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Combination Margetuximab, Retifanlimab, Tebotelimab, and Chemotherapy Phase 2/3 Trial in HER2+ Gastric/GEJ Cancer

Phase 2
Completed
Conditions
Gastric Cancer
Gastroesophageal Junction Cancer
HER2-positive Gastric Cancer
Interventions
Registration Number
NCT04082364
Lead Sponsor
MacroGenics
Brief Summary

This is a Phase 2/3, randomized, open-label study for the treatment of patients with HER2-positive Gastric cancer (GC) or Gastroesophageal Junction (GEJ) cancer conducted in two parts.

Part A is a single-arm cohort (Cohort A, 40 to 110 participants) will evaluate safety and efficacy of margetuximab plus retifanlimab.

Part B Part 1 has 4 arms (50 patients/arm). Participants will be randomized to margetuximab plus retifanlimab plus chemotherapy, margetuximab plus tebotelimab, plus chemotherapy, margetuximab plus chemotherapy, or trastuzumab plus chemotherapy.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
82
Inclusion Criteria
  • Histologically confirmed diagnosis of previously untreated locally advanced unresectable or metastatic HER2+ GC or GEJ adenocarcinoma

    1. Prior systemic perioperative treatment is allowed; however the participants must have had a disease-free interval of at least 6 months from end of chemo/surgery
    2. Participants receiving perioperative anti-HER2 therapy require testing of HER2 status for eligibility
    3. Cohort A: HER2-positive (by IHC 3+) and PD-L1-positive (by IHC with 22C3 CPS ≥ 1%) per central review
    4. Cohort B: HER2-positive (by IHC 3+ or IHC 2+ in combination with FISH+) by local review. PD -L1 status is not required for enrollment.
  • Availability of formalin-fixed, paraffin-embedded tumor specimen, unstained slides or contemporaneous biopsy for tumor target testing

  • Eastern Cooperative Oncology Group performance status of 0 or 1, verified within 3 days of Day 1

  • Life expectancy ≥ 6 months

  • At least one radiographically measurable target lesion

  • Acceptable laboratory parameters and adequate organ function

Key

Exclusion Criteria
  • Other malignancy that is progressing or required treatment within the past 5 years, with certain exceptions

    • Participants with known MSI-H status
  • History of allogeneic stem cell or tissue/solid organ transplant

  • Central nervous system metastases

  • Clinically significant cardiovascular disease, gastrointestinal disorders, pulmonary compromise

    • Prior neoadjuvant or adjuvant treatment with immunotherapy

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Chemotherapy-free armmargetuximabmargetuximab plus retifanlimab
Chemotherapy-free armRetifanlimabmargetuximab plus retifanlimab
Margetuximab, retifanlimab, and chemotherapy armRetifanlimabmargetuximab plus retifanlimab plus investigator choice of chemotherapy options. Chemotherapy options: capecitabine and oxaliplatin (XELOX) or modified 5-FU, leucovorin, and oxaliplatin regimen 6 (mFOLFOX-6)
Trastuzumab and chemotherapy armChemotherapyTrastuzumab plus investigator choice of chemotherapy options. Chemotherapy options: capecitabine and oxaliplatin (XELOX) or modified 5-FU, leucovorin, and oxaliplatin regimen 6 (mFOLFOX-6)
Margetuximab, retifanlimab, and chemotherapy armmargetuximabmargetuximab plus retifanlimab plus investigator choice of chemotherapy options. Chemotherapy options: capecitabine and oxaliplatin (XELOX) or modified 5-FU, leucovorin, and oxaliplatin regimen 6 (mFOLFOX-6)
Margetuximab, retifanlimab, and chemotherapy armChemotherapymargetuximab plus retifanlimab plus investigator choice of chemotherapy options. Chemotherapy options: capecitabine and oxaliplatin (XELOX) or modified 5-FU, leucovorin, and oxaliplatin regimen 6 (mFOLFOX-6)
Margetuximab, tebotelimab and chemotherapy armmargetuximabmargetuximab plus tebotelimab plus investigator choice of chemotherapy options. Chemotherapy options: capecitabine and oxaliplatin (XELOX) or modified 5-FU, leucovorin, and oxaliplatin regimen 6 (mFOLFOX-6)
Margetuximab, tebotelimab and chemotherapy armTebotelimabmargetuximab plus tebotelimab plus investigator choice of chemotherapy options. Chemotherapy options: capecitabine and oxaliplatin (XELOX) or modified 5-FU, leucovorin, and oxaliplatin regimen 6 (mFOLFOX-6)
Margetuximab, tebotelimab and chemotherapy armChemotherapymargetuximab plus tebotelimab plus investigator choice of chemotherapy options. Chemotherapy options: capecitabine and oxaliplatin (XELOX) or modified 5-FU, leucovorin, and oxaliplatin regimen 6 (mFOLFOX-6)
Margetuximab and chemotherapy armmargetuximabmargetuximab plus investigator choice of chemotherapy options. Chemotherapy options: capecitabine and oxaliplatin (XELOX) or modified 5-FU, leucovorin, and oxaliplatin regimen 6 (mFOLFOX-6)
Margetuximab and chemotherapy armChemotherapymargetuximab plus investigator choice of chemotherapy options. Chemotherapy options: capecitabine and oxaliplatin (XELOX) or modified 5-FU, leucovorin, and oxaliplatin regimen 6 (mFOLFOX-6)
Trastuzumab and chemotherapy armTrastuzumabTrastuzumab plus investigator choice of chemotherapy options. Chemotherapy options: capecitabine and oxaliplatin (XELOX) or modified 5-FU, leucovorin, and oxaliplatin regimen 6 (mFOLFOX-6)
Primary Outcome Measures
NameTimeMethod
Number of Participants With Adverse Events of Margetuximab Plus Retifanlimab in Cohort A, as Assessed by CTCAE v5.0Throughout the study, an average of 11 months.

