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Antitumoral Activity and Safety of AEZS-108 in Women With LHRH Receptor Positive Gynecological Tumors

Phase 2
Completed
Conditions
Ovarian Cancer
Endometrial Cancer
Registration Number
NCT00569257
Lead Sponsor
AEterna Zentaris
Brief Summary

The purpose of this study is to determine whether AEZS-108 shows anti-tumor activity and is tolerated in patients with gynecological tumors (ovarian / endometrial cancer) that have been shown to express receptors for the luteinizing hormone releasing hormone (LHRH)

Detailed Description

The ovary and the endometrium are hormone dependent organs. Receptors for different sex hormones are found commonly in epithelial ovarian and endometrial cancers. LHRH and its receptors are expressed in about 80% of human ovarian and endometrial cancers. As binding sites are present on tumors in higher concentrations than on most normal tissues, these receptors represent a specific target for AEZS-108 in which doxorubicin is coupled to an LHRH analog.

Patients whose tumor specimen have shown to be positive for LHRH receptor expression will be investigated for tumor response and tolerability.

Recruitment & Eligibility

Status
COMPLETED
Sex
Female
Target Recruitment
85
Inclusion Criteria
  • LHRH receptor positive tumor status: positive receptor status determined by immunohistochemistry from primary tumor
  • Histologically confirmed epithelial ovarian cancer (Stratum A)
  • Advanced (FIGO III or IV) or recurrent disease
  • Progression during treatment with a platinum-based regimen or within 6 months after receiving a platinum-based regimen
  • Previous treatment with a taxane-containing regimen
  • At least one measurable target lesion (RECIST criteria) OR CA125 level higher than twice the upper limit of normal range (GCIG criteria)
  • Histologically confirmed endometrial cancer (Stratum B)
  • Advanced (FIGO III or IV) or recurrent disease not amenable to potentially curative treatment with local surgery and/or radiation therapy
  • No previous anthracycline-based chemotherapy
  • At least one measurable target lesion according to RECIST criteria
Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Primary Outcome Measures
NameTimeMethod
Tumor response as per RECIST or (for Ovarian CA patients without evaluable target lesion following RECIST) GCIG criteriaup to six 3-weekly treatment cycles
Secondary Outcome Measures
NameTimeMethod
Time-to-progression (TTP); Overall survivalup to observation of event
Safety of AEZS-108 (possibly drug-related adverse events)4 weeks beyond last drug admnistration

Trial Locations

Locations (17)

Klinik für Frauenheilkunde und Geburtshilfe, Universitätsklinikum Carl Gustav Carus

🇩🇪

Dresden, Germany

Frauenklinik, St. Vincentius Kliniken AG

🇩🇪

Karlsruhe, Germany

Klinik für Frauenheilkunde, Universität Erlangen-Nürnberg

🇩🇪

Erlangen, Germany

Universitätsfrauenklinik, Klinikum der JWG Universität Frankfurt

🇩🇪

Frankfurt / Main, Germany

Frauenklinik, Klinikum Bremen-Mitte GmbH

🇩🇪

Bremen, Germany

Frauenklinik, Medizinische Hochschule Hannover

🇩🇪

Hannover, Germany

Klinik für Gynäkologie und Geburtshilfe, Universitätsklinikum Schleswig-Holstein, Campus Kiel

🇩🇪

Kiel, Germany

Klinikum Suedstadt der Hansestadt Rostock, Universitaetsfrauenklinik und Poliklinik

🇩🇪

Rostock, Germany

Klinik f. Gynäkologie u. Gyn. Onkologie, Dr. Horst Schmidt Kliniken GmbH

🇩🇪

Wiesbaden, Germany

Frauenklinik, Klinikum Lüneburg

🇩🇪

Lüneburg, Germany

Universitätsfrauenklinik, Universitätsklinikum

🇩🇪

Essen, Germany

Regional Oncodispensary "M.Markov"

🇧🇬

Varna, Bulgaria

University Hospital "Dr. Georgy Stranski"

🇧🇬

Pleven, Bulgaria

Regional Oncology Hospital Plovdiv

🇧🇬

Plovdiv, Bulgaria

Frauenklinik, Georg-August-Universität Göttingen

🇩🇪

Göttingen, Germany

Klinik für Frauenheilkunde und Geburtshilfe, Charité Campus Virchow-Klinikum

🇩🇪

Berlin, Germany

Klinikum der Ernst-Moritz-Arndt-Universitaet, Klinik und Poliklinik fuer Gynaekologie und Geburtshilfe

🇩🇪

Greifswald, Germany

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