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A Study to Evaluate the Safety and Efficacy of MGD013 in Patients With Melanoma

Phase 1
Terminated
Conditions
Untreated Mucosal or Acral Lentiginous Melanoma
Unresectable, Recurrent or Metastatic Melanoma
Interventions
Registration Number
NCT04653038
Lead Sponsor
Zai Lab (Shanghai) Co., Ltd.
Brief Summary

This is an open-label, multi-cohort, multi-center Phase I clinical trial to evaluate the efficacy and safety of MGD013 in ① Cohort 1: patients with unresectable, recurrent or metastatic melanoma who have failed prior immune checkpoint inhibitor therapy; ② Cohort 2: patients with untreated, unresectable recurrent or metastatic, mucosal or acral lentiginous melanoma.

Detailed Description

The study is conducted in two parts for both Cohort 1 and Cohort 2. Part I: Safety evaluation and efficacy exploration for MGD013. Part II: Efficacy expansion based on results from Part I to further evaluate the efficacy effect of MGD013.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
92
Inclusion Criteria
  • Voluntary and able to provide signed informed consent form

  • Male or female aged ≥ 18 years

  • Patient can comply with protocol requirements as assessed by the investigator

  • Eastern Cooperative Oncology Group (ECOG) performance status score of 0, or 1

  • Histologically confirmed unresectable recurrent or metastatic melanoma:

    • Cohort 1: The pathological type is cutaneous or acral lentiginous, or unknown origin. Progressive or recurrent disease on at least one prior line of systemic therapies. In addition, prior systemic therapies must include one line of anti-PD-(L)1 and/or anti-CTLA-4 immune checkpoint inhibitors. Patients with BRAF-mutated or KIT-mutated/amplified melanoma, and prior treatment with vemurafenib or imatinib is not mandatory;
    • Cohort 2: Histologically confirmed pathological type is acral lentiginous or mucosal. No prior systemic therapy for recurrent or metastatic disease.
  • Patients with at least one measurable lesion according to irRECIST; assessed by investigator per irRECIST criteria to establish a baseline tumor assessment, and should be performed within 28 days prior to the first dose.

Exclusion Criteria
  • The pathological type of patient is:

    • Cohort 1: Mucosal melanoma; uveal melanoma;
    • Cohort 2: Cutaneous melanoma; uveal melanoma; melanoma of unknown origin; known BRAF mutation or KIT mutation/amplification.
  • Central nervous system metastases with clinical symptoms. Patients with prior central nervous system metastases who have received local therapy, have stable disease for ≥ 4 weeks, and meet the following criteria can be enrolled:

    • No treatment for central nervous system metastases during the screening period (e.g., surgery, radiotherapy, mannitol, corticosteroid therapy-prednisolone > 10 mg per day or equivalent dose)
    • No progression of central nervous system lesions on MRI or CT within 14 days prior to start of study treatment
    • No meningeal metastasis or notochord compression
  • Subjects with a history of symptomatic pulmonary fibrosis, interstitial pneumonia, pneumoconiosis, radiation pneumonitis, drug-related pneumonia, severely impaired pulmonary function or may interfere with the detection and treatment of suspected drug-related pulmonary adverse reactions;

  • Prior treatment with any antibody/drug targeting the regulation of T cell function (immune checkpoint) (e.g., anti-LAG-3, anti-0X-40, anti-CD137, anti-TIM-3, anti-TIGIT, IDO)

  • Patients who have previously received immune checkpoint inhibitors (e.g., anti-PD-(L)1, anti-CTLA-4 antibody) are not included if they experience any of the following immune checkpoint-related adverse events, regardless of recovery:

    • ≥ Grade 3 ocular adverse events
    • Grade 4 liver function abnormalities
    • Grade ≥ 3 neurologic adverse reactions
    • ≥ Grade 3 colitis
    • ≥ Grade 3 renal adverse reactions
    • ≥ Grade 3 pneumonitis

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Unresectable, recurrent or metastatic melanomaMGD013Cohort1: patients with unresectable, recurrent or metastatic melanoma who have failed prior immune checkpoint inhibitor therapy
Untreated mucosal or acral lentiginous melanomaMGD013Cohort2: patients with untreated, unresectable recurrent or metastatic, mucosal or acral lentiginous melanoma
Primary Outcome Measures
NameTimeMethod
Objective Response Rate (ORR)Approximately 12 months after dosed

