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A Study of Paclitaxel With GDC-0941 Versus Paclitaxel With Placebo in Participants With Locally Recurrent or Metastatic Breast Cancer

Phase 2
Completed
Conditions
Breast Cancer
Interventions
Registration Number
NCT01740336
Lead Sponsor
Genentech, Inc.
Brief Summary

This multicenter, randomized, single-blind, placebo-controlled, two arm study will evaluate the efficacy and safety of paclitaxel with GDC-0941 versus paclitaxel with placebo in participants with locally recurrent or metastatic breast cancer.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Female
Target Recruitment
183
Inclusion Criteria
  • Histologically or cytologically confirmed adenocarcinoma of the breast, with measurable or non-measurable locally recurrent or metastatic disease
  • Human epidermal growth factor receptor 2 (HER2)-negative and hormone receptor (HR) (estrogen receptor and/or progesterone receptor)-positive disease as defined by local guidelines
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1
  • Adequate hematologic and end organ function
  • Women of childbearing potential must agree to remain abstinent or to use two adequate methods of contraception, including at least one method with a failure rate of less than (<) 1 percent (%) per year, during the treatment period and for at least 30 days after the last dose of study treatment or 6 months after discontinuation of paclitaxel, whichever is longer
Exclusion Criteria
  • Prior non-capecitabine chemotherapy for locally recurrent or metastatic disease
  • Prior treatment with a phosphoinositide 3-kinase (PI3K) inhibitor for advanced or metastatic breast cancer
  • History of intolerance to a taxane-containing therapy
  • History of clinically significant cardiac or pulmonary dysfunction
  • History of malabsorption syndrome or other condition that would interfere with enteral absorption
  • Clinically significant history of liver disease
  • Active autoimmune disease or active inflammatory disease
  • Immunocompromised status due to current known active infection with human immunodeficiency virus (HIV) or due to the use of immunosuppressive therapies for other conditions
  • Need for current chronic corticosteroid therapy
  • Pregnant, lactating, or breastfeeding women
  • Current severe, uncontrolled systemic disease
  • Known untreated or active central nervous system (CNS) metastases

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
B: Paclitaxel, PlaceboPlaceboParticipants will receive placebo matching to GDC-0941 on the 5/7-day schedule along with 90 mg/m\^2 IV weekly for 3 out of 4 weeks in every 28-day cycle.
A: Paclitaxel, GDC-0941GDC-0941Participants will receive GDC-091 260 milligrams (mg) orally in repeated rounds of once daily (QD) dosing for 5 consecutive days followed by 2 consecutive days during which GDC-0941 will not be administered (5/7-day schedule). This 5/7-day schedule will be repeated weekly in each 28-day cycle until disease progression or intolerable toxicity. Participants will receive 90 milligrams per square meter (mg/m\^2) intravenously (IV) weekly for 3 out of 4 weeks in every 28-day cycle.
A: Paclitaxel, GDC-0941PaclitaxelParticipants will receive GDC-091 260 milligrams (mg) orally in repeated rounds of once daily (QD) dosing for 5 consecutive days followed by 2 consecutive days during which GDC-0941 will not be administered (5/7-day schedule). This 5/7-day schedule will be repeated weekly in each 28-day cycle until disease progression or intolerable toxicity. Participants will receive 90 milligrams per square meter (mg/m\^2) intravenously (IV) weekly for 3 out of 4 weeks in every 28-day cycle.
B: Paclitaxel, PlaceboPaclitaxelParticipants will receive placebo matching to GDC-0941 on the 5/7-day schedule along with 90 mg/m\^2 IV weekly for 3 out of 4 weeks in every 28-day cycle.
Primary Outcome Measures
NameTimeMethod
Progression-Free Survival (PFS) Assessed as per Modified Response Evaluation Criteria in Solid Tumors (RECIST) Version 1.1 (v1.1)From the time of randomization until disease progression or death from any cause (up to approximately 3 years)
Secondary Outcome Measures
NameTimeMethod
Population PK for PaclitaxelDay 1 of Cycle 1 (cycle length=28 days)
Duration of Confirmed Objective Response Assessed as per Modified RECIST v1.1From first observation of an objective tumor response until disease progression (up to approximately 3 years)
Percentage of Participants With Adverse EventsFrom randomization up to approximately 3 years
Percentage of Participants With Objective Tumor Response Assessed as per Modified RECIST v1.1From first observation of an objective tumor response until disease progression (up to approximately 3 years)
Percentage of Participants Acheiving Clinical Benefit (Partial Response, Complete Response or Stable Disease Lasting for at Least 6 Months) Assessed as per Modified RECIST v1.1From randomization until disease progression (up to approximately 3 years)
Population Pharmacokinetics (PK) for GDC-0941Day 8 of Cycle 1 and Day 1 of Cycle 6 (cycle length=28 days)

Trial Locations

Locations (97)

Pacific Cancer Medical Center

🇺🇸

Anaheim, California, United States

Helen & Harry Gray Cancer Center-Hartford Hospital-CCD PRIME; Research

🇺🇸

Hartford, Connecticut, United States

Oncology Specialists, S.C.

