MedPath

Clinical Trial Nuedexta in Subjects With ALS

Phase 2
Completed
Conditions
Amyotrophic Lateral Sclerosis (ALS)
Interventions
Drug: Matching Placebo
Registration Number
NCT01806857
Lead Sponsor
Center for Neurologic Study, La Jolla, California,
Brief Summary

The purpose of this study is to determine whether Nuedexta is effective in the treatment of symptoms (impaired speech, swallowing, and saliva control)associated with Amyotrophic Lateral Sclerosis (ALS).

Detailed Description

Muscle weakness, the cardinal feature of ALS, leads to progressive loss of motor function affecting the limbs, tongue, respiratory and pharyngeal muscles. Symptomatic treatments such as the placement of a feeding tube, can compensate for the inability to swallow. Riluzole, the only approved treatment for ALS, may slow disease progression but no treatment is curative and none have improved function.

Unexpectedly, Nuedexta®, approved for the treatment of labile emotionality that occurs in association with ALS and other neurological disorders, has been observed to improve bulbar function, primarily speech and swallowing, in a number of neurological disorders, including ALS. The basis for this is conjectural but likely due to a direct effect of the drug on motor neurons in the part of the brain that controls speech and swallowing. The same part of the brain appears to modulate the expression of emotions and interestingly the site of action of the drug is the same as a site that has been implicated in a juvenile form of ALS.

This is a multicenter, randomized double-blind, placebo controlled, cross over study evaluating the palliative effect of Nuedexta® on bulbar dysfunction. It is expected that approximately 60 ALS patients from 7 clinical centers in the US will be enrolled.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
90
Inclusion Criteria
  • ALS diagnosed as possible, laboratory-supported probable, probable, or definite as defined by revised El Escorial criteria
  • Age 18 years or older
  • Exhibits bulbar dysfunction manifested by dysarthria and/or dysphagia, according to PI judgment, exhibits a score of 55 or above on the CNS-Bulbar Function Scale
  • Capable of providing informed consent and following trial procedures
  • Geographic accessibility to the site
  • Women must not be able to become pregnant for the duration of the study and must be willing to be on two contraceptive therapies
  • Slow vital capacity (SVC) measure ≥50% of predicted for gender, height, and age at the screening visit
  • Must be able to swallow capsules throughout the course of the study, according to PI judgment
  • Subjects must not have taken riluzole for at least 30 days or be on a 50mg BID dose of riluzole for at least 30 days prior to randomization (subjects how have never taken riluzole are permitted in the study)
  • Subjects taking anti-sialorrhea medication(s) must be on a stable dose for at least 30 days prior to randomization (anti-sialorrhea naïve subjects are permitted in the study)
  • Must be able to safely swallow at least 30 milliliters (mLs) of water for the water swallowing test
Exclusion Criteria
  • Prior use of Nuedexta®
  • Current use of dextromethorphan, quinidine, quinine, mefloquine or opioids
  • History of quinidine, quinine, or mefloquine-induced thrombocytopenia, hepatitis, or other hypersensitivity reactions
  • History of known sensitivity or intolerability to dextromethorphan
  • Use of an mono amine oxidase inhibitor (MAOI) or within 14 days of stopping an MAOI
  • Prolonged QT interval, congenital long QT syndrome, history suggestive of torsades de pointes, or heart failure
  • Complete atrioventricular (AV) block without implanted pacemaker, or subjects at high risk of complete AV block
  • Concomitant use with drugs that both prolong QT interval and are metabolized by cytochrome P 2D6 (CYP2D6) (i.e., thioridazine or pimozide)
  • Exposure to any other experimental agent (off-label use or investigational) within 30 days prior to Baseline Visit
  • Invasive ventilator dependence, such as tracheostomy
  • Any history of either substance abuse within the past year, unstable psychiatric disease, cognitive impairment, or dementia, according to PI judgment
  • Placement and/or usage of feeding tube
  • Pregnant women or women currently breastfeeding
  • Unable to turn diaphragm pacing device off during swallowing tests
  • Salivatory Botox within 90 days (3 months) of screening
  • Salivatory radiation within 180 days (6 months) of screening