Objective Response Rate (ORR) is defined as the proportion of patients with a best response of CR or PR in enrolled patients, which is assessed by Independent Review Committee (IRC) per RECIST v1.1

Secondary Outcome Measures
NameTimeMethod
Overall Survival (OS)Approximately 24 months

Overall Survival (OS) is defined as the time from patient enrollment to death due to any cause

Objective Response Rate (ORR)Approximately 12 months after dosed

Objective Response Rate (ORR) as assessed by Investigator and IRC per irRECIST.

Survival RateApproximately 12 months after dosed

Survival Rate is defined as the proportion of surviving patients at the corresponding time point. Survival rates at 6 and 12 months will be analyzed in this study

Incidence of Adverse EventsApproximately 24 months

The incidence of adverse events is defined as the proportion of the patients who have adverse event(s) enrolled in this study.

Progression-free Survival (PFS)Approximately 12 months after dosed

Progression-free Survival (PFS) is defined as the time from patient enrollment to tumor progression or death due to any cause. Progression is assessed per RECIST 1.1 and irRECIST criteria, respectively

Trough Serum Concentration (Ctrough)Approximately 3 months

The through serum concentration (Cmin, ng/ml) is defined as the minimum (or through) serum concentration reached by MGD013 prior to administration of a second dose.

Disease Control Rate (DCR)Approximately 12 months after dosed

Disease Control Rate (DCR) is defined as the time from patient enrollment to tumor progression or death due to any cause. The tumor progression is assessed per RECIST 1.1 and irRECIST criteria, respectively

Duration of Response (DoR)Approximately 12 months after dosed

Duration of Response (DoR) is defined as the time from radiographic response to disease progression or death in patients with a best response of CR or PR, assessed per RECIST 1.1 and irRECIST criteria, respectively

Incidence of Abnormal Laboratory valueApproximately 24 months

Incidence of abnormal laboratory is defined as the proportion of patients who have abnormal laboratory value not prior to the initiation of MGD013 administration

Incidence of Treatment-Emergent Adverse EventsApproximately 24 months.

The incidence of treatment-emergent adverse event is defined as any event not present prior to the initiation of MGD013 treatment or any event already present that worsens in either intensity or frequency following exposure to MGD013 administration.

Maximum Serum Concentration (Cmax)Approximately 3 months.

The maximum serum concentration (Cmax, ng/ml) is defined as the maximum (or peak) serum concentration that MGD013 achieves in patients after the MGD013 administration at a corresponding timepoint.

Immunogenicity of MGD013Approximately 6 months after dosed

Immunogenicity is defined as the positivity measured as the anti-MGD013 antibody induced in serum after MGD013 is administrated into human body at corresponding timepoints.

Trial Locations

Locations (13)

Jiangsu Province Hospital

🇨🇳

Nanjing, Jiangsu, China

Nanjing Drum Tower Hospital

🇨🇳

Nanjing, Jiangsu, China

Beijing Cancer Hospital

🇨🇳

Beijing, Beijing, China

Union Hospital Affiliated to Tongji Medical College of Huazhong University of Science and Technology

🇨🇳

Wuhan, Hubei, China

Hunan Cancer Hospital

🇨🇳

Changsha, Hunan, China

The first hospital of Jilin University

🇨🇳

Chang chun, Jilin, China

Jilin Cancer Hospital

🇨🇳

Changchun, Jilin, China

Tangdu Hospital

🇨🇳

Xi'an, Shanxi, China

Fudan University Shanghai Cancer Center

🇨🇳

Shanghai, Shanghai, China

Tianjin Cancer Hospital

🇨🇳

Tianjin, Tianjin, China

Zhejiang Cancer Hospital

🇨🇳

Hangzhou, Zhejiang, China

Sir Run Shaw Hospital, School Of Medicine ,Zhejiang University

🇨🇳

Hangzhou, Zhejiang, China

Fujian Cancer Hospital

🇨🇳

Fuzhou, Fujian, China

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