🇺🇸

Park Ridge, Illinois, United States

Royal Prince Alfred Hospital

🇦🇺

Camperdown, New South Wales, Australia

Puget Sound Cancer Centers

🇺🇸

Edmonds, Washington, United States

TriHealth Oncology Institute

🇺🇸

Cincinnati, Ohio, United States

Clinique Ste-Elisabeth

🇧🇪

Namur, Belgium

Masarykuv onkologicky ustav

🇨🇿

Brno, Czechia

Kaiser Permanente - San Francisco (2238 Geary)

🇺🇸

San Francisco, California, United States

Klinikum Wels-Grieskirchen

🇦🇹

Wels, Austria

Krankenhaus Hietzing m.Neurolog. Zentrum Rosenhuegel

🇦🇹

Wien, Austria

Arizona Oncology Associates, PC - NAHOA

🇺🇸

Sedona, Arizona, United States

Summa Health System

🇺🇸

Akron, Ohio, United States

Border Medical Oncology

🇦🇺

Wodonga, New South Wales, Australia

Shivers Cancer Center at University Medical Center Brackenridge

🇺🇸

Austin, Texas, United States

Aultman Hospital; Aultman Hospital Cancer Center

🇺🇸

Canton, Ohio, United States

Cancer Specialists of North Florida

🇺🇸

Orange Park, Florida, United States

Texas Oncology

🇺🇸

Bedford, Texas, United States

Mater Adult Hospital

🇦🇺

Mackay, Queensland, Australia

Bendigo Hospital; Oncology

🇦🇺

Bendigo, Victoria, Australia

Shenandoah Oncology Associates

🇺🇸

Winchester, Virginia, United States

Kaiser Permanente - South San Francisco

🇺🇸

South San Francisco, California, United States

ProHEALTH Care Associates LLP

🇺🇸

Lake Success, New York, United States

Texas Oncology, P.A. - El Paso; West

🇺🇸

El Paso, Texas, United States

UZ Antwerpen

🇧🇪

Edegem, Belgium

Swedish Health Services

🇺🇸

Seattle, Washington, United States

Institut Catala d Oncologia Hospital Duran i Reynals

🇪🇸

Barcelona, Spain

Texas Oncology - Memorial City

🇺🇸

Houston, Texas, United States

Hematology and Oncology Associates of Sc

🇺🇸

Greenville, South Carolina, United States

Fakultni nemocnice Brno

🇨🇿

Brno, Czechia

Bay Area Cancer Research Group, LLC

🇺🇸

Pleasant Hill, California, United States

Ashford Cancer Center Research

🇦🇺

Kurralta Park, South Australia, Australia

Port Macquarie Base Hospital;North Coast Cancer Institute

🇦🇺

Port Macquarie, New South Wales, Australia

Krajska nemocnice Liberec a.s.

🇨🇿

Liberec, Czechia

Royal Hobart Hospital

🇦🇺

Hobart, Tasmania, Australia

Abington Memorial Hospital

🇺🇸

Abington, Pennsylvania, United States

Peninsula and South Eastern Haematology and Oncology Grou

🇦🇺

Frankston, Victoria, Australia

Lkh-Univ. Klinikum Graz

🇦🇹

Graz, Austria

UZ Leuven Gasthuisberg

🇧🇪

Leuven, Belgium

Henry Ford Health System

🇺🇸

Detroit, Michigan, United States

Concord Repatriation General Hospital

🇦🇺

Concord, New South Wales, Australia

Nemocnice Na Bulovce

🇨🇿

Prague, Czechia

Vseobecna fakultni nemocnice v Praze

🇨🇿

Praha 2, Czechia

Royal Cornwall Hospital

🇬🇧

Truro, United Kingdom

New Cross Hospital

🇬🇧

Wolverhampton, United Kingdom

The Christie

🇬🇧

Manchester, United Kingdom

Leicester Royal Infirmary

🇬🇧

Leicester, United Kingdom

Freeman Hospital

🇬🇧

Newcastle upon Tyne, United Kingdom

Nottingham University Hospitals City Campus

🇬🇧

Nottingham, United Kingdom

Royal Stoke University Hospital

🇬🇧

Stoke on Trent, United Kingdom

Northern Utah Associates

🇺🇸

Ogden, Utah, United States

Thomayerova nemocnice

🇨🇿

Praha 4 - Krc, Czechia

Royal Brisbane and Women's Hospital

🇦🇺

Herston, Queensland, Australia

Sydney Haematology & Oncology Clinic

🇦🇺

Wahroonga, New South Wales, Australia

California Cancer Associates for Research & Excellence, Inc.

