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Pharmacokinetics of Anacetrapib (MK0859) in Subjects With Impaired Renal Function (MK-0859-038)

Phase 1
Completed
Conditions
Dyslipidemia
Interventions
Registration Number
NCT01122667
Lead Sponsor
Merck Sharp & Dohme LLC
Brief Summary

This study will evaluate the Area Under the Curve (AUC(0 to infinity)) of anacetrapib in subjects with impaired renal function and healthy matched control subjects.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
24
Inclusion Criteria
  • Female subjects of reproductive potential test negative for pregnancy and agree to use two acceptable methods of birth control throughout the study
  • Subject is in good health
  • If Subject is a smoker, smoking is limited to no more than 10 cigarettes per day
Exclusion Criteria
  • Subject has a history of stroke, chronic seizures or major neurological disorder
  • Subject has a history of cancer
  • Subject is unable to refrain from or anticipates the use of any prescription or non-prescription medication during the study
  • Subject consumes excessive amounts of alcohol or caffeine
  • Subject has had major surgery, donated blood or participated in another investigational study within the past 4 weeks
  • Subject is a nursing mother
  • Subject has had a kidney removed or has a functioning renal transplant

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Part 1 - Panel AanacetrapibSubjects with severe renal impairment
Part 2 - Panel CanacetrapibSubjects with moderate renal impairment
Part 2 - Panel DanacetrapibHealthy matched control subjects
Part 2 - Panel EanacetrapibSubjects with mild renal impairment
Part 2 - Panel FanacetrapibHealthy matched control subjects
Part 1 - Panel BanacetrapibHealthy matched control subjects
Primary Outcome Measures
NameTimeMethod
Area Under the Curve (AUC(0 to infinity)) of anacetrapibthrough 168 hours post dose
Secondary Outcome Measures
NameTimeMethod
Safety and tolerability of a single dose administration of 100mg anacetrapib, measured by the number of clinical and laboratory adverse eventsthrough 14 days post dose
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