MedPath

Glesatinib

Generic Name
Glesatinib
Drug Type
Small Molecule
Chemical Formula
C31H27F2N5O3S2
CAS Number
936694-12-1
Unique Ingredient Identifier
7Q29OXD98N
Indication

Investigated for use/treatment in cancer/tumors (unspecified).

Phase 2 Study of Glesatinib, Sitravatinib or Mocetinostat in Combination With Nivolumab in Non-Small Cell Lung Cancer

Phase 2
Terminated
Conditions
Carcinoma, Non-Small-Cell Lung
Interventions
First Posted Date
2016-11-04
Last Posted Date
2024-04-22
Lead Sponsor
Mirati Therapeutics Inc.
Target Recruit Count
161
Registration Number
NCT02954991
Locations
๐Ÿ‡บ๐Ÿ‡ธ

Yuma Regional Medical Center, Yuma, Arizona, United States

๐Ÿ‡บ๐Ÿ‡ธ

USOR - Texas Oncology - Denison Cancer Center, Denison, Texas, United States

๐Ÿ‡บ๐Ÿ‡ธ

Minnesota Oncology Hematology, P.A., Minneapolis, Minnesota, United States

and more 22 locations

Phase 2 Study of MGCD265 in Patients With Non-Small Cell Lung Cancer With Activating Genetic Alterations in MET

Phase 2
Completed
Conditions
Non-Small Cell Lung Cancer
Interventions
First Posted Date
2015-09-09
Last Posted Date
2020-03-04
Lead Sponsor
Mirati Therapeutics Inc.
Target Recruit Count
68
Registration Number
NCT02544633
Locations
๐Ÿ‡บ๐Ÿ‡ธ

Georgetown University Medical Center, Washington, District of Columbia, United States

๐Ÿ‡บ๐Ÿ‡ธ

University of California San Diego, La Jolla, California, United States

๐Ÿ‡บ๐Ÿ‡ธ

Eastern Connecticut Hematology and Oncology Associates, Norwich, Connecticut, United States

and more 90 locations

Safety Study of Two Oral Formulations of MGCD265 Administered in Healthy Subjects in the Fasting State

Phase 1
Completed
Conditions
Advanced Malignancies
Interventions
First Posted Date
2013-08-28
Last Posted Date
2015-01-08
Lead Sponsor
Mirati Therapeutics Inc.
Target Recruit Count
14
Registration Number
NCT01930006
Locations
๐Ÿ‡บ๐Ÿ‡ธ

Vince & Associates Clinical Research, Inc., Overland Park, Kansas, United States

Safety Study of Oral MGCD265 Administered Without Interruption to Subjects With Advanced Malignancies

Phase 1
Completed
Conditions
Advanced Cancer
Interventions
First Posted Date
2008-06-16
Last Posted Date
2019-02-12
Lead Sponsor
Mirati Therapeutics Inc.
Target Recruit Count
180
Registration Number
NCT00697632
Locations
๐Ÿ‡ฐ๐Ÿ‡ท

National Cancer Center, Gyeonggi-do, Korea, Republic of

๐Ÿ‡จ๐Ÿ‡ฆ

Cross Cancer Institute, Edmonton, Alberta, Canada

๐Ÿ‡จ๐Ÿ‡ฆ

British Columbia Cancer Agency, Vancouver Center, Vancouver, British Columbia, Canada

and more 16 locations

Safety Study of Oral MGCD265 Administered With Interruption to Subjects With Advanced Malignancies

Phase 1
Completed
Conditions
Advanced Malignancies
Interventions
First Posted Date
2008-05-16
Last Posted Date
2015-01-08
Lead Sponsor
Mirati Therapeutics Inc.
Target Recruit Count
47
Registration Number
NCT00679133
Locations
๐Ÿ‡บ๐Ÿ‡ธ

Karmanos Cancer Institute, Detroit, Michigan, United States

๐Ÿ‡บ๐Ÿ‡ธ

University of Texas M.D. Anderson Cancer Center, Houston, Texas, United States

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