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Randomized Clinical Trial Of Bococizumab (PF-04950615; RN316) In Subjects With Hyperlipidemia Or Mixed Dyslipidemia At Risk Of Cardiovascular Events

Phase 3
Completed
Conditions
Hyperlipidemia
Interventions
Registration Number
NCT01968954
Lead Sponsor
Pfizer
Brief Summary

This study is a multicenter, randomized study in subjects with high cholesterol receiving highly effective statins to assess the efficacy, safety and tolerability of Bococizumab (PF-04950615;RN316) to lower LDL-C.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
711
Inclusion Criteria
  • Treated with a statin.
  • Fasting LDL-C > 70 mg/dL and triglyceride <=400 mg/dL.
  • High or very high risk of incurring a cardiovascular event.
Exclusion Criteria
  • Pregnant or breastfeeding females.
  • Cardiovascular or cerebrovascular event of procedures during the past 30 days.
  • Congestive heart failure NYHA class IV.
  • Poorly controlled hypertension.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PlaceboPlacebo-
Bococizumab (PF-04950615;RN316)Bococizumab (PF-04950615;RN316)-
Primary Outcome Measures
NameTimeMethod
Percent Change From Baseline in Low Density Lipoprotein-Cholesterol (LDL-C) at Week 12Baseline, Week 12
Secondary Outcome Measures
NameTimeMethod
Percent Change From Baseline in Total Cholesterol (TC) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Percent Change From Baseline in Non- High Density Lipoprotein-Cholesterol (Non HDL-C) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Percent Change From Baseline in Apolipoprotein B (ApoB) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Percent Change From Baseline in Lipoprotein(a) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Percent Change From Baseline in High Density Lipoprotein-Cholesterol (HDL-C) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Percent Change From Baseline in Fasting Low-Density Lipoprotein-Cholesterol (LDL-C) at Week 12 in Participants With Primary HyperlipidemiaBaseline, Week 12

Participants with primary hyperlipidemia are defined as participants with triglycerides (TG) level less than (\<) 200 milligram per decilitre (mg/dL) (2.26 millimoles per litre \[mmol/L\]) at pre-randomization.

Percent Change From Baseline in Fasting Low-Density Lipoprotein-Cholesterol (LDL-C) at Week 12 in Participants With Mixed DyslipidemiaBaseline, Week 12

Participants with mixed dyslipidemia are defined as TG level greater than or equal to (\>=) 200 mg/dL (2.26 mmol/L) at pre-randomization.

Percent Change From Baseline in Fasting Low Density Lipoprotein-Cholesterol (LDL-C) at Week 24 and 52Baseline, Week 24, 52
Percent Change From Baseline in Fasting Low Density Lipoprotein Cholesterol (LDL-C) at Week 24 and 52 by Triglyceride Cut-offBaseline, Week 24, 52

Percent change from baseline in fasting LDL-C among participants with TG cut-off of \<200 mg/dL and \>=200 mg/dL (2.26 mmol/L) were reported in this outcome measure.

Percent Change From Baseline in Fasting Triglyceride (TG) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Percent Change From Baseline in ApolipoproteinA-I (ApoA-I) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Percent Change From Baseline in ApolipoproteinA-II (ApoA-II) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Percent Change From Baseline in Very Low Density Lipoprotein-Cholesterol (VLDL-C) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Absolute Change From Baseline in Fasting Low Density Lipoprotein-C (LDL-C) at Week 12 by Trigylceride Cut-OffBaseline, Week 12

Absolute change from baseline among participants with TG cut-off of \<200 mg/dL and \>=200 mg/dL (2.26 mmol/L) were reported in this outcome measure.