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Nuedexta then Matching PlaceboMatching PlaceboSubjects in this arm will receive treatment with Nuedexta first for 28 days (±3 days) and then crossed over to receive treatment with matching placebo for 28 days (±3 days).
Matching Placebo then NuedextaNuedextaSubjects in this arm will receive treatment with matching placebo first for 28 days (±3 days) and then crossed over to receive treatment with Nuedexta for 28 days (±3 days).
Matching Placebo then NuedextaMatching PlaceboSubjects in this arm will receive treatment with matching placebo first for 28 days (±3 days) and then crossed over to receive treatment with Nuedexta for 28 days (±3 days).
Nuedexta then Matching PlaceboNuedextaSubjects in this arm will receive treatment with Nuedexta first for 28 days (±3 days) and then crossed over to receive treatment with matching placebo for 28 days (±3 days).
Primary Outcome Measures
NameTimeMethod
Bulbar Function Scale (CNS-BFS) Sialorrhea ScoreAverage between Screening Visit to Visit 3

The Center for Neurologic Study-Bulbar Function Scale (CNS-BFS) is a 21-item self report scale that assesses three domains of bulbar function: speech, swallowing and salivation. Scores for each question range from 1 (does not apply) to 5 (applies most of the time). The higher the score, the worse the salivation (sialorrhea). There are 7 salivation (sialorrhea) questions, with a score range of 7 to 35.

Bulbar Function Scale (CNS-BFS) Total ScoreAverage between Screening Visit to Visit 3

The Center for Neurologic Study-Bulbar Function Scale (CNS-BFS) is a 21-item self report scale that assesses three domains of bulbar function: speech, swallowing and salivation. Scores for each question range from 1 (does not apply) to 5 (applies most of the time). The higher the score, the worse the speech, swallowing and salivation (sialorrhea). \[Range of score: 21-105\]

The scale was modeled on the Center for Neurologic Study Emotional Lability Scale (CNS-LS) that has been a robust endpoint in four clinical trials. The scale was validated in a large population of ALS patients (n=122) and detects impaired bulbar function at a sensitivity of 90% and a specificity of 0.97%. Test re-test correlation was 0.92% at six-months (n=53).

Bulbar Function Scale (CNS-BFS) Speech ScoreAverage between Screening Visit to Visit 3

The Center for Neurologic Study-Bulbar Function Scale (CNS-BFS) is a 21-item self report scale that assesses three domains of bulbar function: speech, swallowing and salivation. Scores for each question range from 1 (does not apply) to 5 (applies most of the time). The higher the score, the worse the speech. There are 7 speech questions, with a score range of 7 to 35.

Bulbar Function Scale (CNS-BFS) Swallowing ScoreAverage between Screening Visit to Visit 3

The Center for Neurologic Study-Bulbar Function Scale (CNS-BFS) is a 21-item self report scale that assesses three domains of bulbar function: speech, swallowing and salivation. Scores for each question range from 1 (does not apply) to 5 (applies most of the time). The higher the score, the worse the swallowing. There are 7 swallowing questions, with a score range of 7 to 35.

Secondary Outcome Measures
NameTimeMethod
ALS Functional Rating Scale- Revised (ALSFRS-R) Total ScoreAverage between Screening Visit to Visit 3

The ALSFRS-R is a quickly administered (5 min) ordinal rating scale used to determine a subject's assessment of their capability and independence in 12 functional activities. There are 12 questions, graded by the subject 0-4 (4 is normal). Score of 0 (worst) to 48 (best). Reflects speech and swallowing, fine motor skills, large motor skills, and breathing.

Ashworth Spasticity Scale Score - Right ArmAverage between Baseline Visit to Visit 3

This is a standard measure for spasticity that has been used in numerous ALS clinical trials to assess spasticity due to upper motor neuron dysfunction in ALS. Data is generated from the clinical exam and scored from 1-5, the lowest score indicating normal tone and the highest muscle rigidity.

Visual Analog Scale - Speech ScoresAverage between Baseline Visit to Visit 3

Visual analog scales are useful for measuring complex clinical events and offer the advantage of self-administration and responsiveness to change over time. The scales designed for this study inventory three domains of bulbar function: speech, swallowing and salivation (sialorrhea). For each of these, subjects score themselves by indicating their level of function on a scale of 1 (severe impairment) to 10 (normal). Scores range from 1 to 10; the higher the score, the more normal the function.

