MedPath

CAbotégravir LENacapavir DUal Long Acting

Phase 2
Not yet recruiting
Conditions
HIV1 Infection
Multi-treated Patients Who Have Received Multiple Lines of Antiretroviral Treatment
CABOTEGRAVIR
LENACAPAVIR
Stable Oral Antiretroviral Treatment for At Least 6 Months
Interventions
Registration Number
NCT06657885
Lead Sponsor
Institut de Médecine et d'Epidémiologie Appliquée - Fondation Internationale Léon M'Ba
Brief Summary

This study is a Phase II, prospective, single-arm, multicenter, non-randomized pilot study designed to evaluate the antiretroviral efficacy of lenacapavir in combination with cabotegravir injection over 48 weeks of follow-up in participants who meet the study inclusion criteria. Efficacy is defined as the absence of virologic failure at S48. Virologic success is defined as maintaining or achieving CV \< 50 copies/mL without interruption of long-acting dual therapy with cabotegravir/lenacapavir at the end of 48 weeks. The study will be conducted at several sites in France in adults 18 years of age and older. Minors and persons under legal guardianship will not be included in the study.

Long-acting treatments are evolving thanks to new "long-acting" molecules. These molecules ensure prolonged efficacy without the need for daily dosing thanks to their long half-life by oral / IM or SC injection (cabotegravir, islatravir, lenacapavir, rilpivirine and bNAbs).

Currently, the only available combination is dual therapy with cabotegravir/rilpivirine administered intramuscularly every two months. However, this injectable combination therapy has its limitations, namely previous resistance to rilpivirine, a number of failures due to certain virological subtypes or poor use of the injectable by certain patients (obesity, injection errors, etc.). For many referral centers caring for patients with HIV, it has become necessary to have a long-acting therapeutic alternative for certain patients. A strategy based on lenacapavir combined with cabotegravir could be a validated alternative for undetectable or detectable patients who have received intensive multidrug regimens, for patients with multidrug resistance, or for patients who are unable to take their oral antiretroviral regimens due to intolerance, drug-drug interactions, or non-adherence.

Recently in the US, the case series presented by Dr. Monica Gandhi (Case series examining the Long-Acting combination of Lenacapavir and Cabotegravir: call for a trial-abstract 629 CROI 2024) demonstrated the high virologic efficacy (94%) of this combination in participants who were unobserved, intolerant or had underlying resistance to antiretroviral therapy (NNRTIs).

The experimental drugs used in this study are cabotegravir, marketed as Vocabria®, and lenacapavir, marketed as Sunlenca®. Both are approved in France for the treatment of HIV-1 infection.

Detailed Description

Not available

Recruitment & Eligibility

Status
NOT_YET_RECRUITING
Sex
All
Target Recruitment
30
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
single-armhis is a prospective, single-arm, multicentre, non-randomised phase II, pilot study designed to achieve or maintain virological success in participants who meet the prescribing criteria for lenacapavi-
Primary Outcome Measures
NameTimeMethod
Percentage of participants with virological failureWeek 24
Secondary Outcome Measures
NameTimeMethod
Metabolic parameters (total cholesterol, LDL-c, HDL-c, triglycerides and fasting plasma glucose) from D0 to W48Between day 0 and week 48
Changes in weight and BMI from D0 to W48Between day 0 and week 48
Percentage of participants with virological failureweek24
Percentage of participants achieving therapeutic success at W48 (absence of virological failure and definitive discontinuation of assigned treatment or study continuation due to intolerance). Change of residence, change of treatment due to pregnancy, forweek 48
Percentage of participants with viruses harbouring resistance mutations to the current treatment at the time of virological failure (by Sanger) and description of the resistance mutations selected at the time of virological failure.at the time of virologic failure
Proportion of minority resistance variants archived in DNA at D0 and their impact on the risk of virological failure and on the selection of resistance mutations.D0
Describe the evolution of the proportion of intact and defective proviruses in PBMC at D0 and W48.day 0 and week 48
Percentage of participants with at least one "blip" (viral load greater than 50 copies/mL with a control less than or equal to 50 copies/mL) between D0 and W48.Between day 0 and week 48
Change in CD4 and CD8 T lymphocytes and CD4/CD8 ratio between W-2 and W48Week -2 and week 48
Description of plasma concentrations of antiretroviral treatments between D0 and W48between day0 and week 48
Incidence of clinical and laboratory grade 3 or higher adverse eventsbetwwen Day 0 and week 48
Incidence of adverse events and discontinuation from study to W48Between day 0 and week 48
Change in participants' symptoms as assessed by self-report questionnaire from D0 to W48Between day 0 and week 48
Assessment of participant satisfaction by questionnaire between D0 and W48Between day 0 and week 48

Trial Locations

Locations (12)

Hopital Saint André

🇫🇷

Bordeaux, France

Hopiytal Pellegrin

🇫🇷

Bordeaux, France

Centre hospitalier François Mitterrand

🇫🇷

Dijon, France

Hopital raymond Poincaré

🇫🇷

Garches, France

Hôpital Franco-Britannique

🇫🇷

Levallois Perret, France

CHU de nantes- Hotel Dieu

🇫🇷

Nantes, France

Chu- Nice Archet

🇫🇷

Nice, France

Hopital Saint Antoine

🇫🇷

Paris, France

Hopital Pitié Salpêtrière

🇫🇷

Paris, France

Hopital Necker

🇫🇷

Paris, France

Hopital Bichat Claude Bernard

🇫🇷

Paris, France

Centre hospitalier de Tourcoing

🇫🇷

Tourcoing, France

© Copyright 2025. All Rights Reserved by MedPath