Absolute Change From Baseline in Fasting Low Density Lipoprotein-Cholesterol (LDL-C) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Absolute Change From Baseline in Total Cholesterol (TC) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Absolute Change From Baseline in Non-High Density Lipoprotein Cholesterol (Non-HDL-C) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Absolute Change From Baseline in Apolipoprotein B (ApoB) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Absolute Change From Baseline in Lipoprotein(a) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Absolute Change From Baseline in High Density Lipoprotein-Cholesterol (HDL-C) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Absolute Change From Baseline in Ratio of Fasting Total Cholesterol to High Density Lipoprotein-Cholesterol (TC/HDL-C Ratio) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Absolute Change From Baseline in Ratio of Apolipoprotein B to ApolipoproteinA-I (ApoB/ApoA-I Ratio) at Week 12, 24 and 52Baseline, Week 12, 24, 52
Percentage of Participants Achieving Fasting Low Density Lipoprotein-Cholesterol (LDL-C) Less Than or Equal to (<=) 100 Milligram Per Deciliter (2.59 Millimoles Per Litre) at Week 12, 24 and 52Week 12, 24 and 52
Percentage of Participants Achieving Fasting Low Density Lipoprotein-Cholesterol (LDL-C) Less Than or Equal to (<=) 70 Milligram Per Deciliter (1.81 Millimoles Per Litre) at Week 12, 24 and 52Week 12, 24 and 52
Plasma PF-04950615 Concentrations at Week 12, 24 and 52Week 12, 24, 52
Number of Participants With Adverse Events (AEs) Related to Type 1 or 3 Hypersensitivity Reactions and Injection Site ReactionsBaseline up to the end of study (up to 58 weeks)

Type 1 hypersensitivity or allergic reactions were possible in response to any injected protein and included shortness of breath, urticaria, anaphylaxis and angioedema. Type 3 hypersensitivity reactions were similar to Type 1 hypersensitivity reactions but were likely to be delayed from the time of injection and included symptoms such as rash, urticaria, polyarthritis, myalgia's, polysynovitis, fever and if severe then included glomerulonephritis as well. Injection site reactions included injection site bruising, discolouration, erythema, haematoma, haemorrhage, nodule, induration, pain, pruritus and rash. Participants with type 1 or type 3 hypersensitivity reactions and participants with injection site reactions were reported in this outcome measure.

Percentage of Participants With Anti-Drug Antibodies (ADA) and Neutralizing Antibodies (nAb)Baseline up to the end of study (up to 58 weeks)

Percentage of participants with at least 1 positive ADA titer or 1 positive nAb titer were reported. Participants with their ADA titer \>=6.23 were considered to be ADA positive and participants with their nAb titer \>=1.58 were considered to be nAb positive.

Trial Locations

Locations (103)

Horizon Research Group of Opelousas, LLC

🇺🇸

Eunice, Louisiana, United States

Internal Medicine Associates

🇺🇸

Eunice, Louisiana, United States

Synexus Polska Sp. z o.o. Oddzial w Warszawie

🇵🇱

Warszawa, Poland

Centrum Medyczne AMED

🇵🇱

Warszawa, Poland

Synexus Polska Sp. z o.o. Oddzial we Wroclawiu

🇵🇱

Wroclaw, Poland

Orange County Research Center

🇺🇸

Tustin, California, United States

Soundview Medical Associates

🇺🇸

Norwalk, Connecticut, United States

Montana Medical Research Inc.

🇺🇸

Missoula, Montana, United States

Centre Hospitalier Universitaire de Sherbrooke (CHUS)

🇨🇦

Sherbrooke, Quebec, Canada

Minneapolis Heart Institute Foundation

🇺🇸

Minneapolis, Minnesota, United States

San Diego Family Care

🇺🇸

San Diego, California, United States

Providence Clinical Research

🇺🇸

North Hollywood, California, United States

Prestige Clinical Research Center Inc

🇺🇸

Miami, Florida, United States

Comunity Clinical Research Center

🇺🇸

Anderson, Indiana, United States

East Coast Institute for Research, LLC at Northeast Florida Endocrine & Diabetes Associates

🇺🇸

Jacksonville, Florida, United States

Edgewater Medical Research

🇺🇸

New Smyrna Beach, Florida, United States

Evanston Premier Healthcare Research LLC

🇺🇸

Evanston, Illinois, United States

Midwest Institute for Clinical Research

🇺🇸

Indianapolis, Indiana, United States

University of MN, Lillehei Clinical Trials Unit

🇺🇸

Minneapolis, Minnesota, United States

Rapid Medical Research, Inc.

