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Effisayil™ 1: A Study to Test Spesolimab (BI 655130) in Patients With a Flare-up of a Skin Disease Called Generalized Pustular Psoriasis

Phase 2
Completed
Conditions
Generalized Pustular Psoriasis
Interventions
Drug: Placebo
Drug: Spesolimab
Registration Number
NCT03782792
Lead Sponsor
Boehringer Ingelheim
Brief Summary

To evaluate efficacy, safety, and tolerability of spesolimab (BI 655130) compared to placebo in patients with Generalized Pustular Psoriasis (GPP) presenting with an acute flare of moderate to severe intensity.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
53
Inclusion Criteria
  • Patients with GPPGA of 0 or 1 and a known and documented history of GPP per European Rare And Severe Psoriasis Expert Network (ERASPEN) criteria regardless of IL36RN mutation status, with previous evidence of fever, and/or asthenia, and/or myalgia, and/or elevated C-reactive protein, and/or leucocytosis with peripheral blood neutrophilia (above ULN) OR

    -- Patients with an acute flare of moderate to severe intensity meeting the (ERASPEN) criteria of GPP with a known and documented history of GPP (per ERASPEN criteria) regardless of IL36RN mutation status, with previous evidence of fever, and/or asthenia, and/or myalgia, and/or elevated C-reactive protein, and/or leucocytosis with peripheral blood neutrophilia (above ULN)

  • Male or female patients, aged 18 to 75 years at screening.

  • Signed and dated written informed consent prior to admission to the study in accordance with ICH GCP and local legislation prior to start of any screening procedures.

  • Women of childbearing potential must be ready and able to use highly effective methods of birth control per ICH M3 (R2) that result in a low failure rate of less than 1% per year when used consistently and correctly. Note: A woman is considered of childbearing potential, i.e. fertile, following menarche and until becoming postmenopausal unless permanently sterile. Permanent sterilisation methods include hysterectomy, bilateral salpingectomy and bilateral oophorectomy. Tubal ligation is not a method of permanent sterilization. A postmenopausal state is defined as no menses for 12 months without an alternative medical cause

  • Further inclusion criteria apply

Read More
Exclusion Criteria
  • Patients with SAPHO (Synovitis-acne-pustulosis-hyperostosis-osteitis) syndrome.
  • Patients with primary erythrodermic psoriasis vulgaris.
  • Patients with primary plaque psoriasis vulgaris without presence of pustules or with pustules that are restricted to psoriatic plaques.
  • Drug-triggered Acute Generalized Exanthematous Pustulosis (AGEP).
  • Immediate life-threatening flare of GPP or requiring intensive care treatment, according to the investigator's judgement. Life-threatening complications mainly include, but are not limited to, cardiovascular/cytokine driven shock, pulmonary distress syndrome, or renal failure.
  • Severe, progressive, or uncontrolled hepatic disease, defined as >3- fold Upper Limit of Normal (ULN) elevation in AST or ALT or alkaline phosphatase, or >2-fold ULN elevation in total bilirubin.
  • Further exclusion criteria apply
Read More

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PlaceboPlacebo-
SpesolimabSpesolimab-
Primary Outcome Measures
NameTimeMethod
Proportion of Patients With a Generalized Pustular Psoriasis Physician Global Assessment (GPPGA) Pustulation Subscore of 0 Indicating no Visible Pustules at Week 1At Week 1.

The Generalized Pustular Psoriasis Physician Global Assessment (GPPGA) relies on clinical assessment of the Generalized Pustular Psoriasis (GPP) patient's skin presentation. The investigator (or qualified site personnel) scored the erythema, pustules, and scaling of all GPP lesions from 0 to 4.

The GPPGA pustulation subscore ranges from 0 to 4 where:

0 = clear;

1. = almost clear;

2. = mild:

3. = moderate;

4. = severe. A lower GPPGA pustulation subscore indicates a better outcome. A GPPGA pustulation subscore of 0 means no visible pustules.

The proportion of patients who achieved a GPPGA pustulation subscore of 0 at Week 1 is reported.

