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Safety and Efficacy Study of Contezolid Acefosamil and Contezolid Compared to Linezolid Administered Intravenously and Orally to Adults With Moderate or Severe Diabetic Foot Infections (DFI)

Phase 3
Recruiting
Conditions
Diabetic Foot Infection
Interventions
Registration Number
NCT05369052
Lead Sponsor
MicuRx
Brief Summary

This is a Phase 3, multicenter, randomized, double-blind, safety and efficacy study of contezolid acefosamil (IV)/contezolid (PO) compared with linezolid (IV and PO) administered for a total of 14 to 28 days in adult subjects with moderate or severe DFI.

Detailed Description

Approximately 865 subjects (519 contezolid acefosamil/contezolid: 346 linezolid) will be enrolled with moderate or severe DFI that are confirmed or suspected to be due to a Gram-positive bacterial pathogen (MITT analysis set).

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
865
Inclusion Criteria
  • Have diabetes mellitus (type 1 or 2) per the American Diabetes Association criteria
  • Have a foot infection that started at or below the malleolus and does not extend above the knee
  • Foot infection that meets the IWGDF DFI criteria for classification 3 (moderate infection) or 4 (severe infection)
  • Foot infection had acute onset or worsening of signs and symptoms within the past 14 days
Exclusion Criteria
  • Previous DFI known or suspected to be caused by Gram-positive pathogens that are resistant to oxazolidinone antibiotics
  • DFI with presumptive evidence or suspicion of osteomyelitis
  • Necrotizing fasciitis, crepitant cellulitis, wet gangrene, gas gangrene, ecthyma gangrenosum, septic arthritis, or severely impaired arterial supply to any portion of the affected foot which may need revascularization before the end of the study
  • Evidence of significant hepatic, renal, hematologic, or immunologic disease
  • Females who are pregnant or breastfeeding
  • Prior receipt of any formulation of contezolid acefosamil or contezolid
  • Inability to cooperate fully with the requirements of the study protocol, including the schedule of events, or likely to be noncompliant with any study requirements, or the Investigator determines that the subject should not participate in the study

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
contezolid acefosamil/contezolidcontezolid acefosamil (IV)/contezolid (PO)-
linezolidLinezolid (IV and PO)-
Primary Outcome Measures
NameTimeMethod
Clinical response calculated with percentage of subjects with resolution of DFI signs and symptoms and requiring no further therapy as assessed by InvestigatorsDay 35

The primary objective is to evaluate the Investigator's assessment of clinical response at the D35 visit in subjects receiving contezolid acefosamil/contezolid compared to subjects receiving linezolid in the MITT analysis

Clinical laboratory assessment - complete blood count28-35 days after End-of-Therapy (EOT)

Will be evaluated under safety of contezolid acefosamil (IV)/contezolid (PO) compared with linezolid (IV and PO)

Vital signs - heart rate28-35 days after End-of-Therapy (EOT)

Will be evaluated under safety of contezolid acefosamil (IV)/contezolid (PO) compared with linezolid (IV and PO)

Adverse events - symptoms reported by subjects28-35 days after End-of-Therapy (EOT)

Evaluate safety of contezolid acefosamil (IV)/contezolid (PO) compared with linezolid (IV and PO)

Secondary Outcome Measures
NameTimeMethod
Clinical response calculated with percentage of subjects with resolution of DFI signs and symptoms and requiring no further therapy as assessed by InvestigatorsDay 10, 28-35 days after EOT

Evaluate the Investigator's assessment of clinical response at Day 10 (D10) and Late Follow-Up visits (LFU; 28-35 days after EOT) in the MITT analysis set

Trial Locations

Locations (55)