🇺🇸

Encinitas, California, United States

Kaiser Permanente - Hayward

🇺🇸

Hayward, California, United States

Kaiser Permanente - San Jose

🇺🇸

San Jose, California, United States

Kaiser Permanente - Santa Clara

🇺🇸

Santa Clara, California, United States

Kaiser Permanente - Vallejo

🇺🇸

Vallejo, California, United States

Clinical Research of South Florida

🇺🇸

Coral Gables, Florida, United States

Phoebe Putney Memorial Hospital

🇺🇸

Albany, Georgia, United States

Joliet Oncology-Hematology; Associates, Ltd.

🇺🇸

Joliet, Illinois, United States

Cotton-O'Neil Clinical Research Center, Hematology and Oncology; Cotton O'Neil Cancer Center

🇺🇸

Topeka, Kansas, United States

Hematology Oncology Clinic

🇺🇸

Baton Rouge, Louisiana, United States

Billings Clinic Cancer Center-CCD PRIME

🇺🇸

Billings, Missouri, United States

Texas Oncology, P.A. ;Sherman Cancer Center

🇺🇸

Sherman, Texas, United States

Multiscan s.r.o.

🇨🇿

Pardubice, Czechia

Royal Perth Hospital; Medical Oncology

🇦🇺

Perth, Western Australia, Australia

Chungbuk National University Hospital

🇰🇷

Cheongju-si, Korea, Republic of

Seoul National University Hospital

🇰🇷

Seoul, Korea, Republic of

Samsung Medical Center

🇰🇷

Seoul, Korea, Republic of

Institut Catala d´Oncologia Hospital Germans Trias i Pujol

🇪🇸

Badalona, Barcelona, Spain

Asan Medical Center

🇰🇷

Seoul, Korea, Republic of

Hospital General Univ. Gregorio Maranon

🇪🇸

Madrid, Spain

Complejo Hospitalario de Jaen

🇪🇸

Jaen, Spain

Royal Sussex County Hospital

🇬🇧

Brighton, United Kingdom

Royal Surrey County Hospital

🇬🇧

Guildford, United Kingdom

Kaiser Permanente - Oakland

🇺🇸

Oakland, California, United States

Kaiser Permanente Medical Center - Roseville

🇺🇸

Roseville, California, United States

Kaiser Permanente Sacramento Medical Center

🇺🇸

Sacramento, California, United States

Nebraska Cancer Specialists; Oncology Hematology West, PC

🇺🇸

Omaha, Nebraska, United States

University of California at San Francisco

🇺🇸

San Francisco, California, United States

Kaiser Permanente - Walnut Creek

🇺🇸

Walnut Creek, California, United States

Illinois Cancer Care

🇺🇸

Peoria, Illinois, United States

Hematology - Oncology Associates of Treasure Coast

🇺🇸

Port Saint Lucie, Florida, United States

Calvary Mater Newcastle; Medical Oncology

🇦🇺

Waratah, New South Wales, Australia

Dana Farber Cancer Institute

🇺🇸

Boston, Massachusetts, United States

Metairie Oncologist, LLC

🇺🇸

Metairie, Louisiana, United States

Severance Hospital, Yonsei University Health System

🇰🇷

Seoul, Korea, Republic of

Maine Research Associates

🇺🇸

Auburn, Maine, United States

Beth Israel Deaconess Med Ctr

🇺🇸

Brookline, Massachusetts, United States

START Madrid. Centro Integral Oncologico Clara Campal; CIOCC

🇪🇸

Madrid, Spain

Barts Hospital

🇬🇧

London, United Kingdom

LKH - Universitätsklinikum der PMU Salzburg

🇦🇹

Salzburg, Austria

Sint Augustinus Wilrijk

🇧🇪

Wilrijk, Belgium

CHU Ambroise Paré

🇧🇪

Mons, Belgium

Institut Jules Bordet

🇧🇪

Brussels, Belgium

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