MedPath

Assessment and Monitoring of Renal Proximal Tubular Tolerance of Nucleoside and Nucleotide Analogues Using Early Screening Tools in Patients Chronically Mono-infected With Hepatitis B Virus

Completed
Conditions
Renal Failure With Tubular Necrosis
Hepatitis B
Interventions
Biological: plasma and urine samples, sample with ADN
Registration Number
NCT01500265
Lead Sponsor
University Hospital, Limoges
Brief Summary

Nucleotide analogues are associated in the long term with a risk of proximal tubular nephropathy (PT) with loss of phosphate, and, when compensatory mechanisms are overwhelmed, with osteopenia or osteoporosis. This toxicity has been particularly documented for tenofovir (TDF) in HIV disease, but its prevalence varies widely in the literature and is mainly associated with comorbidities: on average this prevalence is 0.39% after 48 weeks with exceptional cases of Fanconi syndrome described. In HBV monoinfection after 60 months of treatment with TDF, an 11% decrease of creatinine clearance (CreatCl) is observed. A single study showed a significant increase in creatinine level with entecavir (ETV) therapy, a second-generation nucleoside, hitherto not described as nephrotoxic. Furthermore, if the direct renal toxic effect characteristic of HIV in the kidney is well known, the role of HBV is less clear. Thus, HBV treatment appears to have a renal protective effect. The monitoring tools recommended by the SPC, CreatCl and plasma phosphorus level are late markers of tubular damage. The threshold of phosphate tubular reabsorption (TmPi/GFR) and the fractional excretion of uric acid (FEUA) are unexpensive early screening tools. However, the long-term evolution of this subclinical tubular involvement in HBV monoinfection is not known.

Detailed Description

260 naive untreated patients, 220 patients treated with TDF and 220 patients treated with ETV and consecutively recruited in this interventional study, will have at baseline and every three months, a determination of phosphorus, creatinine, uric acid in plasma and urine samples for determination of TMPi / GFR and FEUA, and an evaluation of urinary calcium level. Depending on local opportunities, every six months, a urine sample will be stored in a declared biological collection to perform β2-microglobuline and cystatin dosage. A 25-OHD3 and PTH dosage will be conducted annually. A sample of genomic DNA will be collected after informed consent of the patient from a saliva sample (Saliva autocollection kits) in order to investigate genetic polymorphism in transporters responsible for the renal elimination of TDF and ETV. A serum sample will be stored at baseline, at one year and at endpoint for the retrospective dosage of bone markers (bone PAlk, PINP and CTX).

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
216
Inclusion Criteria
  • Age ≥ 18 years
  • Patients with chronic HBV virus monoinfected
  • For groups of patients treated: Patients with an indication of ETV or TDF
  • For the group of naive patients: treatment-naive patients who have no indication of treatment (or do not want) for the duration of the study
  • globular filtration rate (GFR) ≥ 50 ml / min / 1.73 m2 with no known cause of renal disease
  • Patients who have given their informed and written informed consent
  • Women of childbearing potential with an effective method of contraception without interruption for the duration of the research and during the 4 months after stopping treatment
Exclusion Criteria
  • Patients co-infected with HIV, hepatitis C or hepatitis Delta
  • Patients who have already received the TDF in the group to receive the TDF and having already received ETV in the group to receive ETV
  • Patient with a GFR <50 ml / min / 1.73 m2 or with known causes of renal disease
  • Patient with hypophosphatemia <0.48 mmol / l
  • Patients with hepatocellular carcinoma (diagnosed or suspected)

Study & Design

Study Type
OBSERVATIONAL
Study Design
Not specified
Arm && Interventions
GroupInterventionDescription
Patient naiveplasma and urine samples, sample with ADNPatient with hepatitis B virus naive untreated
Patient with TDFplasma and urine samples, sample with ADNPatient with hepatits B treated with Tenofovir
Patient with ETVplasma and urine samples, sample with ADNPatient with hepatitis B virus treated with Entecavir
Primary Outcome Measures
NameTimeMethod
the prevalence of "subclinical" proximal tubular abnormalities2 years

to compare at 2 years the prevalence of "subclinical" proximal tubular abnormalities (TmPi/GFR and FEUA) in 3 groups of HBV monoinfected patients treated with TDF, ETV or untreated.

Secondary Outcome Measures
NameTimeMethod
the prevalence at baseline of "subclinical" proximal tubular abnormalities1 day

to describe the prevalence at baseline, and the cumulative incidence of these abnormalities during the follow-up and determine the proportion of patients who present at 2 years an impaired CreatCl, an hypophosphatemia and an hypercalciuria (suggesting a bone impact), according to the presence or absence of "subclinical" proximal tubular abnormalities.

Trial Locations

Locations (25)

AP-HP - Hôpital Kremlin Bicêtre

🇫🇷

Le Kremlin Bicêtre, France

CHU de Nice

🇫🇷

Nice, France

CHU de Tours - Hôpital Trousseau

🇫🇷

Tours, France

CHU de Poitiers

🇫🇷

Poitiers, France

CHU de Clermont Ferrand

🇫🇷

Clermont Ferrand, France

Centre Hospitalier d'Hyères

🇫🇷

Hyères, France

CHU de Limoges - Fédération Hépatologie

🇫🇷

Limoges, France

CHU de Bordeaux - Hôpital Haut Levêque

🇫🇷

Pessac, France

AP-HP - Hôpital Beaujon

🇫🇷

Clichy, France

CHU de Point à Pitre

🇫🇷

Point à Pitre, France

CHU d'Angers

🇫🇷

Angers, France

CHU de Besancon

🇫🇷

Besancon, France

CHU de Montpellier - Hôpital Saint Eloi

🇫🇷

Montpellier, France

CHU de Nancy - Hôpital Brabois

🇫🇷

Vandoeuvre les Nancy, France

AP-HP - Hôpital La Pitié Salpétrière

🇫🇷

Paris, France

AP-HP - Hôpital Bichat

🇫🇷

Paris, France

CHU d'Amiens

🇫🇷

Amiens, France

CHU de CAEN

🇫🇷

Caen, France

CHU de Bordeaux - Hôpital Saint André

🇫🇷

Bordeaux, France

CHU de Brest

🇫🇷

Brest, France

Centre Hospitalier Laennec de Creil

🇫🇷

Creil, France

Centre Hospitalier de La Roche sur Yon

🇫🇷

La Roche sur Yon, France

CHU de Lille - Hôpital Huriet

🇫🇷

Lille, France

CHU de Strasbourg - Hôpital Civil

🇫🇷

Strasbourg, France

Hospices Civils de Lyon - Hôpital Croix Rousse

🇫🇷

Lyon, France

© Copyright 2025. All Rights Reserved by MedPath