Evaluation of adverse events and serious adverse events (Cohort A)

Objective Response Rate (ORR) for Non-microsatellite Instability-high (Non-MSI-H) Participants (Cohort A) Using Investigator-assessed Radiology ReviewsThroughout the study, an average of 11 months.

Percent of non MSI-H participants with best overall response of complete response (CR) plus partial response (PR) per RECIST 1.1 (Cohorts A ) based on investigator assessment.

CR is defined as the disappearance of all target and non-target lesions with no new lesions appearing PR is defined as \>= to a 30% decrease in the sum of the longest dimensions of target lesions, non-progression of non- target lesions, with no new lesions appearing.

CR + PR = ORR

Secondary Outcome Measures
NameTimeMethod
Median Progression-free Survival Using Investigator-assessed Radiology Reviews in Cohort AThroughout the study, an average of 11 months.

Time from start of study treatment to the first documented disease progression per RECIST v1.1 or death due to any cause, whichever occurs first. (Cohorts A) based on investigator assessment

Median Duration of Response in Cohort A Using Investigator-assessed Radiology ReviewsThroughout the study, an average of 11 months.

Time from the date of initial response (CR or PR) to the date of first documented progression or death from any cause, whichever occurs first (Cohorts A)

Disease Control RateThroughout the study, an average of 11 months.

Percentage of patients who experienced response of CR, PR or stable disease for at least 3 months from start of study treatment (Cohorts A and B)

ORR for Cohort BThroughout the study, an average of 11 months.

Proportion of participants with best overall response of CR plus PR per RECIST 1.1

Number of Participants Who Have Antidrug Antibodies (ADA) to MargetuximabThroughout the study, an average of 11 months.
Number of Participants Who Have ADA to RetifanlimabThroughout the study, an average of 11 months.
Number of Participants Who Have ADA to TebotelimabThroughout the study, an average of 11 months.

Trial Locations

Locations (73)

Rutgers Cancer Institute of New Jersey

🇺🇸

New Brunswick, New Jersey, United States

Mayo Clinic - Scottsdale

🇺🇸

Scottsdale, Arizona, United States

City of Hope Comprehensive Cancer Center - Duarte

🇺🇸

Duarte, California, United States

Norris Comprehensive Cancer Center (USC)

