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The Study of Omalizumab (CMAB007 and Xolair) in Healthy Subjects to Compare the PK, PD and Safety

Phase 1
Completed
Conditions
Asthma
Interventions
Registration Number
NCT04778137
Lead Sponsor
Taizhou Mabtech Pharmaceutical Co.,Ltd
Brief Summary

A phase 1, randomized, double-blind, parallel group, single-dose study to compare the pharmacokinetics, pharmacodynamics and safety of two formulations of Omalizumab (CMAB007 and Xolair) in healthy subjects.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
114
Inclusion Criteria
  • Healthy subject between the ages of 18 and 45 years.
  • Subject with a body weight of ≥50 kg and ≤ 75kg and a BMI between 19.0~26.0 kg/m2 (both inclusive).
Exclusion Criteria
  • subject has a medical history and/or current presence of disease
  • subject has undergone surgery within three months before signing the informed consent;
  • Alcoholics or regular drinkers within 3 months before the test, i.e. those who drink more than 14 unites of alcohol per week (14 bottles of 360 ml beer or 630 ml spirits with 40% alcohol), or whose alcohol breath test is positive;
  • Those who have used soft drugs within 3 months prior to signing the informed consent or hard drugs within 1 year prior the trial; those who have positive drug abuse test results;
  • Those who smoke more than 10 cigarettes per day on average in the 6 months before signing the informed consent; or those who have positive nocotine results;
  • Those who have a history of drug or food allergy, or who have special allergy history (asthma, urticaria, etc.); those who have allergic rhinitis, or are known to be allergic to any component of the test drug or latex (contained in the syringe needle cover);
  • Those who drinking too much tea, coffee and/or caffeinated beverages (more than 8 cups, 1 cup =250 ml) every day;
  • Those who have received any drug treatment (including prescription drugs, over-the-counter drugs, biological products, Traditional Chinese medicine, etc.) and health care products within 4 weeks befor signing the informed consent;
  • Those who have a blood donation over 400 ml within 3 months, or 200 ml within 1 month before signing the informed consent, or plan to donate blood during the trail;
  • Those who accept any biological drugs within 3 months, or anti-IgE biological drugs within 12 months before signing the informed consent;
  • Those who plan to donate sperm within 6 months after the administration of the test drug;
  • Participants in other clinical trails within 3 months before signing the informed consent;
  • Any one of HIV antibody, HBsAg, HBeAg, HBcAg, HCV antibody and Treponerma pallidum antibody is positive;
  • The results of medical examination (ECG, X-ray, B-ultrasonic, physical and laboratory examination) are clinical significant abnormalities according to the judgment of the researcher;
  • Anti-nuclear antibody or fecal parasite test is positive;
  • Those who have undergone surgery within 1 months before signing the informed consent, or plan to undergo surgery during the trail period;

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
CMAB007Omalizumab75mg×2
XolairOmalizumab150mg
Primary Outcome Measures
NameTimeMethod
Pharmacokinetic Outcome Measures [AUC0-inf]up to day 106

Area Under the Concentration-time Curve from Time zero to infinity (AUC0-inf) of CMAB007 and Xolair in healthy subjects.

Pharmacokinetic Outcome Measures [Cmax]up to day 106

Maximum serum concentration (Cmax) of CMAB007 and Xolair in healthy subjects.

Secondary Outcome Measures
NameTimeMethod
Pharmacokinetic Outcome Measures [Apparent total body clearance (CL/F)]up to day 106

Apparent total body clearance (CL/F) of CMAB007 and Xolair in healthy subjects

Pharmacokinetic Outcome Measures [Tmax]up to day 106

Time to Cmax (Tmax) of CMAB007 and Xolair in healthy subjects

Pharmacokinetic Outcome Measures [λz]up to day 106

Terminal elimination rate constant (λz) of CMAB007 and Xolair in healthy subjects

Incidence of Treatment-Emergent Adverse Events [Safety]up to day 106

Treatment-Emergent Adverse Events (TEAEs) of CMAB007 and Xolair in healthy subjects

Pharmacokinetic Outcome Measures [AUC0-t]up to day 106

Area Under the concentration-time Curve from time zero to the last quantifiable concentration (AUC0-t) of CMAB007 and Xolair in healthy subjects.

Pharmacokinetic Outcome Measures [Vd/F]up to day 106

Apparent total distribution (Cd/F) of CMAB007 and Xolair in healthy subjects

Immunogenicityup to day 106

the Immunogenicity of CMAB007 and Xolair in healthy subjects.

Pharmacokinetic Outcome Measures [t1/2]up to day 106

Terminal half-life (t1/2) of CMAB007 and Xolair in healthy subjects

Pharmacodynamics [IgE levels]up to day 106

Free IgE and total IgE levels (the sum of free and omalizumab-bound IgE) in the serum samples from subjects

Trial Locations

Locations (1)

Shanghai Xuhui Central Hospital

🇨🇳

Shanghai, Shanghai, China

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