MedPath

Masupirdine for the Treatment of Agitation in Dementia of the Alzheimer's Type

Phase 3
Recruiting
Conditions
Agitation
Alzheimer's Type Dementia
Interventions
Drug: Masupirdine 50 mg
Drug: Placebo
Drug: Masupirdine 100 mg
Registration Number
NCT05397639
Lead Sponsor
Suven Life Sciences Limited
Brief Summary

This study will be conducted to evaluate the efficacy, safety, tolerability, and pharmacokinetics of masupirdine compared to placebo for the treatment of agitation in participants with dementia of the Alzheimer's type.

Detailed Description

This is a multicenter, randomized, double-blind, placebo-controlled study, consisting of 12 weeks of treatment.

Approximately 375 participants will be enrolled at approximately 50 centers worldwide.

Study medication will be administered orally once-daily from Day 1 through Day 85. Screening will occur within approximately 4 weeks prior to randomization. Following screening procedures for assessment of inclusion and exclusion criteria, eligible participants will be randomized into the study.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
375
Inclusion Criteria
  • Has a diagnosis of dementia of the Alzheimer's type according to the National Institute on Aging-Alzheimer's Association (NIA-AA) criteria.
  • Has confirmed agitation using the IPA Consensus Provisional Definition of Agitation in Cognitive Disorders.
  • Has a score between 8 and 24 (both inclusive) on Mini-Mental State Examination (MMSE).
Exclusion Criteria
  • Participants with dementia predominantly of the non-Alzheimer's type (e.g., vascular dementia, parkinson's disease, lewy body disease, frontotemporal dementia)
  • Has symptoms of agitation that are not secondary to Alzheimer's disease (eg, pain, other psychiatric disorder, or delirium due to a metabolic disorder, systemic infection, or substance-induced).
  • Participant (or caregiver) is deemed otherwise ineligible for participation in this study in the investigator's judgement.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Low Dose Masupirdine ArmMasupirdine 50 mgTablet
PlaceboPlaceboTablet
High Dose Masupirdine ArmMasupirdine 100 mgTablet
Primary Outcome Measures
NameTimeMethod
Cohen-Mansfield Agitation Inventory (CMAI)From Baseline to Week 12 visit

Change in CMAI items score aligning to the International Psychogeriatric Association (IPA) agitation criteria domains (physical aggression, excessive motor activity, and verbal aggression). CMAI is a validated 29-item questionnaire to assess agitation. Each item is rated on a 7-point scale ranging from 1 "Never" to 7 "Several times per hour". Higher scores indicate worsening agitation.

Secondary Outcome Measures
NameTimeMethod
Modified Alzheimer's Disease Cooperative Study-Clinical Global Impression of Change (mADCS-CGI-C)From Baseline to Week 12 visit

Change in mADCS-CGI-C. The mADCS-CGI-C is a modification of the ADCS-CGI-C instrument that focuses specifically on agitation. It is a 7-point Likert scale that ranges from marked improvement scored as 1 to marked worsening scored as 7. The range is from 1 to 7. Higher scores indicate worsening agitation.

Trial Locations

Locations (51)

Centrum Medyczne Silmedic Sp z o o

๐Ÿ‡ต๐Ÿ‡ฑ

Katowice, Slaskie, Poland

Neuro-Medic Janusz Zbrojkiewicz

๐Ÿ‡ต๐Ÿ‡ฑ

Katowice, Slaskie, Poland

Ocean Medical Research

๐Ÿ‡บ๐Ÿ‡ธ

Toms River, New Jersey, United States

Military Medical Academy, Clinic of Neurology

๐Ÿ‡ท๐Ÿ‡ธ

Belgrade, Serbia

Clinical Hospital Center Rijeka

๐Ÿ‡ญ๐Ÿ‡ท

Rijeka, Croatia

Clinical Hospital Center Dragisa Misovic Dedinje

๐Ÿ‡ท๐Ÿ‡ธ

Belgrade, Serbia

Special Hospital for Psychiatric Diseases ''Dr Slavoljub Bakalovic''

๐Ÿ‡ท๐Ÿ‡ธ

Vrลกac, Serbia

Novel Clinical Research Center, LLC.

๐Ÿ‡บ๐Ÿ‡ธ

Miami, Florida, United States

Brainstorm Research

๐Ÿ‡บ๐Ÿ‡ธ

Miami, Florida, United States

University Clinical Center of Serbia, Clinic for neurology

๐Ÿ‡ท๐Ÿ‡ธ

Belgrade, Serbia

Advanced Research Center, Inc.

๐Ÿ‡บ๐Ÿ‡ธ

Anaheim, California, United States

Neurology Center of North Orange County

๐Ÿ‡บ๐Ÿ‡ธ

Fullerton, California, United States

ATP Clinical Research, Inc.

