MedPath

Low Dose Exemestane Vs Low Dose Tamoxifen in Post-menopausal Women At High Risk for Breast Cancer.

Phase 2
Not yet recruiting
Conditions
Breast Cancer
Interventions
Registration Number
NCT06364267
Lead Sponsor
Andrea DeCensi
Brief Summary

The purpose of the study is to to compare low dose of exemestane (babyexe) versus low dose of tamoxifen (babytam) in terms of change of quality of life from baseline to 12 months.

Detailed Description

This is a multicenter, randomized, double blind phase II trial.

Eligible patients will be randomized in a 1:1 ratio to:

ARM 1: BabyEXE Arm, 25 mg eod, typically every odd day of the monthly calendar for 12 monthsor unless progression, SAE, medical decision, patient withdrawal occur.

ARM 2: BabyTAM Arm, 10 mg eod, typically every odd day of the monthly calendar for 12 months or unless progression, SAE, medical decision, patient withdrawal occur.

Blinding will be guaranteed by over-encapsulation of active tablet agents with an AA capsule in a 6-month bottle.

In both arms, treatment should begin within 30 days from randomization. Exemstane and Tamoxifen will be provided for free by the Study Sponsor.

After study completion, participants will be unblinded and treated according to local guidelines. Clinical visit will be performed every 6 months (±14 days) with physical examination vital signs and weight and girth measurement, ECOG PS, MENQOL questionnaire (0, 6, 12 months), review of self-reported compliance, concomitant medications, AEs assessment, and physical exam. Telephone/video contact may be allowed at 3 and 9 months, whereas baseline, 6 months and 12 months visits are necessary for blood collection and biomarker assessment. Blood serum for centralized storage at IEO, Milan, Italy, will be collected at different time points.

Recruitment & Eligibility

Status
NOT_YET_RECRUITING
Sex
Female
Target Recruitment
140
Inclusion Criteria
  1. Postmenopausal state is defined as no menses for 12 months without an alternative medical cause. A high follicle stimulating hormone (FSH) level in the postmenopausal range may be used to confirm a post- menopausal state in women not using hormonal contraception or hormonal replacement therapy. However, in the absence of 12 months of amenorrhea, a single FSH measurement is insufficient. Permanent sterilization methods include hysterectomy, bilateral salpingectomy and bilateral oophorectomy.

    Any of the following criteria must be met:

    1. Recent (within 12 months from date of consent form signature) histologic diagnosis of ER+ve (>5%) DCIS (patients with DCIS should have undergone breast-conserving therapy i.e. lumpectomy to remove the tumor with negative surgical margins followed by radiotherapy) or diagnosis within 3 years of HRL (ADH, LCIS, ALH), or:
    2. At least 3% breast cancer risk at 5 years (or 5% risk at 10yrs) per one of the following risk models: the Breast Cancer Surveillance Consortium risk calculator V3 or Tyrer-Cuzick model V8 or:
    3. Known carriers of a germline pathogenic/likely pathogenetic variant in the following moderate penetrance genes (CHEK2 or ATM), or women with chest wall irradiation before age of 30 years.
  2. Eastern Cooperative Oncology Group - Performance Status (ECOG-PS) 0-1.

  3. Able to swallow oral medications.

  4. Participants with a prior or concurrent malignancy whose natural history or treatment does not have the potential to interfere with the safety or efficacy assessment of the investigational regimen are eligible for this trial. Specifically, all cancers diagnosed since 3 years or longer except for breast and endometrial are eligible.

  5. Ability to understand and the willingness to sign a written informed consent document.

  6. Mammography performed up to 6 months before the trial consent form signature.

  7. DEXA performed up to 12 months before the trial consent form signature.

  8. Patients with life expectancy ≥ 10 years.

  9. Patients with normal liver function tests and blood cell count.

  10. Negative gynaecological examination performed up to 6 months before the trial consent form signature.

Exclusion Criteria
  1. Pre/perimenopausal women
  2. History of DVT or PE.
  3. Endometrial cancer.
  4. Macular disorders.
  5. Inability to comply with study procedures.
  6. Prior use of antiestrogens within 12 months from the date of the trial consent form signature.
  7. Use of hormone replacement therapy (HRT) within 3 months from the date of the trial consent form signature.
  8. Severe osteoporosis (T score ≤ 2.5 at either spine or hip), or recent vertebral fracture (within 6 months) not treated with zolendronic acid or denosumab.
  9. Use of terbinafine, quinidine, cinacalcet, rifampicin, phenytonin, carbamazepine, phenobarbital, and St. John's wort, warfarin, erythromycin, cyclosporin, nifepidine and any concomitant coumarin-type anticoagulant therapy.
  10. Patients with moderate or severe renal impairment.
  11. Patients with a known hypersensitivity to study drugs.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
ARM 1Exemestane 25 MGBabyEXE Arm, 25 mg eod, typically every odd day of the monthly calendar for 12 months.
ARM 2Tamoxifen 10 MGBabyTAM Arm, 10 mg eod, typically every odd day of the monthly calendar for 12 months
Primary Outcome Measures
NameTimeMethod
Quality of life MEnQol12 months

The primary endpoint is the difference between arms in the score of overall domain of MENQOL after 12 months of treatment.

Secondary Outcome Measures
NameTimeMethod
Sex hormones6 months

The difference in sex hormones (free estradiol: estradiol/SHBG) and IGF system (IGF-I, IGFBP-3 and their ratio) after 6 months, as surrogate endpoint biomarkers.

MenQol score domain6 months

The difference between arms in the overall MENQOL score domain after 6 months of treatment.

Other domains of MenQol6 and 12 months

The difference between arms individual domains of MENQOL (physical, sexual, psychosocial, vasomotor) at 6 and 12 months

Safety profile6 and 12 months

The difference between arms of safety profile according to CTCAE v.5 at 6 and 12 months.

PMAS6 and 12 months

The difference between arms at 6 and 12 months in PMAS, Promise Medication Adherence Scale, a validated tool to measure pill adherence.

BPI6 and 12 months

The difference between arms on BPI Brief Pain Inventory at 6 and 12 months.

Bone biomarker6 and 12 months

The difference between arms in C-telopetide at 6 and 12 months

Customer satisfatcionScreening

Patient uptake at screening/baseline phase will be measured with a questionnaire including factors related to breast cancer worry and presence of life style risk factors, and participant satisfaction for study explanation.

Exemestane toxicity12 months

Toxicity of babyexe in comparison with full dose historical controls treated in the adjuvant setting will also be evaluated

Trial Locations

Locations (1)

E.O. Ospedali Galliera

🇮🇹

Genova, Italy

© Copyright 2025. All Rights Reserved by MedPath