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A Study of Different Doses of Sitagliptin (MK-0431) in Participants With Type 2 Diabetes Mellitus (MK-0431-014)

Phase 2
Completed
Conditions
Type II Diabetes Mellitus
Interventions
Registration Number
NCT00481663
Lead Sponsor
Merck Sharp & Dohme LLC
Brief Summary

A study of different doses of MK-0431 in participants with type 2 diabetes mellitus. There have been 3 extensions to the base study (Extension 1: up to Week 52, Extension 2: up to Week 106, and Extension 3: up to Week 158). The primary hypothesis for the study is that In participants with type 2 diabetes who have inadequate glycemic control, after 12 weeks of treatment, a dose-response will be seen across once-daily doses of MK-0431 in lowering hemoglobin A1C (HbA1c).

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
555
Inclusion Criteria
  • Men and non-pregnant women
  • Fasting plasma glucose >= 130 mg/dL
  • HbA1c >=6.5% and >10.0%
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Exclusion Criteria
  • You have a history of type I diabetes
  • You are on a weight loss program with ongoing weight loss or taking weight loss medication
  • You have had surgery within 30 days
  • You hvae hepatitis B or C.
Read More

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Sitagliptin 25 mg once dailyRescueSitaglipin (MK-0431), 25 mg, once daily for 12 weeks, orally. Due to interim analysis of this study and another Phase IIB study, participants in this arm were switched into the 100-mg once daily arm during either the first or initiation of the second extensions study periods.
Sitagliptin 50 mg once dailyRescueSitagliptin, 50 mg, once daily for 12 weeks, orally. Due to interim analysis of this study and another Phase IIB study, participants in this arm were switched into the 100-mg once daily arm during either the first or initiation of the second extensions study periods.
Sitaglipin 100 mg once dailyRescueSitagliptin, 100 mg, once daily for 158 weeks, orally
Sitagliptin 50 mg twice dailyRescueSitagliptin 50 mg, twice daily for 12 weeks, orally. Due to interim analysis of this study and another Phase IIB study, participants in this arm were switched into the 100-mg once daily arm during either the first or initiation of the second extensions study periods.
Placebo to Sitagliptin → MetforminPlacebo to sitagliptinPlacebo to Sitagliptin, once daily, orally for 12 weeks. Participants randomized to the placebo treatment group during the base study were reallocated to treatment with metformin 850 mg twice daily (b.i.d., initiated with 850 mg q.d. for 4 weeks then force titrated to 850 mg b.i.d.) during either the first or initiation of the second extensions study periods.
Placebo to Sitagliptin → MetforminRescuePlacebo to Sitagliptin, once daily, orally for 12 weeks. Participants randomized to the placebo treatment group during the base study were reallocated to treatment with metformin 850 mg twice daily (b.i.d., initiated with 850 mg q.d. for 4 weeks then force titrated to 850 mg b.i.d.) during either the first or initiation of the second extensions study periods.
Sitagliptin 25 mg once dailySitagliptinSitaglipin (MK-0431), 25 mg, once daily for 12 weeks, orally. Due to interim analysis of this study and another Phase IIB study, participants in this arm were switched into the 100-mg once daily arm during either the first or initiation of the second extensions study periods.
Sitagliptin 50 mg once dailySitagliptinSitagliptin, 50 mg, once daily for 12 weeks, orally. Due to interim analysis of this study and another Phase IIB study, participants in this arm were switched into the 100-mg once daily arm during either the first or initiation of the second extensions study periods.
Sitagliptin 50 mg twice dailySitagliptinSitagliptin 50 mg, twice daily for 12 weeks, orally. Due to interim analysis of this study and another Phase IIB study, participants in this arm were switched into the 100-mg once daily arm during either the first or initiation of the second extensions study periods.
Sitaglipin 100 mg once dailySitagliptinSitagliptin, 100 mg, once daily for 158 weeks, orally
Placebo to Sitagliptin → MetforminMetforminPlacebo to Sitagliptin, once daily, orally for 12 weeks. Participants randomized to the placebo treatment group during the base study were reallocated to treatment with metformin 850 mg twice daily (b.i.d., initiated with 850 mg q.d. for 4 weeks then force titrated to 850 mg b.i.d.) during either the first or initiation of the second extensions study periods.
Primary Outcome Measures
NameTimeMethod
Number of Participants Who Experienced One or More Adverse Events (AE) up to Week 14Up to Week 14
Number of Participants Who Experienced One or More AE up to Week 160Up to Week 160
Change from Baseline in HbA1C at Week 12Baseline and Week 12
Number of participants Who Discontinued Study Treatment Due to An AE up to Week 12Up to Week 12
Number of participants Who Discontinued Study Treatment Due to An AE up to Week 106Up to Week 106
Number of participants Who Discontinued Study Treatment Due to An AE up to Week 158Up to Week 158
Number of Participants Who Experienced One or More AE up to Week 54Up to Week 54
Number of Participants Who Experienced One or More AE up to Week 108Up to Week 108
Number of participants Who Discontinued Study Treatment Due to An AE up to Week 52Up to Week 52
Secondary Outcome Measures
NameTimeMethod
Change from Baseline in HbA1C at Week 106Baseline and Week 106
Change from Baseline in FPG at Week 158Baseline and Week 158
Change from Baseline in Body Weight at Week 106Baseline and Week 106
Change From Baseline in Daily Seven-Point Fingerstick Glucose Average at Week 12Baseline and Week 12
Change From Baseline in Daily Seven-Point Fingerstick Glucose Average at Week 52Baseline and Week 52
Change from Baseline in FPG at Week 52Baseline and Week 52
Change from Baseline in Body Weight at Week 52Baseline and Week 52
Change from Baseline in Body Weight at Week 158Baseline and Week 158
Change From Baseline in Serum Fructosamine at Week 12Baseline and Week 12
Change from Baseline in HbA1C at Week 52Baseline and Week 52
Change from Baseline in HbA1C at Week 158Baseline and Week 158
Change from Baseline in Fasting Plasma Glucose (FPG) at Week 12Baseline and Week 12
Change from Baseline in FPG at Week 106Baseline and Week 106
Change from Baseline in Body Weight at Week 12Baseline and Week 12
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