๐Ÿ‡บ๐Ÿ‡ธ

Costa Mesa, California, United States

Leading Edge Research LA, LLC

๐Ÿ‡บ๐Ÿ‡ธ

Encino, California, United States

Neuro Pain Medical Center

๐Ÿ‡บ๐Ÿ‡ธ

Fresno, California, United States

Mary S Easton Center for Alzheimer's Research and Care UCLA

๐Ÿ‡บ๐Ÿ‡ธ

Los Angeles, California, United States

Ki Health Partners, LLC

๐Ÿ‡บ๐Ÿ‡ธ

Stamford, Connecticut, United States

ClinCloud, LLC

๐Ÿ‡บ๐Ÿ‡ธ

Maitland, Florida, United States

Allied Biomedical Research Institute

๐Ÿ‡บ๐Ÿ‡ธ

Miami, Florida, United States

Central Miami Medical Institute

๐Ÿ‡บ๐Ÿ‡ธ

Miami, Florida, United States

CCM Clinical Research Group

๐Ÿ‡บ๐Ÿ‡ธ

Miami, Florida, United States

Miami Jewish Health

๐Ÿ‡บ๐Ÿ‡ธ

Miami, Florida, United States

Quantum Laboratories Inc

๐Ÿ‡บ๐Ÿ‡ธ

Pompano Beach, Florida, United States

Re:Cognition Health

๐Ÿ‡บ๐Ÿ‡ธ

Fort Worth, Texas, United States

Insight Hospital and Medical Center Chicago

๐Ÿ‡บ๐Ÿ‡ธ

Chicago, Illinois, United States

Dent Neurologic Institute

๐Ÿ‡บ๐Ÿ‡ธ

Amherst, New York, United States

Velocity Clinical Research, Syracuse

๐Ÿ‡บ๐Ÿ‡ธ

East Syracuse, New York, United States

Velocity Clinical Research, Cleveland

๐Ÿ‡บ๐Ÿ‡ธ

Beachwood, Ohio, United States

Baylor College of Medicine

๐Ÿ‡บ๐Ÿ‡ธ

Houston, Texas, United States

Midlands Neurology and Pain Associates

๐Ÿ‡บ๐Ÿ‡ธ

Columbia, South Carolina, United States

Gadolin Research

๐Ÿ‡บ๐Ÿ‡ธ

Beaumont, Texas, United States

Clinical Trial Network

๐Ÿ‡บ๐Ÿ‡ธ

Houston, Texas, United States

Polyclinic Neuron

๐Ÿ‡ญ๐Ÿ‡ท

Zagreb, Croatia

Klinika za psihijatriju Sveti Ivan

๐Ÿ‡ญ๐Ÿ‡ท

Zagreb, Croatia

University Hospital Center Zagreb

๐Ÿ‡ญ๐Ÿ‡ท

Zagreb, Croatia

Klinika za psihijatriju Vrapce

๐Ÿ‡ญ๐Ÿ‡ท

Zagreb, Croatia

EMC Instytut Medyczny S.A.

๐Ÿ‡ต๐Ÿ‡ฑ

Wrocล‚aw, Dolnoslaskie, Poland

Clinical Best Solutions - Lublin

๐Ÿ‡ต๐Ÿ‡ฑ

Lublin, Lubelskie, Poland

Medycyna Milorzab sp. z o.o.

๐Ÿ‡ต๐Ÿ‡ฑ

ลรณdลบ, Lรณdzkie, Poland

FutureMeds Warszawa Centrum

๐Ÿ‡ต๐Ÿ‡ฑ

Warszawa, Mazowieckie, Poland

Osrodek Badan Klinicznych Appletreeclinics

๐Ÿ‡ต๐Ÿ‡ฑ

ลรณdลบ, Lรณdzkie, Poland

MTZ Clinical Research powered by Pratia

๐Ÿ‡ต๐Ÿ‡ฑ

Warszawa, Mazowieckie, Poland

EMC Silesia Sp. z o.o.

๐Ÿ‡ต๐Ÿ‡ฑ

Katowice, Slaskie, Poland

Centrum Leczenia Zaburzen Pamieci Affidea

๐Ÿ‡ต๐Ÿ‡ฑ

Warszawa, Mazowieckie, Poland

Special Hospital for Psychiatric Diseases

๐Ÿ‡ท๐Ÿ‡ธ

Kovin, Serbia

University Clinical Center Kragujevac, Clinic for Psychiatry

๐Ÿ‡ท๐Ÿ‡ธ

Kragujevac, Serbia

University Clinical Center Nis, Clinic for neurology

๐Ÿ‡ท๐Ÿ‡ธ

Niลก, Serbia

Clinical Centre of Vojvodina, Clinic of Neurology

๐Ÿ‡ท๐Ÿ‡ธ

Novi Sad, Serbia

Regional Neurological Associates

๐Ÿ‡บ๐Ÿ‡ธ

Bronx, New York, United States

Combined Research Orlando Phase I-IV

๐Ÿ‡บ๐Ÿ‡ธ

Orlando, Florida, United States

Ralph H. Johnson VA Health Care System

๐Ÿ‡บ๐Ÿ‡ธ

Charleston, South Carolina, United States

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