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A Randomized Study of XEN1101 Versus Placebo in Focal-Onset Seizures

Phase 3
Recruiting
Conditions
Focal Onset Seizures
Interventions
Drug: Placebo
Registration Number
NCT05614063
Lead Sponsor
Xenon Pharmaceuticals Inc.
Brief Summary

The X-TOLE2 Phase 3 clinical trial is a randomized, double-blind, placebo-controlled study that will evaluate the clinical efficacy, safety and tolerability of XEN1101 administered as adjunctive therapy in focal-onset seizures.

Detailed Description

Approximately 360 subjects will be randomized in a blinded manner to one of two active treatment groups or placebo in a 1:1:1 fashion (XEN1101 25 mg : 15 mg : Placebo). Eligible subjects will have up to 9.5 weeks of baseline to assess frequency of seizures, followed by 12 weeks of blinded treatment. In order to be included in the study, subjects must be treated with a stable dose of 1 to 3 allowable antiseizure medications (ASMs) for at least one month prior to screening, during baseline, and throughout the double-blind treatment period (DBP) of the study. During the DBP, subjects will be instructed to orally take XEN1101 or placebo once daily with an evening meal.

Subjects who complete the 12-week DBP will have the opportunity to qualify and enroll in a separate open-label extension (OLE) study for continued treatment with XEN1101. Subjects who do not enroll in the OLE will enter a 8-week post treatment follow-up period.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
360
Inclusion Criteria
  • Be properly informed of the nature and risks of the study and give informed consent in writing, prior to entering the study
  • Diagnosis (≥2 years) of focal epilepsy according to the International League Against Epilepsy (ILAE) Classification of Epilepsy (2017). Subject must have had adequate trials of at least 2 ASMs, which were given (and tolerated) at adequate therapeutic doses, without achieving sustained seizure freedom.
  • Treatment with a stable dose of 1 to 3 allowable current ASMs for at least one month prior to screening, during baseline, and throughout the duration of the DBP
  • Able to keep accurate seizure diaries
Exclusion Criteria
  • Previously documented electroencephalogram which shows any pattern not consistent with focal etiology of seizures.
  • History of focal aware non-motor seizures only, non-epileptic psychogenic seizure, primary generalized seizure, developmental and epileptic encephalopathy, including Lennox-Gastaut syndrome.
  • Seizures secondary to drug or alcohol use, ongoing infection, neoplasia, demyelinating disease, degenerative neurological disease, metabolic illness, progressive structural lesion, encephalopathy, or progressive central nervous system (CNS) disease.
  • History of status epilepticus or repetitive seizures within the 12-month period preceding Visit 1 where the individual seizures cannot be counted.
  • History of neurosurgery for seizures <1 year prior to Visit 1, or radiosurgery <2 years prior to enrollment.
  • Any medical condition or personal circumstance that, in the opinion of the investigator, exposes the subject to unacceptable risk by participating in the study or prevents adherence to the protocol.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
XEN1101 25 mg/dayXEN1101XEN1101 25 mg/day
XEN1101 15 mg/dayXEN1101XEN1101 15 mg/day
PlaceboPlaceboPlacebo
Primary Outcome Measures
NameTimeMethod
Median percent change (MPC) in monthly (28 days) focal seizure frequency from baseline to DBP for XEN1101 versus placebo.From baseline through to the double blind period (week 12)
Secondary Outcome Measures
NameTimeMethod
Proportion of subjects experiencing ≥50% reduction in monthly (28 days) focal seizure frequency from baseline through the DBP for XEN1101 versus placebo.From baseline through to the double blind period (week 12)
MPC in weekly (7 days) focal seizure frequency from baseline to Week 1 for XEN1101 versus placebo.From baseline through to the week 1
Proportion of subjects experiencing "at least much improved" (including "much" and "very much improved") in Patient Global Impression of Change (PGI-C).From baseline through to the double blind period (week 12)
To assess adverse events as criteria for safety and tolerability of XEN1101From screening through to 56 days post-final dose.

Trial Locations

Locations (130)

Universitatsklinikum Bonn

🇩🇪

Bonn, Germany

Hospital Ramón y Cajal

🇪🇸

Madrid, Spain

Hospital Ruber Internacional

🇪🇸

Madrid, Spain

Hospital Vithas La Milagrosa

🇪🇸

Madrid, Spain

Hospital Clinico San Carlos

🇪🇸

Madrid, Spain

IIS-Fundacion Jimenez Diaz/Farmacia

🇪🇸

Madrid, Spain

Hospital Universitario 12 de Octubre

🇪🇸

Madrid, Spain

Hospital Regional De Malaga

🇪🇸

Málaga, Spain

Epilepsy Center Bethel

🇩🇪

Bielefeld, Germany

American Hospital Network LLC

🇬🇪

Tbilisi, Georgia

Institute of Neurology and Neuropsychology

🇬🇪

Tbilisi, Georgia

Vivantes Humboldt Klinikum

🇩🇪

Berlin, Germany

Strada Patient Care Center

🇺🇸

Mobile, Alabama, United States

Xenoscience

🇺🇸

Phoenix, Arizona, United States

St. Joseph's Hospital

🇺🇸

Phoenix, Arizona, United States

University of Arizona, Health Sciences Center

🇺🇸

Tucson, Arizona, United States

Clinical Trials, Inc

🇺🇸

Little Rock, Arkansas, United States

Brain Science Research Institute

🇺🇸

Los Angeles, California, United States

University of California, David Clinical & Translational Science Center Clinical Research (CCRC)

