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A PHASE I STUDY OF ALPS12 IN PATIENTS WITH EXTENSIVE STAGE SMALL CELL LUNG CANCER

Not Applicable
Not yet recruiting
Conditions
Extensive Stage Small Cell Lung Cancer
Interventions
Registration Number
NCT07107490
Lead Sponsor
Chugai Pharmaceutical
Brief Summary

This study is a phase I, open-label, multicenter trial designed to evaluate the safety, tolerability, pharmacokinetics, immunogenicity, and antitumor activity of ALPS12 in patients with extensive-stage small cell lung cancer. The study consists of two parts: a dose-escalation part and an expansion part.

Detailed Description

Not available

Recruitment & Eligibility

Status
NOT_YET_RECRUITING
Sex
All
Target Recruitment
122
Inclusion Criteria
  • Aged >18 years at time of informed consent
  • Eastern Cooperative Oncology Group (ECOG) Performance Status (PS) of 0 or 1
  • Histologically documented extensive stage small cell lung cancer
  • Disease recurrence documented after at least one prior systemic therapy.
  • Confirmed availability of representative archival tumor specimens or fresh tumor specimen.
  • Measurable disease per RECIST v.1.1.
  • Adequate hematologic and end organ function
Exclusion Criteria
  • Pregnant or breastfeeding, or intending to become pregnant or breastfeeding during the study
  • History or complication of clinically significant autoimmune disease
  • a positive HIV antibody test at screening
  • Active hepatitis B or hepatitis C
  • Prior treatment with anti-CD137 antibody drugs, anti-CD3 antibody drugs, and/or DLL3-targeted therapies
  • Patients who have received any investigational or approved anticancer therapy, including hormone therapy and/or radiotherapy, within 21 days prior to the first administration of the investigational drug.
  • History of Grade 4 immune-related adverse events caused by prior anti-PD-L1/PD-1 antibody drugs or anti-CTLA-4 antibody drugs (excluding asymptomatic elevations in serum amylase/lipase)
  • Patients who discontinued immunotherapy due to Grade 3 immune-related adverse events caused by prior anti-PD-L1/PD-1 antibody drugs or anti-CTLA-4 antibody drugs (excluding asymptomatic elevations in serum amylase/lipase), and/or patients who experienced Grade 3 immune-related adverse events caused by immunotherapy within 6 months prior to the first administration of the investigational drug
  • Patients who received a live attenuated vaccine within 4 weeks prior to the first administration of the investigational drug
  • History or clinical evidence of primary central nervous system (CNS) malignancy, symptomatic CNS metastases, CNS metastases requiring any anti tumor treatment, or leptomeningeal disease
  • Current or past CNS diseases (e.g., stroke, epilepsy, CNS vasculitis, neurodegenerative diseases)

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Dose escalation partALPS12Patients will receive ALPS12 as a single agent following pretreatment of obinutuzumab to determine the MTD by evaluating DLTs in patients with extensive stage small cell lung cancer.
Dose escalation partobinutuzumabPatients will receive ALPS12 as a single agent following pretreatment of obinutuzumab to determine the MTD by evaluating DLTs in patients with extensive stage small cell lung cancer.
Expansion partALPS12Patients will receive ALPS12 as a single agent following pretreatment of obinutuzumab to evaluate the antitumor effect.
Expansion partobinutuzumabPatients will receive ALPS12 as a single agent following pretreatment of obinutuzumab to evaluate the antitumor effect.
Primary Outcome Measures
NameTimeMethod
Dose Escalation part : Dose-limiting toxicities (DLTs) and PK profile of ALPS12[safety and tolerability]From Cycle 1 Day 1 to the administration of ALPS12 on Cycle 2 Day 1 (Cycle 1 is 21 days)

Nature and frequency of DLTs, AEs, PK and PD profiles

All part : Adverse events of ALPS12[safety and tolerability]From screening until study completion or treatment discontinuation, assessed up to the end of the study (approximate 42 months)

Incidence, nature, and severity of AEs graded according to National Cancer Institute (NCI) Common Terminology Criteria for Adverse Events (CTCAE) v.5.0, and CRS and Immune effector cell-associated neurotoxicity syndrome (ICANS) graded according to the ASTCT Consensus Grading Criteria

Dose Escalation part : Immunogenicity of ALPS12From screening until study completion or treatment discontinuation, assessed up to the end of the study (approximate 42 months)

Incidence of ADAs to ALPS12 and potential correlation with PK parameters and safety

Expansion part : Preliminary anti-tumor activity of ALPS12 when administered at selected dose(s) based on tumor assessment in patients with extensive stage SCLCFrom screening until study completion or treatment discontinuation, assessed up to the end of the study (approximate 42 months)

Objective response, defined as a confirmed complete response (CR) or partial response (PR) per Response Evaluation Criteria in Solid Tumors (RECIST) v.1.1, as determined by the Investigators

Secondary Outcome Measures
NameTimeMethod
Disease control [preliminary efficacy]From screening until study completion or treatment discontinuation, assessed up to the end of the study (approximate 42 months)

defined as the proportion of patients who have CR, PR, or stable disease (SD) as best overall response per RECIST v.1.1 as determined by the investigator.

Duration of response (DoR)[preliminary efficacy]From screening until study completion or treatment discontinuation, assessed up to the end of the study (approximate 42 months)

Duration of response (DoR), defined as the time from the first occurrence of CR or PR to progression disease (PD) or death from any cause (whichever occurs first), per the investigator according to RECIST v.1.1

Progression-free survival (PFS)[preliminary efficacy]From screening until study completion or treatment discontinuation, assessed up to the end of the study (approximate 42 months)

Progression-free survival (PFS), defined as the time from administration of first study treatment to the first occurrence of disease progression or death from any cause, as determined by the investigator according to RECIST v.1.1

Immunogenicity of obinutuzumabFrom screening until study completion or treatment discontinuation, assessed up to the end of the study (approximate 42 months)

Incidence of ADAs to obinutuzumab and potential correlation with PK parameters and safety

Maximum serum concentration (Cmax) and Area under the concentration time-curve (AUC) of ALPS12 with obinutuzumab[PK profile]From screening until study completion or treatment discontinuation, assessed up to the end of the study (approximate 42 months)

Serum ALPS12 concentration and its PK parameters including Cmax and AUC etc.

Adverse events of obinutuzumab[safety and tolerability]From screening until study completion or treatment discontinuation, assessed up to the end of the study (approximate 42 months)

Incidence, nature, and severity of adverse events graded according to NCI Common Terminology CTCAE v5.0, with severity of CRS determined according to the American Society for Transplantation and Cell Therapy (ASTCT) Consensus Grading Criteria(In parts with obinutuzumab premedication)

Overall survival (OS)[preliminary efficacy]From screening until study completion or treatment discontinuation, assessed up to the end of the study (approximate 42 months)

Overall survival (OS), defined as the time from administration of first study treatment to death from any cause

Objective response rate(ORR)[preliminary efficacy]From screening until study completion or treatment discontinuation, assessed up to the end of the study (approximate 42 months)

ORR assessed per RECIST v.1.1 by the investigators.

Trial Locations

Locations (1)

National Cancer Center Hospital East

🇯🇵

Kashiwa, Chiba, Japan

National Cancer Center Hospital East
🇯🇵Kashiwa, Chiba, Japan

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