Secondary Outcome Measures
NameTimeMethod
Proportion of Patients With a Psoriasis Area and Severity Index for Generalized Pustular Psoriasis (GPPASI) 75 at Week 4At Week 4.

Generalized Pustular Psoriasis Area and Severity Index (GPPASI) provides a numeric scoring for a patient's overall Generalized Pustular Psoriasis (GPP) disease state, ranging from 0 to 72. It is a linear combination of percent of surface area of skin affected by erythema, pustules, and scaling and the severity of erythema, pustules, and scaling (desquamation) over 4 body regions (head, trunk, upper limbs and lower limbs).

A higher score indicates a worse disease state, while a score of 0 indicates no disease. GPPASI 75 is based on the percent reduction from baseline, generally summarized as a dichotomous outcome based on achieving over an 75% reduction.

Proportion of patients with GPPASI 75 at Week 4 is reported.

Proportion of Patients With a Generalized Pustular Psoriasis Area and Severity Index (GPPASI) 50 at Week 1At Week 1.

Generalized Pustular Psoriasis Area and Severity Index (GPPASI) provides a numeric scoring for a patient's overall Generalized Pustular Psoriasis (GPP) disease state, ranging from 0 to 72. It is a linear combination of percent of surface area of skin affected by erythema, pustules, and scaling and the severity of erythema, pustules, and scaling (desquamation) over 4 body regions (head, trunk, upper limbs and lower limbs).

A higher score indicates a worse disease state, while a score of 0 indicates no disease. GPPASI 50 is based on the percent reduction from baseline, generally summarized as a dichotomous outcome based on achieving over an 50 % reduction.

Proportion of patients with GPPASI 50 at Week 1 is reported.

Occurrence of Treatment Emergent Adverse Events (TEAEs) up to Week 1From start of treatment until Day 7, up to 7 days.

TEAEs were all Adverse Events (AEs) occurring between start of treatment and Day 8 (Day 8 excluded). AEs that started before first drug intake and deteriorated under treatment were also considered as 'treatment-emergent'.

The exposure-adjusted incidence rate was calculated as:

Incidence rate \[1/100 patients-years\] = 100 × number of patients with AE / Total AE specific time at risk \[patient-years\] where: Time at risk \[patient-years\] = (date of onset of TEAE - study drug start date + 1) /365.25

Number of Patients With Treatment Emergent Adverse Events (TEAEs) Within the Treatment PhaseFrom start of treatment until end of the residual effect period (REP) but censored at any use of open label spesolimab, up to 16 weeks.

TEAEs were all Adverse Events (AEs) occurring between start of treatment and end of the residual effect period (REP) (16 weeks). AEs that started before first drug intake and deteriorated under treatment were also considered as 'treatment-emergent'.

Change From Baseline in Functional Assessment of Chronic Illness Therapy (FACIT) - Fatigue Score at Week 4Baseline and at Week 4.

The FACIT-Fatigue is a 13-item questionnaire that assesses self-reported fatigue and its impact upon daily activities and function. Each items is scored from 0 to 4. Score range is 0 (extreme fatigue)-52 (no fatigue).

Change from baseline=FACIT Fatigue score at Week 4- FACIT-Fatigue score at baseline. Death, any use of escape medication, OL Spesolimab at Day 8, or rescue medication with Spesolimab after Day 8, prior to observing the endpoint was considered to reflect a failure to achieve the endpoint outcome, i.e. non-response (NR). NR is not a missing value but the worst possible outcome of the endpoint. For example, if the achieved data is s (NR, NR, NR, NR, NR, NR, 2, 3, 3, 3, 5) then Q1 is NR, median is NR and Q3 is 3.

Proportion of Patients With a Generalized Pustular Psoriasis Physician Global Assessment (GPPGA) Score of 0 or 1 at Week 4At Week 4.

