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The Influence of Tramadol on Opioid-induced Bowel Dysfunction

Phase 2
Completed
Conditions
Opioid-Induced Bowel Dysfunction
Constipation
Interventions
Drug: Placebo
Registration Number
NCT06385561
Lead Sponsor
Asbjørn Mohr Drewes
Brief Summary

Tramadol is a weak opioid and widely used to treat moderate to severe pain. Stronger opioids are known to inhibit gastrointestinal motility and secretion, however the effects of tramadol on gastrointestinal function remains less understood. The aim of this study was to determine to what degree tramadol causes opioid-induced bowel dysfunction by using an objective design to explore gastrointestinal transit, motility pattern, secretion, and colonic volume, in a group of healthy male volunteers.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
20
Inclusion Criteria
  • Healthy (assessed by a study-affiliated medical doctor.)
  • Signed informed consent.
  • Able to read and understand Danish.
  • Male (to avoid influence of menstrual cycles)
  • Northern European descent (to minimize genetic variance influences on drug metabolism).
  • The researcher believes that the participant understands the study details, is compliant and is expected to complete the study.
  • Opioid naïve* (who have not taken prescription opioid for one week or longer and at least a year have passed since completion of a previous opioid study.)
  • Between 20 and 40 years of age.
  • A State Trait Anxiety Inventory (STAI) score in the range of 20-37 i.e., classified as "no or low anxiety" at inclusion.
Exclusion Criteria
  • Known hypersensitivity or allergy towards the used pharmaceutical compounds or pharmaceutical compounds similar to those used in the study.
  • Less than three spontaneous bowel movements per week.
  • Participation in other studies within 14 days prior to first visit.
  • Expected need of medical/surgical treatment during the study.
  • Any diagnosed disease, which investigator concludes will affect the trial (including all contraindicated complications: severe chronic obstructive pulmonary disease, pulmonary heart disease, severe bronchial asthma, paralytic ileus, hypercapnia, serious respiratory depression with hypoxia, moderate to severe decreased liver function, gastrointestinal obstruction or perforation, acute surgical abdominal complications such as appendicitis, Mb. Crohn's, ulcerative colitis, and toxic mega colon).
  • History of substance abuse (alcohol, tetrahydrocannabinol (THC), benzodiazepine, central stimulants and/or opioids, urine drug test will be performed prior to treatment start). ¹
  • History of major mental disorders (e.g., major anxiety, major depression or treatment with psychoactive medications etc.) ²
  • Metal implants or pacemaker.
  • Daily use of prescription only medicine
  • Daily alcohol consumption
  • Participation motivated by "wrongful" reasons such as poor economy, or psychosocial issues e.g., problems in the family, loneliness, sadness. People with such problems may be more likely to develop substance dependence.1
  • Intake of alcohol within 48 hours before start of study period or any alcohol consumption during each study period. If consumption takes place during the study the participant will be excluded.
  • Use of any analgesic medication within 48 hours before start as well as for the duration of the study. If consumption takes place during the study the participant will be excluded.
  • Nicotine use

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Placebo treatmentPlaceboPlacebo
Active treatmentTramadolTramadol
Primary Outcome Measures
NameTimeMethod
Total gastrointestinal transit timeFrom day 4 to day 8

Difference in hours from ingestion of a 3D Transit Capsule to expulsion of the capsule during active and placebo treatment

Colorectal transit timeFrom day 4 to day 8

Difference in hours from the entering in the colon of a 3D Transit Capsule to expulsion of the capsule during active and placebo treatment

Secondary Outcome Measures
NameTimeMethod
Bowel movement frequencyFrom day 1 to day 10

Number of spontaneous bowel movements per day

Opiate withdrawal symptomsDay 13, 14 or 15

Measured by the Subjective Opiate Withdrawal Scale (ranging from 0 (not at all) to 4 /extremely)

Colon volumeDay 10

Volumetric quantification of the colon measured using T2-weighted MRI images

Constipation symptomsFrom day 1 to day 10

Measured on the Patient Assessment of Constipation Symptoms (PAC-SYM) questionnaire (ranging from 0 (symptom absent) to 4 (very severe).

Stool consistencyFrom day 1 to day 10

Rated on the Bristol Stool Form Scale (ranging from type 1 (constipation) - type 7 (diarrhea))

Gastrointestinal symptomsDay 1 and day 10

Measured on the Gastrointestinal Symptom Rating Score (GSRS) questionnaire (ranging from 0 (no discomfort) to 6 (very severe discomfort)

Colonic motility patternsFrom day 4 to day 8

Number of motility patterns in the colon measured by the 3D Transit Capsule

Colonic water contentDay 10

Analysis of colonic water content measured using heavily T2-weighted MRI images

Opioid-induced constipationDay 1 and day 10

Measured by the Bowel Function Index (BFI) questionnaire (ranging from 0 (not at all) to 100 (very strong).

Diagnostic evaluation of opioid-induced constipationDay 10

Assessed using the Rome IV C6 criteria consisting of 7 items rated as either true or false. 2 or more items rated as "true" indicates functional constipation

Gastric contraction assessmentDay 1 and day 10

Analysis of gastric contraction frequency after ingestion of a standardized meal measured by MRI

Small bowel motility assessmentDay 1 and day 10

Analysis of small bowel motility after ingestion of a standardized meal measured using dynamic MRI images. A semi-automated analysis software enables registration of small bowel motility with the calculation of regional motility maps and quantification of motility indices.

Gastric half emptying timeDay 1 and day 10

Analysis of gastric half emptying time after ingestion of a standardized meal measured by MRI

Small bowel water contentDay 1 and day 10

Analysis of small bowel water content measured using heavily T2-weighted MRI images

Trial Locations

Locations (1)

Aalborg University Hospital

🇩🇰

Aalborg, Denmark

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