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Study to Evaluate Effects of INL1 in Patients With Heart Failure and Reduced Ejection Fraction

Phase 2
Conditions
Reduced Ejection Fraction
Heart Failure
Interventions
Other: Placebo
Registration Number
NCT03875183
Lead Sponsor
Innolife Co., Ltd.
Brief Summary

This is a multicenter, randomized, double-blind, placebo-controlled, dose-response trial in patients with chronic stable Heart Failure (HF) and reduced Left Ventricular Ejection Fraction (LVEF) to evaluate the efficacy and safety of three INL1 doses compared with placebo. Patients will be treated for approximately 12 weeks with one of three INL1 doses: 50 mg, 150 mg, 300 mg, or, placebo capsules, taken twice daily (BID).

Detailed Description

Not available

Recruitment & Eligibility

Status
UNKNOWN
Sex
All
Target Recruitment
200
Inclusion Criteria
  • Clinical diagnosis of HF requiring chronic treatment of loop diuretics
  • Left Ventricular Ejection Fraction (LVEF) ≤ 40% at screening by echocardiography
  • N-Terminal-prohormone of Brain Natriuretic Peptide (NT-proBNP) ≥400 pg/mL at screening for patients without atrial fibrillation or atrial flutter, or, NT-proBNP ≥ 1,200 pg/mL at screening for patients with atrial fibrillation or atrial flutter
  • Treated for Heart Failure with stable, optimal pharmacological therapy
  • Acceptable screening echocardiographic image quality
Exclusion Criteria
  • Female patients of childbearing potential
  • Patients with a New York Heart Association (NYHA) Class I or IV
  • Heart failure that is clearly caused by toxin / drug such as Adriamycin
  • Significant medical conditions or recent history suggesting the patient's study participation will potentially pose a major risk to patient's safety and well-being
  • Need for routine scheduled outpatient IV infusions for Heart Failure or scheduled ultrafiltration
  • History of rhabdomyolysis or history of autoimmune diseases
  • Severe renal disease
  • Hepatic disease
  • Pulmonary disease limiting exercise capacity
  • Atrial fibrillation with rapid ventricular response
  • Life expectancy of less than 6 months
  • Type 1 diabetes mellitus or Type 2 diabetes mellitus with very poor glycemic control
  • Patients with anemia

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
INL1 50mg BIDINL1INL1 50mg dose to be given twice daily using one 50mg capsule and two matching placebo capsules at each dose
INL1 300 mg BIDINL1INL1 300mg dose to be given twice daily using three 100mg capsules at each dose
PlaceboPlaceboPlacebo dose to be given twice daily using 3 placebo capsules at each dose
INL1 150 mg BIDINL1INL1 150mg dose to be given twice daily using three 50mg capsules at each dose
Primary Outcome Measures
NameTimeMethod
Proportional change in N-terminal prohormone of brain natriuretic peptide (NT-proBNP)Baseline - 12 weeks

Proportional change in N-terminal prohormone of brain natriuretic peptide (NT-proBNP) from Baseline to 12 weeks

Secondary Outcome Measures
NameTimeMethod
Composite Heart Failure (HF) Improvement ScoreBaseline - 12 weeks

Composite HF Improvement Score, summarizing changes in 4 HF outcomes (NT-proBNP, left ventricular end-systolic volume \[LVESV\], NYHA class, and 6 Minute Walk Test) from Baseline to 12 weeks

Change in Left Ventricular End Diastolic (LVED)Baseline - 12 weeks

Echocardiogram finding: change in LVED from Baseline to 12 weeks

Change in ratio of mitral peak velocity of early filling (E) to early diastolic mitral annular velocity (E')Baseline - 12 weeks