GPPGA relied on clinical assessment of the Generalized Pustular Psoriasis (GPP) patient's skin presentation. The GPPGA total score is calculated by taking the mean of the erythema subscore, pustules subscore and scaling/crusting subscore. The severity of each subscore was assessed using a 5 point scale score ranging from 0 to 4 (0=clear, 1=almost clear, 2=mild, 3=moderate, 4=severe). The final GPPGA score is assigned as follows:

* 0, if scores for all three scores are 0,

* 1, if 0 \< mean \< 1.5,

* 2, if 1.5 ≤ mean \< 2.5,

* 3, if 2.5 ≤ mean \< 3.5,

* 4, if mean ≥ 3.5. A lower GPPGA score indicates a better outcome, with 0 being clear and 1 being almost clear.

The proportion of participants with a GPPGA score of 0 or 1 at Week 4 is reported.

Proportion of Patients With a Generalized Pustular Psoriasis Physician Global Assessment (GPPGA) Pustulation Sub-score of 0 Indicating no Visible Pustules at Week 4At Week 4.

The Generalized Pustular Psoriasis Physician Global Assessment (GPPGA) relies on clinical assessment of the Generalized Pustular Psoriasis (GPP) patient's skin presentation. The investigator (or qualified site personnel) scores the erythema, pustules, and scaling of all GPP lesions from 0 to 4.

The GPPGA pustulation subscore ranges from 0 to 4 where:

0 = clear;

1. = almost clear;

2. = mild:

3. = moderate;

4. = severe. A lower GPPGA pustulation subscore indicates a better outcome. The proportion of patients who achieved a GPPGA pustulation subscore of 0 at Week 1 is reported.

Key Secondary: Proportion of Patients With a Generalized Pustular Psoriasis Physician Global Assessment (GPPGA) Score of 0 or 1 at Week 1At Week 1.

GPPGA relied on clinical assessment of the Generalized Pustular Psoriasis (GPP) patient's skin presentation. The GPPGA total score was calculated by taking the mean of the erythema subscore, pustules subscore and scaling/crusting subscore. The severity of each subscore was assessed using a 5 point scale score ranging from 0 to 4 (0=clear, 1=almost clear, 2=mild, 3=moderate, 4=severe). The final GPPGA score is assigned as follows:

* 0, if scores for all three subscores are 0,

* 1, if 0 \< mean \< 1.5,

* 2, if 1.5 ≤ mean \< 2.5,

* 3, if 2.5 ≤ mean \< 3.5,

* 4, if mean ≥ 3.5. A lower GPPGA score indicates a better outcome, with 0 being clear and 1 being almost clear. The proportion of patients with a GPPGA score of 0 or 1 at Week 1 is reported.

Percent Change in Generalized Pustular Psoriasis Area and Severity Index (GPPASI) From Baseline at Week 4Baseline and at Week 4.

GPPASI provides a numeric scoring for a patient's overall Generalized Pustular Psoriasis (GPP) disease state, ranging from 0 (no disease) to 72 (worse disease state). It is a linear combination of percent of surface area of skin affected by erythema, pustules, and scaling and the severity of erythema, pustules, and scaling (desquamation) over 4 body regions (head, trunk, upper limbs and lower limbs).

%GPPASI change from baseline=(GPPASI at Week 4-GPPASI at baseline) \*100/(GPPASI at baseline).

Death, any use of escape medication, OL Spesolimab at Day 8, or rescue medication with Spesolimab after Day 8, prior to observing the endpoint was considered to reflect a failure to achieve the endpoint outcome, i.e. non-response (NR).NR is not a missing value but the worst possible outcome of the endpoint. For example, if the achieved data is (NR, NR, NR, NR, NR, NR, 2, 3, 3, 3, 5) then Q1 is NR, median is NR and Q3 is 3. Planned statistical analysis were not performed due to lack of valid data.

Percent Change in Generalized Pustular Psoriasis Area and Severity Index (GPPASI) From Baseline at Week 1At Week 1.

