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Delta-THC in Behavioral Disturbances in Dementia

Phase 2
Completed
Conditions
Dementia
Interventions
Drug: Delta-THC
Drug: placebo
Registration Number
NCT01302340
Lead Sponsor
Radboud University Medical Center
Brief Summary

Dementia is a common chronic condition, with predicted increasing prevalence. Nearly all patients with dementia will experience neuropsychiatric symptoms (NPS). This causes significant burden for the individual patients and their caregivers. Current treatment has only modest efficacy and important side-effects. Formulations with Δ9-tetrahydrocannabinol (THC), the psycho-active compound of cannabis, are currently being registered for spasms in multiple sclerosis and other diseases, and may have beneficial effects on NPS.

Detailed Description

Design Phase II pilot study, multi-center, repeated cross-over, double blinded randomized trial. The study consists of two weeks baseline measurements to assure that the neuropsychiatric symptoms are stable and six successive treatment blocks of 2 weeks. Each treatment block lasts for two weeks and contains two double-blinded drug periods, each lasting three days of oral THC or placebo, separated by four day washout periods. After three treatment blocks (period A), the dosage of active treatment was increased for the latter three treatment blocks (period B). After the two treatment periods, subjects will proceed to the extension phase if applicable.

Study centers The department of Geriatrics from Radboud University Nijmegen Medical Centre and the department of Elderly from Vincent van Gogh voor Geestelijke Gezondheidszorg Venray (VVG) will participate in this multi center study.

Participants 20 subjects with dementia and NPS. Intervention Namisol® in doses of twice daily 0,75 mg tablet (period A) and twice daily 1.5 mg (period B) THC oral tablets. Placebo of twice daily 0,75 mg and twice daily 1.5 mg oral tablets Outcome measures Primary outcome is NPI score, secondary CMAI, Zarit Burden scale. Other outcomes include vital signs, side-effects, physical exam, mobility and pharmacogenetics.

Visits This study will be assessed fully ambulatory, starting with a 5 hour clinical visit on day 1 and 8 of block 1 and a phone call on day 2 and 9 for assessment of Adverse Events. Furthermore, the research physician will conduct a weekly home visit weekly during the crossover phase for assessment of , among others, the primary outcome measure. These visits will all be repeated in period B of the crossover phase.

During the 6 month open label extension phase, subjects will visit the clinic three times.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
22
Inclusion Criteria
  • Diagnosis of Alzheimer's Disease (AD), Vascular Dementia (VD) or mixed, according to the criteria of NINCDS-ADRDA or NINCDS-AIREN
  • Clinical Dementia Rating score between 0.5 and 3
  • NPS symptoms, with at least agitation or aggression
Exclusion Criteria
  • Diagnosis of Lewy Body Dementia (LBD) or Fronto-Temporal Dementia (FTD)
  • Major psychiatric disorder
  • Severe concomitant illness, seizure, arrhythmias (except sinus arrhythmia and atrial fibrillation), heart failure New York Heart Association (NYHA) class III or IV
  • Tri Cyclic Antidepressives (TCA) or opioids used within 30 days before randomization till the end of the study
  • Changes in dosage of antidepressives within 6 weeks before randomization and during study, and changes in dosage antipsychotics or benzodiazepines within 2 weeks prior to randomization and during study

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Delta-THCDelta-THCTHC will be administered twice daily during three consecutive days per treatment block(0.75 or 1.5 mg twice daily)
placeboplaceboPlacebo will be administered twice daily during three consecutive days per treatment block.
Primary Outcome Measures
NameTimeMethod
Neuropsychiatric Inventory (NPI)At day 3 and 10 during treatment blocks and after 1 month, 3 months and 6 months in the open label extension phase

Improvement in behavior compared to placebo is measured with the NPI, which is the standard measure of Neuro Psychiatric Symptoms in most clinical trials.

Secondary Outcome Measures
NameTimeMethod
Gait rite®At days 1 and 8 during blocks 1 and 4 and at 1, 3 and 6 months during extension phase

Improvement and/or safety compared to placebo and during long term treatment on balance and mobility. It is a non invasive and highly feasible mobility assessment.

Cohen-Mansfield Agitation Inventory (CMAI)At days 1, 3, 8, and 10 during treatment blocks 1 and 4 and weekly during treatment blocks 2, 3, 5 and 6 and months 1, 3, 6 and 6 during extension phase

Improvement in agitation compared to placebo and during long term treatment is measured with CMAI. It is useful in determining fluctuations in behaviors and emotional states in Alzheimer's Disease

Zarit Burden Scale (ZBS)At days 3 and 10 during treatment blocks and months 1, 3 and 6 during extension phase

Reducing caregiver stress compared to placebo and during long term treatment by focusing on the patients' behavior compared to Zarit burden interviews with the caregiver.

Visual Analogue Scale (VAS) Bowdle for feeling highAt days 1, 3, 8, and 10 during treatment blocks 1 and 4 and weekly during treatment blocks 2, 3, 5 and 6 and months 1, 3, 6 and 6 during extension phase

severity and duration of feeling high episodes

Sway Star®At days 1 and 8 during blocks 1 and 4 and at 1, 3 and 6 months during extension phase

Improvement and/or safety compared to placebo and during long term treatment on balance and mobility. It is a non invasive and highly feasible mobility assessments.

Time up and goAt days 1, 3, 8, and 10 during treatment blocks 1 and 4 and weekly during treatment blocks 2, 3, 5 and 6 and months 1, 3, 6 and 6 during extension phase

Improvement and/or safety compared to placebo and during long term treatment on balance and mobility in elderly patients.

Tinetti Balance Assessment ToolAt days 1, 3, 8, and 10 during treatment blocks 1 and 4 and weekly during treatment blocks 2, 3, 5 and 6 and months 1, 3, 6 and 6 during extension phase

Improvement and/or safety compared to placebo and during long term treatment on balance and mobility in elderly patients. It is a performance-oriented assessment of mobility problems in elderly patients.

pharmacogeneticsday 1

The following polymorphisms will be genotyped:

* CYP2C9\*2

* CYP2C9\*3

* CYP2C19\*2

* CYP2C19\*3

* CYP2C19\*17

To investigate the role of CYP2C9 and CYP2C19 genetic polymorphisms in the interindividual variation in pharmacokinetics, efficacy and adverse events of THC.

Trial Locations

Locations (2)

Radboud university medical center

🇳🇱

Nijmegen, Gelderland, Netherlands

Vincent van Gogh Institute for Psychiatry, department of Elderly

🇳🇱

Venray, Limburg, Netherlands

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