🇺🇸

Sacramento, California, United States

California Pacific Medical Center (CPMC)

🇺🇸

San Francisco, California, United States

Anschutz Health Sciences

🇺🇸

Aurora, Colorado, United States

Floridian Community Research Center

🇺🇸

Coral Gables, Florida, United States

Serenity Research

🇺🇸

Miami, Florida, United States

Research Institute of Orlando, LLC

🇺🇸

Orlando, Florida, United States

Panhandle Research & Medical Clinic

🇺🇸

Pensacola, Florida, United States

Medsol Clinical Research Center

🇺🇸

Port Charlotte, Florida, United States

University of South Florida

🇺🇸

Tampa, Florida, United States

Encore Medical Research of Weston, LLC

🇺🇸

Weston, Florida, United States

Emory Brain Health Center

🇺🇸

Atlanta, Georgia, United States

Georgia Neurology and Sleep Medicine Associates

🇺🇸

Suwanee, Georgia, United States

Hawaii Pacific Neuroscience

🇺🇸

Honolulu, Hawaii, United States

Consultants in Epilepsy and Neurology

🇺🇸

Boise, Idaho, United States

Rush University Medical Center

🇺🇸

Chicago, Illinois, United States

Indiana University, IU Health Partners, Adult Neurology Clinic

🇺🇸

Indianapolis, Indiana, United States

The University of Kansas Medical Center

🇺🇸

Kansas City, Kansas, United States

Bluegrass Epilepsy Research, LLC

🇺🇸

Lexington, Kentucky, United States

University of Kentucky, Dept. of Neurology

🇺🇸

Lexington, Kentucky, United States

MaineHealth Neurology - Scarborough

🇺🇸

Scarborough, Maine, United States

University of Maryland Medical Center

🇺🇸

Baltimore, Maryland, United States

Mid-Atlantic Epilepsy and Sleep Center

🇺🇸

Bethesda, Maryland, United States

MedStar Health Research Institute

🇺🇸

Clinton, Maryland, United States

Medstar Health Research Institute

🇺🇸

Hyattsville, Maryland, United States

Brigham and Women's Hospital

🇺🇸

Boston, Massachusetts, United States

UMass Memorial Medical Center

🇺🇸

Worcester, Massachusetts, United States

University of Michigan

🇺🇸

Ann Arbor, Michigan, United States

Michigan State University

🇺🇸

East Lansing, Michigan, United States

Cornwell Health

🇺🇸

Grand Rapids, Michigan, United States

Minneapolis Clinic of Neurology

🇺🇸

Burnsville, Minnesota, United States

Saint Louis University Medical School - Neurosciences Clinical Research Unit

🇺🇸

Saint Louis, Missouri, United States

Washington University, St. Louis

🇺🇸

Saint Louis, Missouri, United States

Northeast Epilepsy Group

🇺🇸

Hackensack, New Jersey, United States

Montefiore Medical Center

🇺🇸

Bronx, New York, United States

Dent Neurosciences Research Center

🇺🇸

Buffalo, New York, United States

NYU Comprehensive Epilepsy Center (CEC)

🇺🇸

New York, New York, United States

Weill Cornell Medicine/ New York-Presbyterian Hospital

🇺🇸

New York, New York, United States

Mount Sinai Medical Center

🇺🇸

New York, New York, United States

SUNY Upstate Medical University

🇺🇸

Syracuse, New York, United States

Onsite Clinical Solutions, LLC

🇺🇸

Charlotte, North Carolina, United States

Duke Neurology

🇺🇸

Durham, North Carolina, United States

Meridian Clinical Research, LLC

🇺🇸

Raleigh, North Carolina, United States

Wake Forest Baptist Health

🇺🇸

Winston-Salem, North Carolina, United States

Summa Health

🇺🇸

Akron, Ohio, United States

University of Toledo Medical Center

🇺🇸

Toledo, Ohio, United States

Providence Brain & Spine Institute

🇺🇸

Portland, Oregon, United States

Thomas Jefferson University

🇺🇸

Philadelphia, Pennsylvania, United States

Temple University Hospital

🇺🇸

Philadelphia, Pennsylvania, United States

Austin Epilepsy Care Center (AECC)

🇺🇸

Austin, Texas, United States

ANESC Research

🇺🇸

El Paso, Texas, United States

UT Physicians Epilepsy Clinic

🇺🇸

Houston, Texas, United States

UT Health San Antonio

🇺🇸

San Antonio, Texas, United States

Carilion Clinic - Neurology

🇺🇸

Roanoke, Virginia, United States

Sentara Neurology Specialists

🇺🇸

Virginia Beach, Virginia, United States

University of Washington Main Hospital

🇺🇸

Seattle, Washington, United States

Aurora St. Luke's Medical Center

🇺🇸

Milwaukee, Wisconsin, United States

Hospital General de Agudos J.M. Ramos Mejia

🇦🇷

Buenos Aires, Argentina

STAT Research S.A.