Generalized Pustular Psoriasis Area and Severity Index (GPPASI) provides a numeric scoring for a patient's overall Generalized Pustular Psoriasis (GPP) disease state, ranging from 0 to 72. It is a linear combination of percent of surface area of skin affected by erythema, pustules, and scaling and the severity of erythema, pustules, and scaling (desquamation) over 4 body regions (head, trunk, upper limbs and lower limbs).

A higher score indicates a worse disease state, while a score of 0 indicates no disease.

The percent change from baseline at Week 1 is calculated as:

% GPPASI change from baseline = (GPPASI at Week 1 - GPPASI at baseline) \*100/GPPASI at baseline. If % GPPASI change from baseline is positive, it means the disease is becoming worse.

Occurrence of Treatment Emergent Adverse Events (TEAEs) Within the Treatment PhaseFrom start of treatment until end of the residual effect period (REP) but censored at any use of open label spesolimab, up to 16 weeks.

TEAEs were all Adverse Events (AEs) occurring between start of treatment and end of the residual effect period (REP) (16 weeks). AEs that started before first drug intake and deteriorated under treatment were also considered as 'treatment-emergent'.

The exposure-adjusted incidence rate was calculated as:

Incidence rate \[1/100 patients-years\] = 100 × number of patients with AE / Total AE specific time at risk \[patient-years\] where Time at risk where: Time at risk \[patient-years\] = (date of onset of TEAE - study drug start date + 1) /365.25 If, for a patient, the selected TEAE did not occur then the time at risk was censored at min

* Date of death

* For patients who did not roll over into the Open Label Extension (OLE) study: last contact date Visit14/15

* For patients who rolled over into the OLE study: the 1st dose in the OLE study

* Drug stop date + 112 days

* Date of Day 8 if OL spesolimab was given

* Date of rescue medication if spesolimab was given.

Change From Baseline in Pain Visual Analog Scale (VAS) Score at Week 4Baseline and at Week 4.

The pain Visual Analogue Scale (VAS) is a participant-administered single-item scale designed to measure skin pain intensity from generalized pustular psoriasis (GPP) using a 100 millimeter (mm) horizontal VAS. Overall severity of participant's skin pain from GPP is indicated by placing a single mark on the horizontal 100 mm scale from 0 mm (no pain) to 100 mm (pain as bad as one can imagine).

Change from baseline was calculated by subtracting the VAS score at baseline from the VAS score at Week 4. A negative change indicates an improvement from baseline.

Death, any use of escape medication, OL Spesolimab at Day 8, or rescue medication with Spesolimab after Day 8, prior to observing the endpoint was considered to reflect a failure to achieve the endpoint outcome, i.e. non-response (NR).

NR is not a missing value but the worst possible outcome of the endpoint. For example, if the achieved data is (NR, NR, NR, NR, NR, NR, 2, 3, 3, 3, 5) then Q1 is NR, median is NR and Q3 is 3.

Proportion of Patients With a Generalized Pustular Psoriasis Area and Severity Index (GPPASI) 50 at Week 4At Week 4.

Generalized Pustular Psoriasis Area and Severity Index (GPPASI) provides a numeric scoring for a patient's overall Generalized Pustular Psoriasis (GPP) disease state, ranging from 0 to 72. It is a linear combination of percent of surface area of skin affected by erythema, pustules, and scaling and the severity of erythema, pustules, and scaling (desquamation) over 4 body regions (head, trunk, upper limbs and lower limbs).

A higher score indicates a worse disease state, while a score of 0 indicates no disease. GPPASI 50 is based on the percent reduction from baseline, generally summarized as a dichotomous outcome based on achieving over an 50 % reduction.

Proportion of patients with GPPASI 50 at Week 4 is reported.

Change From Baseline in Psoriasis Symptom Scale (PSS) Score at Week 4Baseline and at Week 4.

