amendment 06/04/2021)TEDDITEDDI-R with cytarabine, and isavuconazole
Arm 1-A (original study design - prior to Amendment G)RituximabTEDD-R (cycle 1) with ibrutinib; TEDDI-R with cytarabine (cycles 2-6)
Arm 1-B (original study design-prior to Amendment G)RituximabTEDDI-R with cytarabine
Arm 2 (Dose Escalation; prior to Amendment 06/04/2021)IsavuconazoleTEDDI-R with cytarabine, and isavuconazole
Arm 1-B (original study design-prior to Amendment G)CytarabineTEDDI-R with cytarabine
Arm 2 (Dose Escalation; prior to Amendment 06/04/2021)RituximabTEDDI-R with cytarabine, and isavuconazole
Arm 2 (Dose Escalation; prior to Amendment 06/04/2021)CytarabineTEDDI-R with cytarabine, and isavuconazole
Arm 4 (Dose Expansion; Amendment 06/04/21)CytarabineTEDDI-R, cytarabine or methotrexate, isavuconazole, ibrutinib for 10 days
Arm 3 (Dose Expansion; prior to Amendment 06/04/2021)IsavuconazoleTEDDI-R with cytarabine and isavuconazole
Arm 3 (Dose Expansion; prior to Amendment 06/04/2021)RituximabTEDDI-R with cytarabine and isavuconazole
Arm 3 (Dose Expansion; prior to Amendment 06/04/2021)CytarabineTEDDI-R with cytarabine and isavuconazole
Arm 4 (Dose Expansion; Amendment 06/04/21)IsavuconazoleTEDDI-R, cytarabine or methotrexate, isavuconazole, ibrutinib for 10 days
Arm 4 (Dose Expansion; Amendment 06/04/21)RituximabTEDDI-R, cytarabine or methotrexate, isavuconazole, ibrutinib for 10 days
Primary Outcome Measures
NameTimeMethod
safety and feasibility in untreated PCNSL patientsInitiation of ibrutinib until 30 days after treatment

Incidence of adverse events (i.e., grade and frequency)

MTD of ibrutinib with anti-fungal prophylaxis when given with TEDD-Rafter one cycle

AEs will be tabulated and reported

MTD of ibrutinib when given with TEDD-Rafter one cycle

AEs will be tabulated and reported

Complete Response rate in untreated PCNSL patientsevery 3 months for 1 year, every 4 months year 2, every 6 months year 3 then yearly

The response rate will be determined and reported along with a 95% confidence interval

Secondary Outcome Measures
NameTimeMethod
Safety and TolerabilityInitiation of ibrutinib until 30 days after treatment

Incidence of adverse events (i.e., grade and frequency)

Progression-free survivalevery 3 months for 1 year, every 4 months year 2, every 6 months year 3 then yearly

The response rate will be determined and reported along with a 95% confidence interval

Overall survivalevery 3 months for 1 year, every 4 months year 2, every 6 months year 3 then yearly

The response rate will be determined and reported along with a 95% confidence interval

Trial Locations

Locations (1)

National Institutes of Health Clinical Center

🇺🇸

Bethesda, Maryland, United States

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