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A Study to Evaluate MEDI5752 in Subjects With Advanced Solid Tumors

Phase 1
Active, not recruiting
Conditions
Selected Advanced Solid Tumors
Interventions
Biological: MEDI5752
Biological: Pembrolizumab
Registration Number
NCT03530397
Lead Sponsor
MedImmune LLC
Brief Summary

The purpose of this study is to evaluate MEDI5752 and carboplatin and pemetrexed or paclitaxel or nab-paclitaxel in adult subjects with advanced solid tumors, when administered as a single agent or combined with chemotherapy.

Detailed Description

This is a phase 1, first-time-in-human, multicenter, open-label, dose-escalation and dose-expansion study to evaluate the safety and tolerability, and efficacy, pharmacokinetics and Immunogenicity of MEDI5752 and carboplatin and pemetrexed or paclitaxel or nab-paclitaxel in adult subjects with advanced solid tumors, when administered as a single agent or combined with chemotherapy.

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
All
Target Recruitment
401
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Arm A: MEDI5752MEDI5752MEDI5752
Arm B: MEDI5752 and chemotherapyPaclitaxel or Nab-PaclitaxelMEDI5752, pemetrexed, carboplatin and paclitaxel.
Arm B: MEDI5752 and chemotherapyMEDI5752MEDI5752, pemetrexed, carboplatin and paclitaxel.
Arm B: MEDI5752 and chemotherapyPemetrexedMEDI5752, pemetrexed, carboplatin and paclitaxel.
Arm C: Pembrolizumab and chemotherapyPembrolizumabpembrolizumab, pemetrexed, and carboplatin
Arm B: MEDI5752 and chemotherapyCarboplatinMEDI5752, pemetrexed, carboplatin and paclitaxel.
Arm C: Pembrolizumab and chemotherapyCarboplatinpembrolizumab, pemetrexed, and carboplatin
Arm C: Pembrolizumab and chemotherapyPemetrexedpembrolizumab, pemetrexed, and carboplatin
Primary Outcome Measures
NameTimeMethod
Preliminary anti-tumor activitiy of MEDI5752 (versus pembrolizumab, where applicable) using Objective Response based on RECIST v1.1 (Dose-expansion phase)From the first dose of study drug through the date of first documented progression, end of study, date of death, or two years after the last patient starts treatment, whichever should occur first

The primary endpoint of antitumor activity include Objective Response and will be based on all post baseline disease assessments that occur prior to initiation of subsequent anticancer therapy.

The number of subjects experiencing abnormal laboratory evaluations (Dose-escalation phase)From the time of informed consent through 114 days following termination of treatment with investigational product

The primary endpoint is as assessed as the number of subjects experiencing changes in laboratory parameters from baseline.

The number of subjects experiencing dose-limiting toxicities (DLTs) (Dose-escalation phase)Up to 21 days following the first dose

The primary endpoint is as assessed by the number of subjects experiencing dose limiting toxicities (DLTs) as defined by the protocol.

The number of subjects experiencing treatment related adverse events (AEs) (Dose-escalation phase)From the time of informed consent through 114 days following termination of treatment with investigational product

The primary endpoint is as assessed by the number of subjects experiencing adverse events (AEs) graded per NCI CTCAE v4.03

The number of subjects experiencing abnormal electrocardiograms (ECG) reported as Adverse Events (Dose-escalation phase)From the time of informed consent through 114 days following termination of treatment with investigational product

The primary endpoint is as assessed by the the number of subjects experiencing clinically significant changes in ECG parameters from baseline.

The number of subjects experiencing changes from baseline in vital signs reported as adverse events (Dose-escalation phase)From the time of informed consent through 114 days following termination of treatment with investigational product

The primary endpoint is as assessed by the number of subjects experiencing clinically significant changes in vital signs from baseline.

The number of subjects experiencing treatment related serious adverse events (SAEs) (Dose-escalation phase)From the time of informed consent through 114 days following termination of treatment with investigational product

The primary endpoint is as assessed by the number of subjects with serious adverse events (SAEs) graded per NCI CTCAE v4.03.

Secondary Outcome Measures
NameTimeMethod
Ability of MEDI5752 to generate immune response in subjects with advanced solid tumorsTo be assessed at Day 1, 8, 15, 22, 29, 43, 64, 85, and 106 over the first 4 months of treatment and up to 114 days following end of treatment.

