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The Efficacy and Safety of Third-generation TKIs Combined With Azacitidine and Bcl-2 Inhibitor in Patients With CML-MBP

Not yet recruiting
Conditions
Chronic Myeloid Leukemia
Interventions
Registration Number
NCT06390306
Lead Sponsor
Peking University People's Hospital
Brief Summary

This is a prospective multi-center study to investigate efficacy and safety of the third generation tyrosine kinase inhibitors (TKIs) combined with azacitidine and B-cell lymphoma-2 (Bcl-2) inhibitor in patients with myeloid blast phase chronic myeloid leukemia (CML-MBP).

Detailed Description

CML-MBP has dismal outcome. Currently, there is no standardized induction treatment approach in CML-MBP. The European LeukemiaNet (ELN) recommendations and NCCN guideline recommended the combination of TKI and chemotherapy in CML-MBP. The previous study revealed that TKI combined with hypomethylating agents had promising efficacy. However, imatinib and second generation TKI are the most widely applied in combination treatment, there is limited data in third generation TKI.

Currently, venetoclax in combination with hypomethylating agents such as azacitidine is standard treatment for patients with AML unsuitable for intensive induction chemotherapy. Maiti et al. reported that TKI combined with venetoclax and detectable had promising efficacy in CML-MBP. Therefore, the investigator conducted a study to explore the efficacy and safety of a third generation TKI in combination with azacitidine and Bcl-2 inhibitor in CML-MBP and multi-omics exploratory analysis was performed to identify potential biomarkers correlated with the outcome.

Recruitment & Eligibility

Status
NOT_YET_RECRUITING
Sex
All
Target Recruitment
30
Inclusion Criteria
  1. age ≥ 18 years old;
  2. philadelphia chromosome (Ph)-positive or BCR::ABL-positive;
  3. serum creatinine ≤ 1.5 × upper limit of normal (ULN) or 24h creatinine clearance ≥ 50 mL/min when serum creatinine was > 1.5 × ULN;
  4. serum total bilirubin ≤ 1.5 × ULN;
  5. aspartate aminotransferase and alanine aminotransferase ≤ 2.5 × ULN;
  6. amylase ≤ 1.5 × ULN; (7) lipase ≤ 1.5 × ULN;
  7. ejection fraction > 50%; corrected QT interval on electrocardiographic evaluation was ≤ 450 ms in men or ≤ 470 ms in women.
Exclusion Criteria
  1. concurrent diseases requiring treatment(s) with potential to interact with 3G-TKI;
  2. diagnosis of other primary malignancies;
  3. history of allogeneic HSCT;
  4. extramedullary disease only.

Study & Design

Study Type
OBSERVATIONAL
Study Design
Not specified
Arm && Interventions
GroupInterventionDescription
3G-TKI + AZA + Ven groupPonatinibAdult CML-MBP
3G-TKI + AZA + Ven groupVenetoclaxAdult CML-MBP
3G-TKI + AZA + Ven groupAzacitidineAdult CML-MBP
3G-TKI + AZA + Ven groupOlverembatinibAdult CML-MBP
Primary Outcome Measures
NameTimeMethod
Major hematologic response (MaHR)At the end of Cycle 2 (each cycle is 28 days)

either a complete hematologic response (CHR) or no evidence of leukemia (NEL).

Secondary Outcome Measures
NameTimeMethod
Return to chronic phaseAt the end of Cycle 2 (each cycle is 28 days)

\< 10% blasts in blood and bone marrow with no extra-medullary leukemia and last for ≥ 4 weeks

SurvivalUp to 3 years

interval from therapy start to death from any cause or censored at the last follow-up

Major cytogenetic response (MCyR)Up to 3 years

Ph-positive cells ≤ 35%

Major molecular response (MMR)Up to 3 years

BCR::ABL1IS ≤ 0.1%

Event-free survival (EFS)Up to 3 years

interval from therapy start to lacking RCP after 1 cycle, MaHR after 2 cycles, loss of hematologic response, progression to blast phase again, or death from any causes

CML-related survivalUp to 3 years

interval from therapy start to death from blast phase, or censored at the last follow-up

Incidence of adverse eventsUp to 3 years

Adverse effects (AEs) were graded according to the National Cancer Institute Common Terminology Criteria for Adverse Events, version 5.0. and assessed continuously.

Complete cytogenetic response (CCyR)Up to 3 years

no Ph-positive cell

Trial Locations

Locations (1)

Peking university people's hospital

🇨🇳

Beijing, Beijing, China

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