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Study to Compare Conivaptan in Subjects With Mild & Moderate Liver Impairment Versus Subjects With Normal Liver Function

Phase 1
Completed
Conditions
Liver Disease
Hyponatremia
Interventions
Registration Number
NCT00851227
Lead Sponsor
Cumberland Pharmaceuticals
Brief Summary

A study to compare a 48-hour continuous infusion of conivaptan in subjects with mild and moderate liver impairment versus subjects with normal liver function

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
26
Inclusion Criteria
  • Subjects with Normal Hepatic Function:

    • Weighs at least 45 kg
    • Body mass index between 18 and 40 kg/m2 inclusive
    • Must have normal hepatic function
  • Hepatic Impaired Subjects:

    • Weighs at least 45 kg
    • Meets criteria for mild or moderate hepatic impairment defined by Child-Pugh method
    • Body mass index between 18 and 40 kg/m2 inclusive
Exclusion Criteria
  • Subjects with Normal Hepatic Function:

    • Smokes more than 10 cigarettes per day
    • Known to be HIV positive or has HIV antibodies
    • Has clinically significant history or presence of illness, malignancy, or immunodeficiency
    • Is Hepatitis A, B, or C positive
    • Has had a blood transfusion or donated/lost more than 550ml of blood within 8 weeks of study drug administration
    • History of substance abuse within 6 months prior to screening
  • Hepatic Impaired Subjects:

    • Has history or presence of biliary obstruction or biliary disease, hepatic encephalopathy, advanced acidities, portal hypertension, or biliary liver cirrhosis
    • Is hypovolemic or has evidence of orthostatic hypotension
    • Smokes more than 10 cigarettes per day
    • Known to be HIV positive or has HIV antibodies
    • Has clinically significant history or presence of illness, malignancy, or immunodeficiency
    • Has clinically significant history or presence of GI symptoms other than those associated with moderate hepatic impairment
    • Has had a blood transfusion or donated/lost more than 550ml of blood within 8 weeks of study drug administration
    • History of substance abuse within 6 months prior to screening

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
1. Mildly Hepatic Impaired Subjectsconivaptan hydrochloride-
2. Moderately Hepatic Impaired Subjectsconivaptan hydrochloride-
3. Subjects with Normal Hepatic Functionconivaptan hydrochloride-
Primary Outcome Measures
NameTimeMethod
Measure PK and protein binding of conivaptan5 days
Secondary Outcome Measures
NameTimeMethod
Measure tolerability of conivaptan5 days
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