Average Water Swallowing Test (WST)Average between Baseline Visit to Visit 3

The Water Swallowing Test (WST) estimates swallowing speed, a useful and reproducible measure. While sitting, subjects are asked to drink 30 milliliters (mL) of liquid. The time for subjects to complete this task is a sensitive measure for the detection of swallowing dysfunction and is a simple measure for serial assessment of subjects. The test will be completed three times, with the best two scores recorded to obtain an average score. Following completion of the WST, the subject's swallowing abilities (choking, spillage, and effort) will be observed.

Ashworth Spasticity Scale Score - Left LegAverage between Baseline Visit to Visit 3

This is a standard measure for spasticity that has been used in numerous ALS clinical trials to assess spasticity due to upper motor neuron dysfunction in ALS. Data is generated from the clinical exam and scored from 1-5, the lowest score indicating normal tone and the highest muscle rigidity.

Center for Neurologic Study - Lability Scale (CNS-LS) Total ScoreAverage between Screening Visit to Visit 3

The Center for Neurologic Study-Lability Scale (CNS-LS) is a 7-item self report scale that assesses pseudobulbar affect (PBA) by measuring the perceived frequency of PBA episodes (laughing or crying). Each item is scored using a 5-point Likert scale, from 1 (applies never) to 5 (applies most of the time). Scores range from 5-35. The higher the score, the worse the PBA.

Timed Reading of Test Paragraph ResultAverage between Baseline Visit to Visit 3

Subjects will be asked to read 'The Rainbow Passage' a commonly used test paragraph utilized by speech pathologists to assess speech rate (words/minute). Study staff will time the subject to determine how many words the subject reads per minute. It is used primarily because it contains every sound in the English language. Subjects will also be observed for loudness, nasality, and intelligibility.

Average Solids Swallowing TestAverage between Baseline Visit to Visit 3

The Time Swallowing Test assesses the subject's ability to swallow solids. For this test, the subject will be asked to consume a tablespoon of cereal containing 5 cheerios. The subject will be instructed to close their mouth, chew and subsequently swallow the bolus. The time to complete this task will be recorded. The test will be completed three times to obtain an average score.

Ashworth Spasticity Scale Score - Right LegAverage between Baseline Visit to Visit 3

This is a standard measure for spasticity that has been used in numerous ALS clinical trials to assess spasticity due to upper motor neuron dysfunction in ALS. Data is generated from the clinical exam and scored from 1-5, the lowest score indicating normal tone and the highest muscle rigidity.

Visual Analog Scale - Swallowing ScoreAverage between Baseline Visit to Visit 3

Visual analog scales are useful for measuring complex clinical events and offer the advantage of self-administration and responsiveness to change over time. The scales designed for this study inventory three domains of bulbar function: speech, swallowing and salivation (sialorrhea). For each of these, subjects score themselves by indicating their level of function on a scale of 1 (severe impairment) to 10 (normal). Scores range from 1 to 10; the higher the score, the more normal the function.

Visual Analog Scale - Salivation (Sialorrhea) ScoreAverage between Baseline Visit to Visit 3

Visual analog scales are useful for measuring complex clinical events and offer the advantage of self-administration and responsiveness to change over time. The scales designed for this study inventory three domains of bulbar function: speech, swallowing and salivation (sialorrhea). For each of these, subjects score themselves by indicating their level of function on a scale of 1 (severe impairment) to 10 (normal). Scores range from 1 to 10; the higher the score, the more normal the function.

Ashworth Spasticity Scale Score - Left ArmAverage between Baseline Visit to Visit 3

This is a standard measure for spasticity that has been used in numerous ALS clinical trials to assess spasticity due to upper motor neuron dysfunction in ALS. Data is generated from the clinical exam and scored from 1-5, the lowest score indicating normal tone and the highest muscle rigidity.

Trial Locations

Locations (7)

Neurology Associates, P.C.

🇺🇸

Lincoln, Nebraska, United States

California Pacific Medical Center

🇺🇸

San Francisco, California, United States

The Cleveland Clinic

🇺🇸

Cleveland, Ohio, United States

Hennepin County Medical Center

🇺🇸

Minneapolis, Minnesota, United States

Georgetown University Medical Center

🇺🇸

Washington D.C., District of Columbia, United States

Saint Mary's Health Care

🇺🇸

Grand Rapids, Michigan, United States

Providence ALS Center

🇺🇸

Portland, Oregon, United States

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