MedPath
HSA Approval

NALDEBAIN® EXTENDED RELEASE INJECTION 75MG/ML

SIN16058P

NALDEBAIN® EXTENDED RELEASE INJECTION 75MG/ML

NALDEBAIN® EXTENDED RELEASE INJECTION 75MG/ML

December 15, 2020

INTEGA PTE LTD

INTEGA PTE LTD

Regulatory Information

HSA regulatory responsibility and product classification details

Regulatory Responsibility

RegistrantINTEGA PTE LTD
Licence HolderINTEGA PTE LTD

Product Classification

D
Drug Type
Therapeutic
F
Forensic Class
Prescription Only
HSA Singapore Classification

Formulation Information

INJECTION, SOLUTION

**2 DOSAGE AND ADMINISTRATION** **2.1 General Dosing Information** Administer intramuscularly at a dose of 150 mg single dose. It is not necessary to adjust dosage based on body surface area or body weight. NALDEBAIN is an extended-release formulation, it should be taken into consideration that it takes 12~24 hours to achieve therapeutic concentration. NALDEBAIN is not adequate for administration in patients with urgent analgesics need. NALDEBAIN is fixed-dose package and only for single-dose use. Safety and effectiveness for repeat-dose use have not been established. Except for nalbuphine and ketorolac, studies of concomitant use with other drugs including general anesthetic have not been conducted. **2.2 Instructions for Use** NALDEBAIN should be administered only via the intramuscular route. Instructions for administration: 1. Clean the vial top with an alcohol swab before use. 2. Draw up 2 mL of drug into syringe. 3. After preparing the skin, inject in the upper outer quadrant of the gluteus maximus. The solution is viscous and oily. Slow injection is recommended. 4. Slightly applying pressure to the injection site to prevent drug solution leakage. 5. Do not massage the injection site.

INTRAMUSCULAR

Medical Information

**1 INDICATIONS AND USAGE** **NALDEBAIN** is indicated for the relief of moderate to severe acute postsurgical pain. _\[see Clinical studies (13)_ – _please refer to the Product Insert/Patient Information Leaflet published on HSA for the full drug information_ _\]_.

**4 CONTRAINDICATION** NALDEBAIN is for administration via the intramuscular route. It is prohibited for intravenous administration. NALDEBAIN is contraindicated in patients with: - Significant respiratory depression - Acute or severe bronchial asthma in an unmonitored setting or in the absence of resuscitative equipment - Known or suspected gastrointestinal obstruction, including paralytic ileus - Hypersensitivity to nalbuphine, sesame oil or benzyl benzoate in NALDEBAIN.

Pending

xpending

Manufacturer Information

INTEGA PTE. LTD.

Hsinchu Plant of UBI Pharma Inc.

Active Ingredients

Dinalbuphine sebacate

75mg/ ml

Dinalbuphine sebacate

Documents

Package Inserts

Naldebain Extended Release Injection PI.pdf

Approved: September 21, 2022

Download

MedPath

Empowering clinical research with data-driven insights and AI-powered tools.

© 2025 MedPath, Inc. All rights reserved.