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Pilocarpine

Generic Name
Pilocarpine
Brand Names
Betoptic Pilo, Isoptocarpine, Minims Pilocarpine Nitrate, Salagen, Vuity
Drug Type
Small Molecule
Chemical Formula
C11H16N2O2
CAS Number
92-13-7
Unique Ingredient Identifier
01MI4Q9DI3

Overview

Pilocarpine is a cholinergic muscarinic receptor agonist.

Background

Pilocarpine is a cholinergic muscarinic receptor agonist.

Indication

Pilocarpine oral tablets are indicated for the treatment of dry mouth caused by Sjogren's Syndrome or radiotherapy for cancer of the head and neck. Pilocarpine ophthalmic formulations are used to treat presbyopia in adults, reduce elevated intraocular pressure (IOP) in patients with open-angle glaucoma or ocular hypertension, manage acute angle-closure glaucoma, prevent postoperative elevated IOP associated with laser surgery, and induce miosis.

Associated Conditions

  • Acute angle-closure glaucoma
  • Dry Mouth
  • Glaucoma, Closed-Angle
  • Increased Intra Ocular Pressure (IOP)
  • Narrow-angle glaucoma
  • Ocular Hypertension
  • Open Angle Glaucoma (OAG)
  • Presbyopia
  • Chronic open-angle glaucoma

FDA Approved Products

Pilocarpine Hydrochloride
Manufacturer:Amneal Pharmaceuticals NY LLC
Route:OPHTHALMIC
Strength:20 mg in 1 mL
Approved: 2023/12/30
NDC:69238-1746
Pilocarpine Hydrochloride
Manufacturer:Bryant Ranch Prepack
Route:ORAL
Strength:5 mg in 1 1
Approved: 2023/08/30
NDC:72162-1078
Pilocarpine Hydrochloride
Manufacturer:Bryant Ranch Prepack
Route:ORAL
Strength:5 mg in 1 1
Approved: 2020/06/11
NDC:63629-8351
Pilocarpine Hydrochloride
Manufacturer:Aurobindo Pharma Limited
Route:ORAL
Strength:7.5 mg in 1 1
Approved: 2021/04/29
NDC:59651-225
Pilocarpine Hydrochloride
Manufacturer:Aurobindo Pharma Limited
Route:ORAL
Strength:5 mg in 1 1
Approved: 2021/04/29
NDC:59651-224

Singapore Approved Products

No Singapore products found for this drug

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