🇦🇷

Buenos Aires, Argentina

CENyR

🇦🇷

Caba, Argentina

Hospital Córdoba

🇦🇷

Córdoba, Argentina

Sanatorio del Sur S.A.

🇦🇷

Tucumán, Argentina

St Vincent's Hospital Melbourne

🇦🇺

Fitzroy, Melbourne, Australia

Royal Prince Alfred Hospital (RAPH)

🇦🇺

Camperdown, New South Wales, Australia

Prince of Wales Hospital

🇦🇺

Sydney, New South Wales, Australia

Southern Neurology

🇦🇺

Sydney, New South Wales, Australia

Westmead Hospital

🇦🇺

Westmead, New South Wales, Australia

The University of Queensland (UQ) - Mater Research Institute (MRI)

🇦🇺

Brisbane, Queensland, Australia

Austin Health Pharmacy Clinical Trials

🇦🇺

Heidelberg, Victoria, Australia

The Alfred Hospital (Alfred Health)

🇦🇺

Melbourne, Victoria, Australia

The Royal Melbourne Hospital

🇦🇺

Melbourne, Australia

MHAT Puls AD

🇧🇬

Blagoevgrad, Bulgaria

First Multiprofile Hospital for Active Treatment

🇧🇬

Sofia, Bulgaria

Center For Neurologic Research

🇨🇦

Lethbridge, Alberta, Canada

London Health Sciences Centre

🇨🇦

London, Ontario, Canada

Le Centre Hospitalier de l'Universite' de Montreal (CHUM)

🇨🇦

Montréal, Quebec, Canada

FORBELI s.r.o., Neurologicka ambulance

🇨🇿

Prague, Czechia

Epilepsiezentrum Frankfurt Rhein-Main

🇩🇪

Frankfurt, Germany

University Medical Center Freiburg

🇩🇪

Freiburg im Breisgau, Germany

Philipps-Universität Marburg

🇩🇪

Marburg, Germany

LMU Munich, Department of Neurology

🇩🇪

Munich, Germany

Epilepsiezentrum Kleinwachau Gemeinnutzige eGmbH

🇩🇪

Radeberg, Germany

Universitätsklinikum Tübingen

🇩🇪

Tübingen, Germany

Universitatsklinik fur neurologie, universitats - und Rehabilitationskliniken Ulm

🇩🇪

Ulm, Germany

Beaumont Hospital

🇮🇪

Dublin, Ireland

Istituto delle Scienze Neurologiche di Bologna

🇮🇹

Bologna, Italy

Università Degli Studi Gabriele d'Annunzio Di Chieti

🇮🇹

Pescara, Italy

Azienda Ospedaliero Universitaria Pisana

🇮🇹

Pisa, Italy

Ospedale Pediatrico Bambino Gesu

🇮🇹

Roma, Italy

Azienda Ospedaliero-Universitaria Policlinico Umberto I

🇮🇹

Rome, Italy

Pauls Stradina Clinical university hospital

🇱🇻

Riga, Latvia

Riga East University Hospital

🇱🇻

Riga, Latvia

University of Auckland

🇳🇿

Auckland, New Zealand

Waikato Hospital

🇳🇿

Hamilton, New Zealand

Centrum Medyczne Neuromed

🇵🇱

Bydgoszcz, Poland

NZOZ Novo-Med

🇵🇱

Katowice, Poland

Clinical Best Solutions

🇵🇱

Lublin, Poland

Twoja Przychodnia NCM

🇵🇱

Nowa Sól, Poland

Neurosphera Sp. z o.o.

🇵🇱

Warszawa, Poland

Unidade Local de Saúde de São João

🇵🇹

Porto, Portugal

Hospital Pedro Hispano

🇵🇹

Porto, Portugal

Unitat d'Assaigs Clínics. Servei de Farmàcia

🇪🇸

Barcelona, Spain

Hospital Universitario y Politecnico La Fe

🇪🇸

Valencia, Spain

Hospital Clínico Universitario Valladolid

🇪🇸

Valladolid, Spain

Mid Yorkshire Hospitals NHS Trust

🇬🇧

Wakefield, West Yorkshire, United Kingdom

University Hospitals Birmingham NHS Foundation Trust

🇬🇧

Birmingham, United Kingdom

University Hospital of Wales

🇬🇧

Cardiff, United Kingdom

Ninewells Hospital and Medical School

🇬🇧

Dundee, United Kingdom

Leeds Teaching Hospitals NHS Trust

🇬🇧

Leeds, United Kingdom

St. George's Hospital NHS Foundation Trust

🇬🇧

London, United Kingdom

Royal London Hospital for Integrated Medicine

🇬🇧

London, United Kingdom

John Radcliffe Hospital

🇬🇧

Oxford, United Kingdom

Northern Care Alliance NHS Foundation Trust, Salford Care Organisation

🇬🇧

Salford, United Kingdom

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