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A Comparison of Saquinavir Hard- and Soft-Gelatin Capsules in HIV-Infected Patients

Phase 1
Completed
Conditions
HIV Infections
Registration Number
NCT00002383
Lead Sponsor
Hoffmann-La Roche
Brief Summary

To compare the antiviral activity, safety, and pharmacokinetics of saquinavir hard gel capsule (HGC) formulation, to 1 of 3 doses of saquinavir soft gel capsule (SGC) formulation administered orally every 8 hours for 4 weeks.

Detailed Description

Patients are randomly assigned to one of the four treatment groups as follows:

Group 1: 10 patients receive saquinavir HGC. Group 2: 10 patients receive saquinavir SGC. Group 3: 30 patients receive saquinavir SGC at an intermediate dose. Group 4: 30 patients receive saquinavir SGC at the highest study dose. Upon completion of the initial 4 weeks, all patients may have the option to continue their originally-assigned therapy as monotherapy unless significant drug toxicity intervenes. If the analysis of the initial 4 week data identifies an optimal dose of saquinavir SGC, patients may have the option to change to this optimal dose in a treatment extension phase of the protocol. Patients in this extension phase may choose to remain on monotherapy unless they experience significant drug toxicity, their CD4 count or HIV-RNA levels return to baseline, until saquinavir is approved by the FDA or study termination, whichever comes first.

NOTE: A washout \>= 28 days is required for patients on antiretroviral therapy.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
80
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
Not specified
Primary Outcome Measures
NameTimeMethod
Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (10)

Harkness Pavilion

🇺🇸

New York, New York, United States

Mt Zion Hosp of UCSF / HIV Research Ctr

🇺🇸

San Francisco, California, United States

Davis Med Ctr

🇺🇸

San Francisco, California, United States

Oregon Health Sciences Univ

🇺🇸

Portland, Oregon, United States

Univ of Alabama at Birmingham / 1917 Rsch Cln

🇺🇸

Birmingham, Alabama, United States

Pacific Oaks Med Group / Research & Scientific Investiga

🇺🇸

Sherman Oaks, California, United States

Kansas City AIDS Research Consortium

🇺🇸

Kansas City, Missouri, United States

Univ of Texas Med Branch / Virology Clinic

🇺🇸

Galveston, Texas, United States

New England Med Ctr

🇺🇸

Boston, Massachusetts, United States

Tulane Univ Med Ctr / Infectious Diseases Sect

🇺🇸

New Orleans, Louisiana, United States

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