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Dose Escalation Study of LGH447 in Japanese Patients With Relapsed and/or Refractory Hematologic Malignancies

Phase 1
Completed
Conditions
Multiple Myeloma
Interventions
Registration Number
NCT02160951
Lead Sponsor
Novartis Pharmaceuticals
Brief Summary

This is a multi-center, open-label, dose escalation, Phase 1 study of oral LGH447 in Japanese patients with relapsed and/or refractory multiple myeloma for which no standard effective treatment options exist.

The study consists of a dose escalation part to estimate the maximum tolerated dose and/or the recommended dose for expansion and a dose expansion part to further assess safety and preliminary anti-cancer activity of LGH447 at the maximum tolerated dose and/or the recommended dose for expansion.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
13
Inclusion Criteria

-Confirmed diagnosis of relapsed and/or refractory MM for which no standard effective treatment options exist.

Exclusion Criteria

-Uncontrolled cardiovascular condition, including ongoing cardiac arrhythmias, congestive heart failure, angina, or myocardial infarction within the past 6 months.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
LGH447LGH447LGH447, QD
Primary Outcome Measures
NameTimeMethod
Incidence rate of dose limiting toxicities28 days

Estimate the maximum tolerated dose and/or recommended dose for expansion of LGH447 in Japanese patients

Secondary Outcome Measures
NameTimeMethod
Pharmacokinetics profile of LGH447 and its metabolites if appropriateBaseline, 0.5, 1, 2, 3, 4, 5, 6, 8, 24 hours on Cycle1Day1, 14 and 28 and baseline on Cycle2Day14 and Cycle3Day1

PK parameters such as AUC, Cmax, Tmax, T1/2. Cycle = 28 days

Number of patients with adverse events as a measure of safety and tolerability of LGH44728 days and till the end of the study, an average of 84 days

Adverse events, serious adverse events, changes in laboratory values, and electrocardiograms

Duration of ResponseEvery 28 days till the end of the study, an average of 84 days, from the first documented onset of confirmed PR or better response to the date of documented disease progression/relapse or death due to multiple myeloma

Describe any preliminary anti-cancer activity associated with LGH447 based on International Myeloma Working group Criteria with modification.

Overall Response RateEvery 28 days till the end of the study, an average of 84 days

Describe any preliminary anti-cancer activity associated with LGH447 based on International Myeloma Working group Criteria with modification.

Disease control rateEvery 28 days till the end of the study, an average of 84 days

Describe any preliminary anti-cancer activity associated with LGH447 based on International Myeloma Working group Criteria with modification.

Clinical benefit rateEvery 28 days till the end of the study, an average of 84 days

Describe any preliminary anti-cancer activity associated with LGH447 based on International Myeloma Working group Criteria with modification.

Progression Free SurvivalEvery 28 days till the end of the study, an average of 84 days, from start of treatment to the date of event defined as the first documented disease progression/relapse, or death due to any cause

Describe any preliminary anti-cancer activity associated with LGH447 based on International Myeloma Working group Criteria with modification.

Time to responseEvery 28 days till the end of the study, an average of 84 days, from start of treatment until first documented best overall response

Describe any preliminary anti-cancer activity associated with LGH447 based on International Myeloma Working group Criteria with modification.

Trial Locations

Locations (1)

Novartis Investigative Site

🇯🇵

Okayama-city, Okayama, Japan

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