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Adagrasib in Patients With KRASG12C-mutant NSCLC Who Are Elderly or Have Poor Performance Status

Phase 2
Recruiting
Conditions
NSCLC Stage IV
KRAS P.G12C
Interventions
Registration Number
NCT05673187
Lead Sponsor
ETOP IBCSG Partners Foundation
Brief Summary

ADEPPT is an international, multicentre, single-arm phase II trial. The protocol treatment consists of adagrasib, which is administered at a dose of 600 mg orally, twice daily until progression or unacceptable toxicity.The primary objective of this trial is to assess the clinical efficacy of adagrasib treatment, in terms of objective response, in patients with KRASG12C-mutant NSCLC, including the elderly (≥70 years) or patients with poor performance status (ECOG PS=2).

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
68
Inclusion Criteria
  1. Histologically or cytologically confirmed stage IV NSCLC.
  2. KRASG12C-mutation by local testing (by tissue or ctDNA).
  3. Prior treatment with at least one line of systemic therapy for NSCLC (e.g., platinum-based doublet chemotherapy and/or immune-checkpoint inhibition or both).
  4. Life expectancy ≥12 weeks.
  5. Measurable disease according to RECIST v1.1.
  6. Age ≥18 years with ECOG PS 2 (cohort 1), or age ≥70 years with ECOG PS 0-1 (cohort 2).
  7. Adequate haematological, renal and liver function
  8. Men and women of childbearing potential must agree to use use highly effective contraceptive methods.
  9. Women of childbearing potential, including women who had their last menstruation in the last 2 years, must have a negative urinary or serum beta HCG pregnancy test within 5 weeks before enrolment. Pregnancy test must be repeated within 7 days before the first dose of adagrasib treatment.Ability to comply with the trial protocol, in the investigator's judgment.
  10. Written IC for study participation must be signed and dated by the patient and the investigator prior to any study-related intervention, including the submission of mandatory biomaterial.
Exclusion Criteria
  1. Prior investigational therapy within 28 days or at least 5 half-lives before enrolment.

  2. Prior treatment with an agent targeting KRASG12C.

  3. Leptomeningeal disease or untreated brain metastases.

    • Patient should be neurologically stable for at least 2 weeks before enrolment, without the need for corticosteroids, except for prednisone (or its equivalent) at a dose of ≤10 mg daily.
    • For patients with definitively treated brain metastases, a time period of minimum of 2 weeks must have elapsed from the last day of radiotherapy.
  4. History of intestinal disease or major gastric surgery likely to alter absorption of study treatment or inability to swallow oral medications.

  5. Any of the following cardiac abnormalities:

    • Unstable angina pectoris or myocardial infarction within 6 months prior to enrolment.
    • Symptomatic or uncontrolled atrial fibrillation within 6 months prior to enrolment.
    • Congestive heart failure ≥NYHA Class 3 within 6 months prior to enrolment.
    • Prolonged QTc interval >480 ms or family or medical history of congenital Long QT Syndrome.
  6. History of stroke or transient ischemic attack within 6 months prior to enrolment.

  7. Ongoing need for treatment with concomitant medication with any of the following characteristics: known risk of Torsades de Pointes; substrate of CYP3A with narrow therapeutic index; strong inducer of CYP3A and/or P-gp; strong inhibitor of BCRP; and proton pump inhibitors that cannot be switched to alternative treatment prior to enrolment.

  8. Known human immunodeficiency virus (HIV) infection.

  9. Acute or chronic hepatitis B or C infection.

  10. Women who are pregnant or in the period of lactation.

  11. Sexually active men and women of childbearing potential who are not willing to use an effective contraceptive method during the study.

  12. Judgement by the investigator that the patient should not participate in the study if the patient is unlikely to comply with study procedures, restrictions and requirements.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Treatment ArmAdagrasibAdagrasib to be administered at a dose of 600 mg orally, twice daily until progression or unacceptable toxicity.
Primary Outcome Measures
NameTimeMethod
Objective Response Rate (ORR) per RECIST v1.1, assessed at 12 weeks.From date of enrolment until 12 weeks post-enrolment

The primary objective of this trial is to assess the clinical efficacy of adagrasib treatment, in terms of objective response as defined as the rate of patients achieving a best overall response \[complete response (CR) or partial response (PR)\] according to RECIST v1.1

Secondary Outcome Measures
NameTimeMethod
Durable clinical benefitFrom date of enrolment until at least the 24-week assessment.

Durable clinical benefit (DCB) is defined as the rate among all enrolled patients who are alive and without disease progression who achieve CR or PR, according to RECIST v1.1, or stable disease (SD) lasting for at least 24 weeks.

Time-to-progression (TTP)From the date of enrolment until last tumour assessment (approximately 20-26 months after enrolment of the first patient)

Time-to-progression (TTP) is defined as the time from the date of enrolment until the date of documented progression (according to RECIST v1.1). Censoring for patients without documented progression will occur at the date of last tumour assessment without PD. Patients without a post-baseline tumour assessment will be censored at the date of enrolment plus 1 day.

