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Alternative Dosing Regimens in the Pharmacotherapy of Insomnia

Phase 3
Terminated
Conditions
Insomnia
Interventions
Registration Number
NCT02139098
Lead Sponsor
Philipps University Marburg Medical Center
Brief Summary

The purpose of this study is to evaluate whether drug efficiency of zolpidem and amitriptyline can be conditioned according to learning theory in patients with primary insomnia.

Detailed Description

Previous research has shown that repeated drug treatments can be regarded as conditioning processes. Sleep disorders are especially of interest to be investigated under the perspective of conditioning with drugs, since sleep quality can be defined both in terms of subjective ratings (self-rated sleep quality parameters) and objective measures (via polysomnographic assessment PSG; e.g., total sleep time, sleep onset, sleep architecture). By using two different drugs (zolpidem, amitriptyline) that modulate sleep differentially, the investigators intend to implement a conditioning paradigm in sleep disorders dissociating conditioning effects on subjective and objective sleep parameters. Both drugs should affect objective and subjective sleep parameters positively, while only amitriptyline should modulate the objectively assessed sleep architecture by REM-suppression (latency of REM-sleep onset, percentage of REM-sleep).Patients with mild to moderate insomnia will undergo a classical conditioning paradigm with one of two study medications: amitriptyline or zolpidem. After an acquisition period and a wash-out period, conditioned sleep changes are assessed in an evocation trial. During a second treatment phase of 7 days, patients receive different doses of amitriptyline (between 0mg and 50mg per night) or zolpidem (between 0mg and 5mg per night) to evaluate alternative dosing regimens in the pharmacotherapy of mild to moderate Insomnia.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
23
Inclusion Criteria
  1. age between 18 years to 69 years
  2. fluent in German language
  3. provide written informed consent
  4. ability to understand the explanations and instructions given by the study physician and the investigator
Exclusion Criteria
  1. Sleep disorders caused by medical factors (e.g. sleep apnea, restless legs syndrome, narcolepsy, substance-induced insomnia)

  2. Contraindications to study medication intake according to the information sheet for health professionals (Summary of medicinal Product Characteristics, SmPC; Fachinformation in Germany) assessed by physical examination (including ECG) and medical history

    • allergies to amitriptyline hydrochloride or any of its ingredients
    • allergies to zolpidem or any of its ingredients
    • acute intoxication with alcohol, analgetics, hypnotics or any other psychotropic drug
    • urinary retention
    • delirium
    • untreated closed-angle glaucoma
    • prostatic hyperplasia
    • pyloric stenosis
    • paralytic ilius
    • suicidal thoughts
    • liver/ kidney/ pulmonary insufficiency
    • myasthenia gravis
    • hypokalemia
    • bradycardia
    • coronary heart disease, cardiac arrhythmias, long QT syndrome or other clinically relevant cardiac disorders
    • increased risk of seizures/ history of seizures
    • substance dependence syndrome/ history of substance dependence syndrome
  3. Allergies to ingredients of placebo or novel-tasting drink (CS)

  4. currently pregnant (verified by urine pregnancy test) or lactating

  5. patients scoring ≥12 on the Epworth Sleepiness Scale

  6. patients scoring below 8 or above 21 on the Insomnia Severity Index

  7. patients suffering from a mental disorder as verified by the SCID (major depression; psychosis; brain injury; substance abuse or dependency syndrome during the last 6 months before V1)

  8. nicotine consumption > 10 cigarettes/day

  9. unwillingness to refrain from alcohol consumption throughout the study

  10. Concomitant medication interfering with study medication intake due to potential interactions (all psychotropic medication including analgetics and muscle relaxants, hypericum derivatives; antihypertensives; anti-arrhythmic agents; antibiotics; cisaprid; anti-malaria drugs; diuretics; imidazole antifungals; cumarin derivatives; antihistaminics; calcium channel blockers; medications that enlarge the QT interval or may lead to hypokalemia)

  11. change in concomitant medication regime during the last 2 weeks prior to visit 1 or after randomization

  12. intake of psychotropic medication during the last 3 months

  13. participation in any other clinical trial 3 months prior to visit 1

  14. women of childbearing age not using 2 highly effective contraceptive methods

  15. employee of the Sponsor or the principal investigator

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Amitriptyline flexible dosingPlacebo50 mg capsule amitriptyline before going to bed on 8 out of 17 nights/placebo
Zolpidem flexible dosingPlacebo5 mg capsule zolpidem before going to bed on 8 out of 17 nights/placebo
Amitriptyline flexible dosingAmitriptyline50 mg capsule amitriptyline before going to bed on 8 out of 17 nights/placebo
Amitriptyline fixed dosingAmitriptyline50 mg capsule amitriptyline before going to bed on 8 out of 17 nights
Zolpidem flexible dosingZolpidem5 mg capsule zolpidem before going to bed on 8 out of 17 nights/placebo
Zolpidem fixed dosingZolpidem5 mg capsule zolpidem before going to bed on 8 out of 17 nights
Amitriptyline continuous dosingAmitriptyline50 mg capsule amitriptyline before going to bed on 13 out of 17 nights
Primary Outcome Measures
NameTimeMethod
Objective Total Sleep TimeChange from baseline to day 10 after first medication intake

assessed by polysomnography

Objective Sleep Onset LatencyChange from baseline to day 10 after first medication intake

assessed by polysomnography

Self-reported Total Sleep TimeChange from baseline to day 10 after first medication intake

assessed by sleep diary

Self-Reported Sleep Onset LatencyChange from baseline to day 10 after first medication intake

assessed by sleep diary

Secondary Outcome Measures
NameTimeMethod
Percentage of REM sleepChange from baseline to day 10 after first medication intake

assessed by polysomnography

REM onset latencyChange from baseline to day 10 after first medication intake

assessed by polysomnography

Objective Sleep EfficiencyChange from baseline to day 17 after first medication intake

assessed by actigraphy

Objective Total Sleep TimeChange from baseline to day 17 after first medication intake

assessed by actigraphy

Self-Reported Total Sleep TimeChange from baseline to day 18 after first medication intake

assessed by sleep diary

Self-reported Sleep Onset Latency (min)Change from baseline to day 18 after first medication intake

assessed by sleep diary

Self-reported Sleep Onset Latency (evaluation)Change from baseline to day 18 after first medication intake

assessed by sleep diary

Trial Locations

Locations (1)

Clinical Psychology and Psychotherapy, Department of Psychology, Philipps University Marburg

🇩🇪

Marburg, Hessen, Germany

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