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Effect of Rifampin on the Pharmacokinetics of Dapagliflozin in Healthy Subjects

Phase 1
Terminated
Conditions
Type 2 Diabetes Mellitus
Interventions
Registration Number
NCT01068756
Lead Sponsor
AstraZeneca
Brief Summary

The purpose of the study is to assess the effects of rifampin on the pharmacokinetics of dapagliflozin

Detailed Description

Not available

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
14
Inclusion Criteria
  • Healthy subjects
  • Body Mass Index (BMI) of 18 to 32 inclusive
  • Women who are not of childbearing potential and men, ages 18 to 45
Exclusion Criteria
  • Evidence of organ dysfunction or any clinically significant deviation from normal in physical examination, vital signs, electrocardiogram (ECG) or clinical laboratory determinations
  • Glucosuria
  • Abnormal liver function tests

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Dapagliflozin/RifampinDapagliflozin-
Dapagliflozin/RifampinRifampin-
Primary Outcome Measures
NameTimeMethod
AUC (area under the concentration-time curve) Single dose pharmacokinetic parameter will be derived from plasma concentration versus time dataDays 1 to 3 and Days 9 to 11
Secondary Outcome Measures
NameTimeMethod
Cmax (maximum observed concentration) Single dose pharmacokinetic parameter will be derived from plasma concentration versus time dataDays 1 to 3 and Days 9 to 11
Tmax (time of maximum observed concentration) Single dose pharmacokinetic parameter will be derived from plasma concentration versus time dataDays 1 to 3 and Days 9 to 11

Trial Locations

Locations (1)

Ppd Development

🇺🇸

Austin, Texas, United States

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