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Tarloxotinib

Generic Name
Tarloxotinib
Drug Type
Small Molecule
Chemical Formula
C24H24BrClN9O3
CAS Number
1636938-13-0
Unique Ingredient Identifier
H8768UL06V
Background

Tarloxotinib is under investigation in clinical trial NCT03743350 (NSCLC Exon 20 or HER2-activating Mutations).

Study of Tarloxotinib in Pts With NSCLC (EGFR Exon 20 Insertion, HER2-activating Mutations) & Other Solid Tumors With NRG1/ERBB Gene Fusions

Phase 2
Terminated
Conditions
EGFR Exon 20 Insertion Mutation
HER2-activating Mutation
ERBB Fusion
NSCLC Stage IIIB
NRG1 Fusion
NSCLC, Stage IV
NSCLC, Stage IIIC
NSCLC, Recurrent
Interventions
First Posted Date
2019-01-16
Last Posted Date
2023-06-28
Lead Sponsor
Rain Oncology Inc
Target Recruit Count
41
Registration Number
NCT03805841
Locations
🇺🇸

Pacific Shores Medical Group, Long Beach, California, United States

🇺🇸

Providence Cancer Institute, Portland, Oregon, United States

🇺🇸

University of California San Francisco, Helen Diller Cancer Center, San Francisco, California, United States

and more 6 locations

A Dose Escalation Trial of PR610 Treating Patients With Solid Tumors

Phase 1
Terminated
Conditions
Unspecified Adult Solid Tumor, Protocol Specific
Interventions
First Posted Date
2012-06-29
Last Posted Date
2014-06-16
Lead Sponsor
Proacta, Incorporated
Target Recruit Count
33
Registration Number
NCT01631279
Locations
🇳🇿

Waikato Hospital, Waikato, New Zealand

🇺🇸

University of California-Davis Comprehensive Cancer Ctr, Sacramento, California, United States

🇺🇸

Scottsdale Healthcare, Scottsdale, Arizona, United States

and more 3 locations
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