🇺🇸

Cleveland, Ohio, United States

Clinical Trials of America, Inc.

🇺🇸

Winston Salem, North Carolina, United States

The Office of Daniel G. Williams, MD

🇺🇸

Perrysburg, Ohio, United States

Great Lakes Medical Research, LLC

🇺🇸

Willoughby, Ohio, United States

Perelman Center for Advanced Medicine Heart & Vascular Center

🇺🇸

Philadelphia, Pennsylvania, United States

Internal Medicine and Pediatric Associates of Bristol, PC

🇺🇸

Bristol, Tennessee, United States

3 rd Coast Research Associates

🇺🇸

Corpus Christi, Texas, United States

Texas Center For Drug Development, Inc.

🇺🇸

Houston, Texas, United States

Pioneer Research Solutions, Inc.

🇺🇸

Houston, Texas, United States

Protenium Clinical Research

🇺🇸

Hurst, Texas, United States

Utah Cardiology, P.C.

🇺🇸

Layton, Utah, United States

National Clinical Research - Norfolk, Inc.

🇺🇸

Norfolk, Virginia, United States

Premier Clinical Research

🇺🇸

Spokane, Washington, United States

Australian Clinical Research Network

🇦🇺

Maroubra, New South Wales, Australia

Core Research Group Pty Ltd

🇦🇺

Milton, Queensland, Australia

Dipartimento di Medicina Interna e Specialita Mediche Policlinico Umberto I

🇮🇹

Roma, RM, Italy

Lekarsky dum Ormiga

🇨🇿

Zlin, Czech Republic

MD Studies, Inc.

🇺🇸

Fountain Valley, California, United States

Southwest Heart Group

🇺🇸

Tucson, Arizona, United States

Eastern Research, Inc.

🇺🇸

Hialeah, Florida, United States

Fellows Research Alliance, Inc.

🇺🇸

Savannah, Georgia, United States

Encompass Clinical Research North Coast

🇺🇸

Encinitas, California, United States

PMG Research of Raleigh, LLC d/b/a PMG Research of Cary

🇺🇸

Cary, North Carolina, United States

Harleysville Medical Associates

🇺🇸

Harleysville, Pennsylvania, United States

Expresscare Clinical Research

🇺🇸

Colorado Springs, Colorado, United States

Alliance Research Centers

🇺🇸

Laguna Hills, California, United States

Elite Clinical Trials

🇺🇸

Wildomar, California, United States

Radiant Research, Inc

🇺🇸

Akron, Ohio, United States

Care Partners Clinical Research, LLC

🇺🇸

Jacksonville, Florida, United States

The Avenue Cardiovascular Centre

🇦🇺

St. Kilda East, Victoria, Australia

Medexa Recherche

🇨🇦

Victoriaville, Quebec, Canada

ALPHA Recherche Clinique

🇨🇦

Quebec City, Quebec, Canada

IRCCS Centro Cardiologico Fondazione Monzino

🇮🇹

Milano, MI, Italy

Integrated Medical Research, PC

🇺🇸

Ashland, Oregon, United States

Berks Cardiologists, Ltd.

🇺🇸

Wyomissing, Pennsylvania, United States

Klinische Forschung Berlin-Mitte GmbH

🇩🇪

Berlin, Germany

Beacon Clinical Research, LLC

🇺🇸

Quincy, Massachusetts, United States

SouthCoast Medical Group

🇺🇸

Savannah, Georgia, United States

Allina Health System, dba Abbott Northwestern Hospital

🇺🇸

Minneapolis, Minnesota, United States

American Health Network of Indiana, LLC

🇺🇸

Avon, Indiana, United States

Ecogene-21

🇨🇦

Chicoutimi, Quebec, Canada

Berkeley Family Practice

🇺🇸

Moncks Corner, South Carolina, United States

Montreal Heart Institute

🇨🇦

Montreal, Quebec, Canada

Diex Research Montreal Inc.

