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A Formulation Screening Study of Dalcetrapib and Atorvastatin in Healthy Volunteers

Phase 1
Completed
Conditions
Healthy Volunteer
Interventions
Registration Number
NCT01363999
Lead Sponsor
Hoffmann-La Roche
Brief Summary

A single-center, crossover study to evaluate the pharmacokinetics of dalcetrapib and atorvastatin from prototype fixed dose combination formulations in healthy volunteers. Volunteers will receive a single dose of dalcetrapib with atorvastatin in each of four treatment periods.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
24
Inclusion Criteria
  • Healthy volunteers, 18 to 55 years of age, inclusive
Exclusion Criteria
  • Any concomitant disease or ongoing condition that in the investigator's opinion could interfere with the study or could pose an unacceptable risk to the patient
  • Clinically significant abnormal laboratory values

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
DdalcetrapibRO4607381/F49 tablet
AdalcetrapibRO5317116/F01 bilayer tablet
AatorvastatinRO5317116/F01 bilayer tablet
BdalcetrapibRO5317116/F03 bilayer tablet
BatorvastatinRO5317116/F03 bilayer tablet
CatorvastatinRO5317116/F04 active-coated tablet
CdalcetrapibRO5317116/F04 active-coated tablet
DatorvastatinRO4607381/F49 tablet
Primary Outcome Measures
NameTimeMethod
Plasma Concentration of Dalcetrapib Active Form3 days
Plasma Concentration of Atorvastatin3 days
Secondary Outcome Measures
NameTimeMethod
Safety: Incidence of Serious Adverse Events9 weeks
Plasma Concentration of Atorvastatin Metabolites3 days

Measuring the amount of byproducts of the metabolization of Atorvastatin in the blood plasma.

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