The endpoints for the immunogenicity of MEDI5752 include the number of subjects who develop detectable anti-drug antibodies (ADAs)

Preliminary Antitumor Activity: Progression Free SurvivalFrom the first dose of study drug through the date of first documented progression, end of study, date of death, or two years after last subject starts treatment whichever should occur first

The endpoints for assessment of antitumor activity include progression free survival (PFS) and is defined as the duration measured from the start of treatment with investigational product to the first documentation of disease progression or death due to any cause.

The number of subjects experiencing abnormal laboratory evaluations (Dose-expansion phase)From the time of informed consent through 114 days following termination of treatment with investigational product

The secondary endpoint is as assessed by the number of subjects experiencing changes in laboratory parameters from baseline.

Pharmacokinetics of MEDI5752: AUCTo be assessed at Day 1, 2, 3, 8, 15, 22, 29, 43, 64, 85, and 106 over the first 4 months of treatment and up to 114 days following end of treatment

The endpoints for the assessment of PK of MEDI5752 include individual MEDI5752 concentrations at different time points after administration. PK parameters that may be modeled on this data include area under the concentration-time curve (AUC)

Preliminary Antitumor Activity: Disease ControlFrom the first dose of study drug through the date of first documented progression, end of study, date of death, or two years after last subject starts treatment whichever should occur first

The endpoints for assessment of antitumor activity include disease control (DC) and is defined as CR, PR, or SD according to RECIST v1.1.

The number of subjects experiencing treatment related adverse events (AEs) (Dose-expansion phase)From the time of informed consent through 114 days following termination of treatment with investigational product

The secondary endpoint is as assessed by the number of subjects experiencing adverse events (AEs) graded per NCI CTCAE v4.03

The number of subjects experiencing Changes from baseline in vital signs reported as adverse events (Dose-expansion phase)From the time of informed consent through 114 days following termination of treatment with investigational product

The secondary endpoint is as assessed by the number of subjects experiencing clinically significant changes in vital signs from baseline.

Pharmacokinetics of MEDI5752: CmaxTo be assessed at Day 1, 2, 3, 8, 15, 22, 29, 43, 64, 85, and 106 over the first 4 months of treatment and up to 114 days following end of treatment

The endpoints for the assessment of PK of MEDI5752 include individual MEDI5752 concentrations at different time points after administration. PK parameters that may be modeled on this data include maximum observed concentration (Cmax)

The number of subjects experiencing treatment related serious adverse events (SAEs) (Dose-expansion phase)From the time of informed consent through 114 days following termination of treatment with investigational product

The secondary endpoint is as assessed by the number of subjects with serious adverse events (SAEs) graded per NCI CTCAE v4.03

Pharmacokinetics of MEDI5752: ClearanceTo be assessed at Day 1, 2, 3, 8, 15, 22, 29, 43, 64, 85, and 106 over the first 4 months of treatment and up to 114 days following end of treatment

The endpoints for the assessment of PK of MEDI5752 include individual MEDI5752 concentrations at different time points after administration. PK parameters that may be modeled on this data include clearance (CL)

Pharmacokinetics of MEDI5752: t 1/2To be assessed at Day 1, 2, 3, 8, 15, 22, 29, 43, 64, 85, and 106 over the first 4 months of treatment and up to 114 days following end of treatment.

The endpoints for the assessment of PK of MEDI5752 include individual MEDI5752 concentrations at different time points after administration. PK parameters that may be modeled on this data include terminal phase half life (t 1/2)

PD-L1 Expression in subjects with advanced solid tumorsTo be assessed at baseline

The endpoint for the PD-L1 expression will be determined by Immunohistochemistry characterization.

Preliminary Antitumor Activity: Duration of ResponseFrom the date of response through the date of first documented progression, end of study, date of death, or two years after last subject starts treatment whichever should occur first

The endpoints for assessment of antitumor activity include duration of response (DoR) and is defined as the duration from the documentation of OR to the first documentation of disease progression or death due to any cause.

Preliminary Antitumor Activity: Overall SurvivalFrom the first dose of study drug through the end of study, or date of death, or two years after last subject starts treatment whichever should occur first

The endpoints for assessment of antitumor activity include overall survival (OS) and is defined as the duration measured from the start of treatment with investigational product until death due to any cause.

The number of subjects experiencing abnormal ECGs reported as adverse events (Dose-expansion phase)From the time of informed consent through 14 days following termination of treatment with investigational product

The secondary endpoint is as assessed by the number of subjects experiencing clinically significant changes in ECG parameters from baseline.

Trial Locations

Locations (1)

Research Site

🇨🇳

Taipei, Taiwan

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