Progression-free survival (PFS)From the date of enrolment until last tumour assessment (approximately 20-26 months after enrolment of the first patient)

Progression-free survival (PFS) is defined as the time from the date of enrolment until the date of documented progression (according to RECIST v1.1) or death, if progression is not documented. Censoring (for patients without progression or death) will occur at the date of last tumour assessment. Patients without a post-baseline tumour assessment will be censored at the date of enrolment plus 1 day.

Overall survival (OS)From the date of enrolment until last patient last visit (approximately 20-26 months after enrolment of the first patient)

Overall survival (OS) is defined as the time from the date of enrolment until the date of death from any cause. Censoring for patients who are not reported as dead will occur at the last date they are known to be alive. Data for patients who do not have post-baseline information will be censored at the date of enrolment plus 1 day.

Safety and tolerabilityFrom the date of enrolment until last patient last visit (approximately 20-26 months after enrolment of the first patient)

The toxicity and safety profile of the protocol treatment will be evaluated by:

* Adverse events (AEs) according to CTCAE v5.0 (any-cause, as well as treatment-related) including AEs leading to dose delays and/or interruptions, withdrawal of protocol treatment, and death

* Severe and serious AEs

* Deaths

Laboratory parameters and abnormalities 1From the date of enrolment until last patient last visit (approximately 20-26 months after enrolment of the first patient)

Hemoglobin \[g/dl\]

Laboratory parameters and abnormalities 2From the date of enrolment until last patient last visit (approximately 20-26 months after enrolment of the first patient)

Platelet count \[G/L\]

Laboratory parameters and abnormalities 3From the date of enrolment until last patient last visit (approximately 20-26 months after enrolment of the first patient)

White blood cell count \[G/L\]

Vital signs 1From the date of enrolment until last patient last visit (approximately 20-26 months after enrolment of the first patient)

Blood pressure systolic \[mmHg\]

Vital signs 2From the date of enrolment until last patient last visit (approximately 20-26 months after enrolment of the first patient)

Blood pressure diastolic \[mmHG\]

Vital signs 3From the date of enrolment until last patient last visit (approximately 20-26 months after enrolment of the first patient)

Heart rate \[beats/min\]

Vital signs 4From the date of enrolment until last patient last visit (approximately 20-26 months after enrolment of the first patient)

Body temperature \[°C\]

Patient-reported outcomes NFLSI-17From the date of screening until patient's end of treatment (approximately 20-26 months after enrolment of the first patient)

Patient-reported symptoms and functioning will be assessed by NCCN-Functional Assessment of Cancer Therapy (FACT) Lung Symptom Index-17 (NFLSI-17).

Patient-reported outcomes PRO-CTCAE®From the date of screening until patient's end of treatment (approximately 20-26 months after enrolment of the first patient)

The most commonly reported treatment-related adverse effects of adagrasib (diarrhoea and vomiting) that are not covered by the NFLSI-17 will be assessed by the NCI Patient-Reported Outcomes version of the Common Terminology Criteria for Adverse Events (PRO-CTCAE®).

Trial Locations

Locations (22)

St James's Hospital

🇮🇪

Dublin, Ireland

University Hospital Limerick

🇮🇪

Limerick, Ireland

Instiute Jules Bordet

🇧🇪

Brussels, Belgium

AULSS2 Marca Trevigiana Treviso

🇮🇹

Treviso, Italy

Le Mans - CHG

🇫🇷

Le Mans, France

Beaumont Hospital

🇮🇪

Dublin, Ireland

Caen - CHU

🇫🇷

Caen, France

Centre Hospitalier d'Avignon

🇫🇷

Avignon, France

Hôpital de Marseille

🇫🇷

Marseille, France

University Hospital Waterford

🇮🇪

Waterford, Ireland

Santa Maria della Misericordia Hospital

🇮🇹

Perugia, Italy

Fondazione IRCCS Policlinico S. Matteo

🇮🇹

Pavia, Italy

Istituto Nazionale Tumori "Regina Elena"

🇮🇹

Rome, Italy

Complejo Hospitalario Universitario a Coruña

🇪🇸

A Coruña, Spain

Alicante University Hospital

🇪🇸

Alicante, Spain

ICO Badalona - Hospital Germans Trias i Pujol

🇪🇸

Badalona, Spain

Hospital Universitario Fundacion Jimenez Diaz

🇪🇸

Madrid, Spain

ICO Bellvitge -H. Duran i Reynals / H. Bellvitge

🇪🇸

L'Hospitalet De Llobregat, Spain

Hospital de Basurto

🇪🇸

Bilbao, Spain

Hospital General Universitario de Valencia (University Hospital Valencia)

🇪🇸

Valencia, Spain

Hospital Universitario Puerta de Hierro

🇪🇸

Madrid, Spain

Christie NHS Manchester

🇬🇧

Manchester, United Kingdom

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