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AGN-151586 Dose-Ranging Study for Treatment of Glabellar Lines

Phase 2
Completed
Conditions
Glabellar Lines
Interventions
Drug: Placebo
Registration Number
NCT04096326
Lead Sponsor
Allergan
Brief Summary

The purpose of this study is to evaluate the safety and efficacy of AGN-151586 over a range of doses for the treatment of moderate to severe glabellar lines (GL).

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
198
Inclusion Criteria

-Female participants willing to minimize the risk of inducing pregnancy for the duration of the clinical study and follow-up period (at least 10 weeks after study intervention).

Exclusion Criteria
  • Known immunization or hypersensitivity to any botulinum neurotoxin serotype
  • Any medical condition that may put the participant at increased risk with exposure to AGN-151586, including diagnosed myasthenia gravis, Eaton-Lambert syndrome, amyotrophic lateral sclerosis, or any other condition that might interfere with neuromuscular function
  • Marked facial asymmetry, dermatochalasis, deep dermal scarring, excessively thick sebaceous skin, or the inability to substantially lessen facial lines even by physically spreading them apart, as determined by the investigator
  • Any brow or eyelid ptosis, as determined by the investigator
  • Infection or skin disorder at the injection sites
  • History of facial nerve palsy
  • Any uncontrolled systemic disease
  • Anticipated need for treatment with botulinum neurotoxin of any serotype for any reason during the study (other than study intervention)
  • Anticipated need for surgery or overnight hospitalization during the study
  • Prior periorbital surgery, facial lift (full face or mid-face), thread lift, brow lift, or related procedures (eg, eyelid [blepharoplasty] and/or eyebrow surgery)
  • Prior facial treatment with permanent soft tissue fillers, synthetic implantation (eg, Gore-Tex®), and/or autologous fat transplantation
  • Current enrollment in an investigational drug or device study or participation in such a study within 30 days of Screening

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Cohort 1: PlaceboPlaceboParticipants received AGN-151586-matching placebo, intramuscular (IM) injections in the glabellar complex on Day 1 in Cohort 1.
Cohort 2: PlaceboPlaceboParticipants received AGN-151586-matching placebo, IM injections in the glabellar complex on Day 1 in Cohort 2.
Cohort 2: AGN-151586AGN-151586Participants received AGN-151586, IM injections in the glabellar complex on Day 1.
Cohort 3: PlaceboPlaceboParticipants received AGN-151586-matching placebo, IM injections in the glabellar complex on Day 1 in Cohort 3.
Cohort 4: PlaceboPlaceboParticipants received AGN-151586-matching placebo, IM injections in the glabellar complex on Day 1 in Cohort 4.
Cohort 5: PlaceboPlaceboParticipants received AGN-151586-matching placebo, IM injections in the glabellar complex on Day 1 in Cohort 5.
Cohort 5: AGN-151586AGN-151586Participants received AGN-151586 highest dose, IM injections in the glabellar complex on Day 1.
Cohort 1: AGN-151586AGN-151586Participants received AGN-151586 lowest dose, IM injections in the glabellar complex on Day 1.
Cohort 3: AGN-151586AGN-151586Participants received AGN-151586, IM injections in the glabellar complex on Day 1.
Cohort 4: AGN-151586AGN-151586Participants received AGN-151586, IM injections in the glabellar complex on Day 1.
Primary Outcome Measures
NameTimeMethod
Percentage of Participants With ≥ 2-grade Improvement From Baseline on the FWS According to Investigator's Assessment at Any Postintervention Timepoint Through Day 7Baseline (Day 1) through Day 7

Percentage of participants achieving a ≥ 2-grade improvement from baseline on the FWS according to investigator assessments of GL severity at maximum frown at any postintervention timepoint through Day 7 were reported. Investigators' assessments of the severity of GL at rest and maximum frown using the validated FWS was assessed using the 4-grade FWS, where 0=none, 1=mild, 2=moderate, and 3=severe. Higher scores indicate more severity. Percentages are rounded off to nearest single decimal.

Number of Participants Who Experience One or More Treatment Emergent Adverse Events (TEAEs)From first dose of study drug until the end of study (up to 42 days)

An adverse event (AE) was defined as any untoward medical occurrence in a participant or clinical study participant, temporally associated with the use of study intervention, whether considered related to the study intervention or not. TEAEs were defined as events event began on or after the date and time of the study intervention; or the adverse event was present before the date and time of the study intervention, but increased in severity or became serious on or after the date and time of the study intervention.

Number of Participants With Potentially Clinically Significant Laboratory Parameters Post InterventionFrom first dose of study drug until the end of study (up to 42 days)

Potentially clinically significant post intervention laboratory values included hematology, chemistry, and urinalysis as defined in the SAP.

Number of Participants With Potentially Clinically Significant Vital Signs Post InterventionFrom first dose of study drug until the end of study (up to 42 days)

Potentially clinically significant post intervention vital sign measurements included systolic and diastolic blood pressure, pulse rate, respiration rate, body temperature as defined in the SAP.

Number of Participants With Potentially Clinically Significant Electrocardiogram Findings Post InterventionFrom first dose of study drug until the end of study (up to 42 days)

Potentially clinically significant post intervention values in 12-lead ECG recordings included heart rate and measures PR, QRS, QT and QTcF intervals. 12-lead ECG recordings were obtained after the participants have rested for at least 10 minutes in semi-supine or supine position as defined in the SAP. A post-baseline value is considered potentially clinically significant if it meets either the observed-value or the change-from-baseline criteria such as QRS interval observed value: ≥ 150 msec; PR interval observed value: ≥ 250 msec; QTcB observed value: \> 500 msec or change from baseline value: increase of \> 60 msec; QTcF observed value: \> 500 msec or change from baseline value: increase of \> 60 msec.

Number of Participants With Anti-drug Antibodies (ADAs)Up to Day 42

Number of participants with positive anti-drug antibodies are reported. Binding and neutralizing anti-bodies are evaluated as anti-drug antibodies. Only participants with positive samples for binding antibodies have been analyzed for presence of neutralizing antibodies.

Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (9)

DermResearch Inc. /ID# 234483

🇺🇸

Austin, Texas, United States

Austin Institute for Clinical Research /ID# 237135

🇺🇸

Pflugerville, Texas, United States

Center for Dermatology Clinical Research /ID# 237798

🇺🇸

Fremont, California, United States

Wilmington Dermatology Center /ID# 237055

🇺🇸

Wilmington, North Carolina, United States

Kgl, Llc /Id# 234798

🇺🇸

Newtown Square, Pennsylvania, United States

Ava T. Shamban MD - Santa Monica. /ID# 235353

🇺🇸

Santa Monica, California, United States

Skin and Cancer Associates, LLP /ID# 236231

🇺🇸

Miami, Florida, United States

Austin Institute for Clinical Research at SBA Dermatology /ID# 236646

🇺🇸

Houston, Texas, United States

Laser and Skin Surgery Center of Indiana /ID# 236588

🇺🇸

Indianapolis, Indiana, United States

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