New Hope Research Development

🇺🇸

Corona, California, United States

Clemente Clinical Research

🇺🇸

Los Angeles, California, United States

VA Greater Los Angeles Healthcare System

🇺🇸

Los Angeles, California, United States

PIH Health Whittier Hospital

🇺🇸

Whittier, California, United States

University Medical and Research Center, LLC

🇺🇸

Miami, Florida, United States

Infectious Diseases Consultants of the Treasure Coast

🇺🇸

Vero Beach, Florida, United States

South Jersey Infectious Disease

🇺🇸

Somers Point, New Jersey, United States

Hospital Italiano de Buenos Aires

🇦🇷

Buenos Aires, Argentina

Sanatorio Guemes

🇦🇷

Buenos Aires, Argentina

Centro Universitario de Investigacion Clinica

🇦🇷

Corrientes, Argentina

Clinica Chutro

🇦🇷

Córdoba, Argentina

Hospital Rawson

🇦🇷

Córdoba, Argentina

Hospital San Roque

🇦🇷

Córdoba, Argentina

Instituto Medico Platense

🇦🇷

La Plata, Argentina

Centro de Investigaciones Medicas Mar Del Plata

🇦🇷

Mar Del Plata, Argentina

Hospital Ernesto Dornelles

🇧🇷

Porto Alegre, Brazil

Hospital Sao Lucas da PUCRS

🇧🇷

Porto Alegre, Brazil

Centro de Estudos e Pesquisas Em Molestias Infecciosas Ltda CPCLIN

🇧🇷

Rio Grande, Brazil

Affiliated Hospital of Yunnan University

🇨🇳

Kunming, Yunnan, China

MHAT Sveti Nikolay Chudotvorets EOOD

🇧🇬

Lom, Bulgaria

UMHAT - Sveti Georgi EAD

🇧🇬

Plovdiv, Bulgaria

Multiprofile Hospital for Active Treatment - KANEV

🇧🇬

Ruse, Bulgaria

Medical Institute Ministry of Interior Central Clinical Base

🇧🇬

Sofia, Bulgaria

University Multidisciplinary Hospital for Active Treatment and Emergency Medicine 'N. I. Priogov´

🇧🇬

Sofia, Bulgaria

UMHAT - Prof. Stoyan Kirkovich

🇧🇬

Stara Zagora, Bulgaria

Biomedica Research Group

🇨🇱

Santiago, Chile

Hospital Gustavo Fricke

🇨🇱

Viña Del Mar, Chile

The Second Affiliated Hospital of Shantou University Medical Center

🇨🇳

Shantou, Guangdong, China

The Second Affiliated Hospital of Guangxi Medical University

🇨🇳

Nanning, Guangxi, China

Union Hospital Tongji Medical College Huazhong University

🇨🇳

Wuhan, Hubei, China

The Third Xiangya Hospital of Central South University

🇨🇳

Changsha, Hunan, China

Zhongda Hospital Southeast University

🇨🇳

Nanjing, Jiangsu, China

Affiliated Hospital of Jiangsu University

🇨🇳

Zhenjiang, Jiangsu, China

Xi'an Medical University First Affiliated Hospital

🇨🇳

Xi'an, Shaanxi, China

West China Hospital Sichuan University

🇨🇳

Chengdu, Sichuan, China

West China Hospital

🇨🇳

Chengdu, Sichuan, China

Chongqing No. 4 People's Hospital

🇨🇳

Chongqing, Sichuan, China

Chu Hsien-I Memorial Hospital of Tianjin Medical University

🇨🇳

Tianjing, Tianjin, China

General Hospital Slavonski Brod

🇭🇷

Slavonski Brod, Croatia

Clinical Hospital Merkur

🇭🇷

Zagreb, Croatia

Ida-Viru Central Hospital

🇪🇪

Kohtla-Järve, Estonia

Tartu University Hospital

🇪🇪

Tartu, Estonia

South-Estonian Hospital Ltd.

🇪🇪

Võru, Estonia

LTD High Technology Hospital Med Center

🇬🇪

Batumi, Georgia

JSC Vian - West Georgia Medical Center

🇬🇪

Kutaisi, Georgia

Healthycore

🇬🇪

Tbilisi, Georgia

Tbilisi Heart Center

🇬🇪

Tbilisi, Georgia

Daugavpils Regional Hospital

🇱🇻

Daugavpils, Latvia

Riga East Clinical University Hospital

🇱🇻

Riga, Latvia

Clinical Hospital Center Zvezdara

🇷🇸

Belgrade, Serbia

Institute of Cardiovascular Diseases Dedinje

🇷🇸

Belgrade, Serbia

Univerzitna Nemocnica Bratislava

🇸🇰

Bratislava, Slovakia

Fakultna Nemocnica Trnava

🇸🇰

Trnava, Slovakia

Hospital Universitario Donostia

🇪🇸

San Sebastián, Gipuzkoa, Spain

Hospital del Mar

🇪🇸

Barcelona, Spain

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