PSS is a 4-item patient-reported outcome instrument that assesses the severity of psoriasis symptoms in moderate to severe psoriasis patients. The symptoms included are: pain, redness, itching, and burning. The symptom severity was assessed using a 5 point scale ranging from 0 to 4 where 0=none, 1=mild, 2=moderate, 3=severe, 4=very severe. The symptom scores are added to an unweighted total score (range: 0 to 16). A lower PSS score indicates a better outcome. Change from baseline =PSS score at Week 4 - PSS score at baseline. Death, any use of escape medication, OL Spesolimab at Day 8, or rescue medication with Spesolimab after Day 8, prior to observing the endpoint was considered to reflect a failure to achieve the endpoint outcome, i.e. non-response (NR). NR is not a missing value but the worst possible outcome of the endpoint. For example, if the achieved data is (NR, NR, NR, NR, NR, NR, 2, 3, 3, 3, 5) then Q1 is NR, median is NR and Q3 is 3.

Number of Patients With Treatment Emergent Adverse Events (TEAEs) up to Week 1From start of treatment until Day 7, up to 7 days.

TEAEs were all Adverse Events (AEs) occurring between start of treatment and Day 8 (Day 8 excluded). AEs that started before first drug intake and deteriorated under treatment were also considered as 'treatment-emergent'.

Trial Locations

Locations (37)

Tianjin Medical University General Hospital

🇨🇳

Tianjin, China

HOP Robert Debré

🇫🇷

Reims, France

Hedi Chaker Hospital, Department of Dermatology

🇹🇳

Tunisia, Tunisia

Huashan Hospital, Fudan University

🇨🇳

Shanghai, China

University of Alabama at Birmingham

🇺🇸

Birmingham, Alabama, United States

The First Hospital of Dalian Medical University

🇨🇳

Dalian, China

2nd Affiliated Hosp Zhejiang University College of Medical

🇨🇳

Hangzhou, China

Shanghai Skin Disease Hospital

🇨🇳

Shanghai, China

HOP Saint-André

🇫🇷

Bordeaux, France

Universitätsklinikum Essen AöR

🇩🇪

Essen, Germany

Nagoya City University Hospital

🇯🇵

Aichi, Nagoya, Japan

Asahikawa Medical University Hospital

🇯🇵

Hokkaido, Asahikawa, Japan

Hospital Sultan Ismail

🇲🇾

Johor Bahru, Malaysia

University of Miami

🇺🇸

Miami, Florida, United States

Universitätsklinikum Bonn AöR

🇩🇪

Bonn, Germany

HOP Saint-Louis

🇫🇷

Paris, France

Hospital Sultanah Aminah

🇲🇾

Johor Bahru, Malaysia

Hospital Pakar Sultanah Fatimah

🇲🇾

Muar, Malaysia

Severance Hospital

🇰🇷

Seoul, Korea, Republic of

University of South Florida

🇺🇸

Tampa, Florida, United States

Tohoku University Hospital

🇯🇵

Miyagi, Sendai, Japan

Hospital Raja Permaisuri Bainun

🇲🇾

Negeri Perak/Ipoh, Malaysia

Hospital Selayang

🇲🇾

Selangor, Malaysia

National University Hospital

🇸🇬

Singapore, Singapore

Charité - Universitätsmedizin Berlin

🇩🇪

Berlin, Germany

Klinikum der Universität München - Campus Innenstadt

🇩🇪

München, Germany

University Hospital of Lausanne

🇨🇭

Lausanne, Switzerland

Fukuoka University Hospital

🇯🇵

Fukuoka, Fukuoka, Japan

Tokyo Medical University Hachioji Medical Center

🇯🇵

Tokyo, Hachioji, Japan

Tokyo Medical University Hospital

🇯🇵

Tokyo, Shinjuku-ku, Japan

Hospital Kuala Lumpur

🇲🇾

Kuala Lumpur, Malaysia

Hospital Pulau Pinang

🇲🇾

Pulau Pinang, Malaysia

Farhat Hached Hospital

🇹🇳

Sousse, Tunisia

La Rabta Hospital

🇹🇳

Tunis, Tunisia

National Taiwan University Hospital

🇨🇳

Taipei, Taiwan

Ramathibodi Hospital

🇹🇭

Ratchatewi, Bangkok, Thailand

Icahn School of Medicine at Mount Sinai

🇺🇸

New York, New York, United States

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