🇺🇸

Los Angeles, California, United States

UCLA School of Medicine

🇺🇸

Santa Monica, California, United States

Salinas Memorial

🇺🇸

Salinas, California, United States

Florida Cancer Specialists South

🇺🇸

Fort Myers, Florida, United States

Mayo Clinic - Jacksonville

🇺🇸

Jacksonville, Florida, United States

Ocala Oncology Center PL DBA Florida Cancer Affiliates - Ocala

🇺🇸

Ocala, Florida, United States

Cancer & Hematology Centers of Western Michigan - Lemmen-Holton Cancer Pavilion

🇺🇸

Grand Rapids, Michigan, United States

Florida Cancer Specialists North

🇺🇸

Saint Petersburg, Florida, United States

Azienda Ospedaliero-Universitaria Pisana

🇮🇹

Pisa, Italy

University of Chicago

🇺🇸

Chicago, Illinois, United States

Massachusetts General Hospital Cancer Center

🇺🇸

Boston, Massachusetts, United States

Swedish Cancer Institute

🇺🇸

Seattle, Washington, United States

SIR RUN RUN SHAW Hospital, Zhejiang University school of medicine

🇨🇳

Hangzhou, China

Zhejiang Cancer Hospital

🇨🇳

Hangzhou, China

The First Affiliated Hospital of Anhui Medical University

🇨🇳

Hefei, China

Anhui Provincial Cancer Hospital

🇨🇳

Hefei, China

Henan Cancer Hospital

🇨🇳

Zhengzhou, China

The First Affiliated Hospital of Zhengzhou University

🇨🇳

Zhenzhou, China

Henry Ford Health System

🇺🇸

Detroit, Michigan, United States

Stephenson Cancer Center at OUHSC

🇺🇸

Oklahoma City, Oklahoma, United States

Sarah Cannon Research Institute

🇺🇸

Nashville, Tennessee, United States

Oncology Consultants

🇺🇸

Houston, Texas, United States

Utah Cancer Specialists

🇺🇸

Salt Lake City, Utah, United States

SPSK nr 1 in Lublin

🇵🇱

Lublin, Poland

Kaohsiung Chang Gung MemorialHospital

🇨🇳

Kaohsiung, Taiwan

National Cancer Center Singapore

🇸🇬

Singapore, Singapore

Liuying Chi MeiMedical Hospital

🇨🇳

Tainan city, Taiwan

Chang Gung Memorial Hospital, Keelung

🇨🇳

Keelung, Taiwan

National Taiwan University

🇨🇳

Taipei, Taiwan

Centrum Medyczne MrukMed

🇵🇱

Rzeszów, Poland

Taipei Medical University Hospital

🇨🇳

Taipei City, Taipei, Taiwan

Edward H. Kaplan MD & Associates

🇺🇸

Skokie, Illinois, United States

Nebraska Heme Onc

🇺🇸

Lincoln, Nebraska, United States

Washington University School of Medicine

🇺🇸

Saint Louis, Missouri, United States

Beijing Cancer Hospital

🇨🇳

Beijing, China

Jilin Cancer Hospital (Second People's Hospital Of Jilin Province)

🇨🇳

Changchun, China

Affiliated Tumor Hospital of Harbin Medical University- the 3rd Affiliated Hospital of Harbin

🇨🇳

Harbin, China

Fujian Medical University - Fujian Provincial Cancer Hospital (Fujian Provincial Tumor Hospital)

🇨🇳

Fuzhou, China

Hebei cancer hospital (The Fourth Affiliate)

🇨🇳

Shijiazhuang, China

Jinan Center Hospital

🇨🇳

Jinan, China

Wuhan Union Hospital

🇨🇳

Wuhan, China

Zhongshan Hospital Fudan University

🇨🇳

Shanghai, China

Liaoning cancer hospital

🇨🇳

Shenyang, China

Institute of Clinical Cancer Research Krankenhaus Nordwest (IKF)

🇩🇪

Frankfurt, Germany

Haematologisch-Onkologische Praxis Eppendorf

🇩🇪

Hamburg, Germany

Korea University, Anam Hospital

🇰🇷

Seoul, Korea, Republic of

Istituto Europeo Di Oncologia

🇮🇹

Milan, Italy

Universitätsmedizin Mainz

🇩🇪

Mainz, Germany

Ospedale San Raffaele

🇮🇹

Milan, Italy

Kliniken Maria Hilf GmbH

🇩🇪

Monchengladbach, Germany

CHA bundang

🇰🇷

Gyeonggi-do, Korea, Republic of

Inje University Haeundae Paik Hospital

🇰🇷

Haeundae, Korea, Republic of

Hallym University Sacred Heart Hospital

🇰🇷

Anyang-Si, Korea, Republic of

Seoul National University Bundang Hospital

🇰🇷

Seongnam-si, Korea, Republic of

Samsung Medical Center

🇰🇷

Seoul, Korea, Republic of

Korea University Guro

🇰🇷

Seoul, Korea, Republic of

Seoul National University Hospital

🇰🇷

Seoul, Korea, Republic of

Asan Medical Center

🇰🇷

Seoul, Korea, Republic of

Catholic University of Korea St. Vincent Hospital

🇰🇷

Suwon, Korea, Republic of

Yonsei University College of Medicine (Severance Hospital)

🇰🇷

Seoul, Korea, Republic of

National University Hospital (Cancer Institute) -Singapore

🇸🇬

Singapore, Singapore

The Christie Hospital NHS Foundation Trust

🇬🇧

Manchester, United Kingdom

Cambridge University Hospitals NHS Foundation Trust Addenbrooke's Hospital

🇬🇧

Cambridge, United Kingdom

Virginia Cancer Specialists

🇺🇸

Fairfax, Virginia, United States

Yale University

🇺🇸

New Haven, Connecticut, United States

Mayo Clinic - Rochester

🇺🇸

Rochester, Minnesota, United States

Kaiser Permanente

🇺🇸

Honolulu, Hawaii, United States

University of Wisconsin

🇺🇸

Madison, Wisconsin, United States

The University of New Mexico Comprehensive Cancer Center

🇺🇸

Albuquerque, New Mexico, United States

Nanjing University Medical School; Nanjing Drug Tower

🇨🇳

Nanjing, China

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