🇨🇦

Montreal, Quebec, Canada

Fakultni nemocnice Hradec Kralove

🇨🇿

Hradec Kralove, Czech Republic

Kardiologie a interni lekarstvi

🇨🇿

Praha 5, Czech Republic

IRCCS Istituto Auxologico Italiano

🇮🇹

Milano, MI, Italy

Severance Hospital, Yonsei University Health System

🇰🇷

Seoul, Korea, Republic of

Klinikum der Stadt Ludwigshafen am Rhein gGmbH

🇩🇪

Ludwigshafen, Germany

The Catholic University of Korea, Seoul St. Mary's Hospital

🇰🇷

Seoul, Korea, Republic of

IRCCS Ospedale San Raffaele

🇮🇹

Milano, MI, Italy

Ajou University Hospital

🇰🇷

Suwon, Korea, Republic of

Seoul National University Hospital

🇰🇷

Seoul, Korea, Republic of

Gangnam Sevrance Hospital, Yeonsei University Health System

🇰🇷

Seoul, Korea, Republic of

The Catholic University of Korea, Uijeongbu St. Mary's Hospital

🇰🇷

Uijeongbu-si, Gyeonggi-do, Korea, Republic of

Synexus Polska Sp. z o.o. Oddzial w Gdyni

🇵🇱

Gdynia, Poland

Niepubliczny Zaklad Opieki Zdrowotnej CEREO-MED Sp. z o.o.

🇵🇱

Lodz, Poland

Synexus Polska Sp. z o.o Oddzial w Poznaniu

🇵🇱

Poznan, Poland

Centrum Medyczne Ogrodowa Sp. z o.o.

🇵🇱

Skierniewice, Poland

Yonsei University Wonju Severance Christian Hospital

🇰🇷

Gangwon-Do, Korea, Republic of

Klinische Forschung Schwerin GmbH

🇩🇪

Schwerin, Germany

Klinische Forschung Hannover - Mitte GmbH

🇩🇪

Hannover, Germany

Ulsan University Hospital

🇰🇷

Ulsan, Korea, Republic of

Chonnam National University Hospital

🇰🇷

Gwangju, Korea, Republic of

SYNEXUS Polska Sp. z o.o. Oddzial w Katowicach

🇵🇱

Katowice, Mazowieckie, Poland

NZOZ Terapia Optima

🇵🇱

Katowice, Slaskie, Poland

Medicus w Opolu Sp z o.o.

🇵🇱

Opole, Poland

Medicome Sp. z o.o.

🇵🇱

Oswiecim, Poland

Centrum Medyczne "SOPMED" Sp. z o.o.

🇵🇱

Sopot, Poland

CSK MSW w Warszawie, Klinika Kardiologii Zachowawczej i Nadcisnienia Tetniczego

🇵🇱

Warszawa, Poland

Diagnamics, Inc.

🇺🇸

Encinitas, California, United States

St. Joseph's Medical Associates

🇺🇸

Stockton, California, United States

Prime Care Clinical Research

🇺🇸

Laguna Hills, California, United States

Clinical Research Advantage, Inc./Cassidy Medical Group - Vista

🇺🇸

Vista, California, United States

Azienda Ospedaliera Universitaria Policlinico "Paolo Giaccone"

🇮🇹

Palermo, PA, Italy

ARA-Arizona Research Associates

🇺🇸

Tucson, Arizona, United States

Achieve Clinical Research, LLC

🇺🇸

Birmingham, Alabama, United States

Cardiovascular Associates of the Southeast, LLC

🇺🇸

Birmingham, Alabama, United States

Gulfcoast Medical Research Center, LLC

🇺🇸

Tampa, Florida, United States

South Oklahoma Heart Research LLC

🇺🇸

Oklahoma City, Oklahoma, United States

Columbia Research Group, Inc.

🇺🇸

Portland, Oregon, United States

Medical Research South,LLC

🇺🇸

Charleston, South Carolina, United States

The Chinese University of Hong Kong

🇭🇰

Shatin, Hong Kong

Department of Medicine & Therapeutics-The Chinese University of Hong Kong

🇭🇰

Shatin, NT, Hong Kong

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