MedPath

Test Albuvirtide in Experienced Patients

Phase 3
Completed
Conditions
HIV Infections
AIDS
Interventions
Registration Number
NCT02369965
Lead Sponsor
Frontier Biotechnologies Inc.
Brief Summary

The purpose of this study is to evaluate the efficacy and safety of albuvirtide combined with lopinavir-ritonavir (LPV/r) in HIV-1-infected patients who failed first-line antiretroviral therapy (ART).

Detailed Description

This was a 48-week, multi-center, open-label, randomized and controlled, non-inferiority phase 3 clinical trial to evaluate the safety and efficacy of albuvirtide combined with LPV/r in HIV-1 infected patients who failed their first-line ART and had HIV-1 RNA levels ≥ 1000 copies/mL at screening.

The trial was conducted in 12 sites in China. Subjects meeting inclusion criteria were randomized in a 1:1 ratio to ABT group and NRTI group, in which the ABT group received albuvirtide and LPV/r combination therapy, and NRTI group received the standard 3-drug regimen of LPV/r + Lamivudine (3TC) + Tenofovir (TDF). If TDF was used in the previous regimen or genotypic resistance histories showed primary mutation to TDF, zidovudine (AZT) or abacavir (ABC) would be used. Albuvirtide was given by weekly intravenous infusion and LPV/r was given twice daily orally. A total of 418 subjects were randomized, of whom 401 received at least one treatment.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
418
Inclusion Criteria
  1. 16-60 years old, male or female.
  2. Those who meet the Diagnostic Criteria of AIDS and HIV Infection, the Health Industry Standard of the People's Republic of China (WS 293-2008).
  3. Those who have been undergoing antiretroviral treatment with nucleosides and non-nucleoside reverse transcriptase inhibitors (NRTIs+NNRTIs) for at least 6 months.
  4. HIV-RNA ≥ 1000 copies/mL.
  5. Those who have no serious hepatic or renal functional impairment and other parameters are generally in the normal ranges according to the comprehensive physical examinations (including general physical examination, routine blood and urine tests, blood chemistry tests, ECG, etc.).
  6. The subjects should have a full understanding of the objective, nature, methods of the trial and the possible reactions. He/She should participate in the trial voluntarily and should sign the informed consent form.
Exclusion Criteria
  1. Those who are in an acute stage of infection, or have suffered from AIDS-related diseases (e.g. opportunistic infections or malignant tumors, etc.) at enrollment; or have suffered from opportunistic infections within 3 months prior to enrollment and the conditions have not reached a stable state within 2 weeks prior to enrollment.
  2. Those who have used protease inhibitors or HIV fusion inhibitors for antiretroviral treatment, and who have participated in HIV vaccine clinical trials or have participated in other drug trials within recent 3 months.
  3. Those who have been co-administered antiviral treatment for hepatitis.
  4. Those whose screening test results meet one of the following: hemoglobin < 9 g/dL, WBC count <2×109/L, neutrophil count < 1×109/L, PLT count < 75×109/L, transaminase > 3×ULN, total bilirubin > 2×ULN, creatinine > 1×ULN, serum creatine phosphokinase > 2×ULN.
  5. Those with allergic constitution or known allergic to ingredients of the investigational drug or ART drugs prescribed in the protocol.
  6. Currently suffering from serious chronic diseases, metabolic diseases (such as diabetes mellitus), neurological and psychiatric disorders.
  7. Patients with hemophilia A or B.
  8. Those with suspected or confirmed history of alcohol or drug abuse.
  9. Pregnant or lactating women; or women of childbearing age who refuse to take contraceptive measures during the trial.
  10. Those for whom the possibility of being enrolled is low according to the judgment of the investigator (e.g. weak physical condition, poor compliance, etc.).

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
albuvirtide, lopinavir-ritonaviralbuvirtidealbuvirtide once a week and lopinavir-ritonavir twice daily for 48 weeks
albuvirtide, lopinavir-ritonavirlopinavir-ritonaviralbuvirtide once a week and lopinavir-ritonavir twice daily for 48 weeks
lopinavir-ritonavir,tenofovir,lamivudinelopinavir-ritonavirlopinavir-ritonavir twice daily, tenofovir once daily and lamivudine once daily for 48 weeks
lopinavir-ritonavir,tenofovir,lamivudinetenofovirlopinavir-ritonavir twice daily, tenofovir once daily and lamivudine once daily for 48 weeks
lopinavir-ritonavir,tenofovir,lamivudinelamivudinelopinavir-ritonavir twice daily, tenofovir once daily and lamivudine once daily for 48 weeks
Primary Outcome Measures
NameTimeMethod
Percentage of participants of virological suppression at Week 48Through Week 48

Percentage of participants with HIV-1 RNA \< 50 copies/mL at Week 48

Secondary Outcome Measures
NameTimeMethod
Changes of viral loadBaseline to Week 48

Changes of HIV-1 RNA relative to baseline at Week 48

Percentage of participants with HIV-1 RNA < 400 copies/mL at Week 48Through Week 48

Percentage of participants with HIV-1 RNA \< 400 copies/mL at Week 48

Changes of CD4 cell countBaseline to Week 48

Changes of CD4 cell count relative to baseline at Week 48

Trial Locations

Locations (12)

The Third People'S Hospital Of Shenzhen

🇨🇳

Shenzhen, Guangdong, China

The Second Xiangya Hospital of Central South University

🇨🇳

Changsha, Hunan, China

Beijing Youan Hospital, Capital medical university

🇨🇳

Beijing, Beijing, China

Affiliated Hangzhou Xixi Hospital,Zhejiang University School Of Medicine

🇨🇳

Hangzhou, Zhejiang, China

Beijing Ditan Hospital, Capital Medical University

🇨🇳

Beijing, Beijing, China

Tangdu Hospital, Fourth Military Medical University

🇨🇳

Xi'an, Shanxi, China

The First Hospital of Changsha

🇨🇳

Changsha, Hunan, China

302 Hospital People's Liberation Army Of China

🇨🇳

Beijing, Beijing, China

Henan Infectious Disease Hospital

🇨🇳

Zhengzhou, Henan, China

Guangzhou Eighth People's Hospital

🇨🇳

Guangzhou, Guangdong, China

Shanghai Public Health Clinical Center

🇨🇳

Shanghai, Shanghai, China

The First Affiliated Hospital Zhejiang University School Of Medicine

🇨🇳

Hangzhou, Zhejiang, China

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