Echocardiogram finding: change in E/E' ratio from Baseline to 12 weeks

Change in Left Atrial Volume (LAV)Baseline - 12 weeks

Echocardiogram finding: change in LAV from Baseline to 12 weeks

Change in Left Ventricular End Systolic (LVES)Baseline - 12 weeks

Echocardiogram finding: change in LVES from Baseline to 12 weeks

Change in Left Ventricular End Diastolic Volume (LVEDV)Baseline - 12 weeks

Echocardiogram finding: change in LVEDV from Baseline to 12 weeks

Change in Left Ventricular End Systolic Volume (LVESV)Baseline - 12 weeks

Echocardiogram finding: change in LVESV from Baseline to 12 weeks

Change in Left Ventricular Systolic Volume (LVSV)Baseline - 12 weeks

Echocardiogram finding: change in LVSV from Baseline to 12 weeks

Change in Left Ventricular Ejection Fraction (LVEF)Baseline - 12 weeks

Echocardiogram finding: change in LVEF from Baseline to 12 weeks

Change in Left Ventricular Mass (LVM)Baseline - 12 weeks

Echocardiogram finding: change in LVM from Baseline to 12 weeks

Change in Left Ventricular End Diastolic Diameter (LVEDD)Baseline - 12 weeks

Echocardiogram finding: change in LVEDD from Baseline to 12 weeks

Change in Left Ventricular End Systolic Diameter (LVESD)Baseline - 12 weeks

Echocardiogram finding: change in LVESD from Baseline to 12 weeks

Change in Left Ventricular Fractional Shortening (LVFS)Baseline - 12 weeks

Echocardiogram finding: change in LVFS from Baseline to 12 weeks

Change in Tricuspid Annular Plane Systolic Excursion (TAPSE)Baseline - 12 weeks

Echocardiogram finding: change in TAPSE from Baseline to 12 weeks

Change in Tricuspid Regurgitation (TR) peak velocityBaseline - 12 weeks

Echocardiogram finding: change in TR peak velocity from Baseline to 12 weeks

Change in Tricuspid Regurgitation (TR) gradientBaseline - 12 weeks

Echocardiogram finding: change in TR gradient from Baseline to 12 weeks

Change in Tricuspid Regurgitation (TR) severityBaseline - 12 weeks

Echocardiogram finding: change in TR severity from Baseline to 12 weeks

Change in Inferior Vena Cava (IVC) DiameterBaseline - 12 weeks

Echocardiogram finding: change IVC Diameter from Baseline to 12 weeks

Change in New York Heart Association (NYHA) classBaseline to 12 weeks

Change in NYHA class from Baseline to 12 weeks

Change in 6 minute walk distanceBaseline to 12 weeks

Change in 6 minute walk distance from Baseline to 12 weeks

Quality of Life (QoL) based on Kansas City Cardiomyopathy Questionnaire (KCCQ) changeBaseline to 12 weeks

QoL based on change in KCCQ from Baseline to 12 weeks. Quality of Life scale can range from 0 to 100, with higher values indicating a better outcome. Change will be calculated by subtraction.

Time to earliest event among the composite of cardiovascular (CV) death, hospitalization for HF, and unplanned use of intravenous diuretics or intensification of oral diuretic doseBaseline to 12 weeks

Time to earliest event among the composite of CV death, hospitalization for HF, and unplanned use of intravenous diuretics or intensification of oral diuretic dose from Baseline to 12 weeks

Trial Locations

Locations (13)

Stern Cardiovascular

🇺🇸

Germantown, Tennessee, United States

UCLA School of Medicine

🇺🇸

Torrance, California, United States

Innovative Research of West Florida, Inc.

🇺🇸

Clearwater, Florida, United States

Universal Axon Clinical Research

🇺🇸

Doral, Florida, United States

Via Christi Research, a division of Via Christi Hospitals Wichita, Inc.

🇺🇸

Wichita, Kansas, United States

Grady Clinical Research Center

🇺🇸

Atlanta, Georgia, United States

Clinical Trials of America LA, LLC

🇺🇸

Monroe, Louisiana, United States

Clinical Research of Gastonia

🇺🇸

Gastonia, North Carolina, United States

St Louis Heart and Vascular

🇺🇸

Saint Louis, Missouri, United States

East Texas Cardiology

🇺🇸

Houston, Texas, United States

Angiocardiac Care of Texas

🇺🇸

Houston, Texas, United States

Chongqing University 3 Gorges Hospital

🇨🇳

Chongqing, China

Medication Management, LLC

🇺🇸

Greensboro, North Carolina, United States

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