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Study of Chemotherapy in Combination With IDO Inhibitor in Metastatic Breast Cancer

Phase 2
Completed
Conditions
Metastatic Breast Cancer
Interventions
Registration Number
NCT01792050
Lead Sponsor
NewLink Genetics Corporation
Brief Summary

The purpose of this study is to compare the effects, good and/or bad, of standard of care therapy (docetaxel or paclitaxel) with or without the addition of 1-Methyl-D-tryptophan (referred to as indoximod) an experimental drug to find out which treatment is better.

Detailed Description

It is estimated that 232,340 US women will be diagnosed with and 40,030 women will die of breast cancer in 2013. Metastatic breast cancer is a terminal condition and treatments are palliative in nature. The median survival for patients with metastatic breast cancer is approximately 2.5 years. The standard therapies currently in use include anti-estrogen therapies (anastrazole, letrozole, fulvestrant, tamoxifen), chemotherapy agents (taxanes, capecitabine, navelbine, gemcitabine, eribulin, ixabepilone), targeted therapies (trastuzumab, lapatinib), and supportive care agents (zolendronic acid, denosumab). While breast cancer typically responds well to treatment, the response is transient and their disease becomes more refractory with continued therapy. Also, quality of life is a significant issue for these patients as many of these therapies are associated with significant side effects. Well tolerated, novel agents which improve the efficacy of existing chemotherapy agents would prove quite useful in managing metastatic breast cancer.

Preclinical data derived from MMTV-Neu mice with autochthonous tumors studied the interaction between indoximod and various chemotherapeutic agents. Mice with 5-10mm tumors were enrolled into control and treatment groups. Mice were treated with indoximod alone, chemotherapy alone (paclitaxel, doxorubicin, cyclophosphamide, and others), and the combination of indoximod and chemotherapy. treatment with indoximod or paclitaxel alone caused retardation of tumor growth in this model but no regressions were seen. the combination of indoximod plus paclitaxel caused 30% tumor regression and histologically there was significantly enhanced tumor cell death with the combination versus either agent alone. This synergism was abrogated when the mice underwent CD4+ T cell depletion prior to treatment with the combination, suggesting the immune response played a role in the observed effect. Based on this data and other reports suggesting systemic immunomodulating drugs like indoximod can synergize with chemotherapy agents such as taxanes, the decision was made to devise this combination of therapy of docetaxel or paclitaxel with indoximod in metastatic breast cancer.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
169
Inclusion Criteria
  • Histologically or cytologically confirmed estrogen/progesterone receptors (ER/PR) +/-; human epidermal growth factor receptor 2 (HER2)-, metastatic breast cancer.
  • Metastatic disease that is evaluable on imaging. May have measureable disease, defined as at least one lesion that can be accurately measured in at least one dimension (longest diameter to be recorded for non-nodal lesions and short axis for nodal lesions) as ≥20 mm with conventional techniques or as ≥10 mm with spiral CT scan, MRI, or calipers by clinical exam. Patients can also have non-measurable disease including bone only metastatic disease, evaluated by bone scan, PET or MRI.
  • Any number of prior endocrine therapies in the metastatic setting are allowed. The patient must not have received any prior chemotherapy agents in the metastatic setting. Prior treatment with adjuvant docetaxel or paclitaxel is allowed if disease relapse occurred greater than 12 months from the completion of adjuvant therapy.
  • Age ≥18 years.
  • Eastern Cooperative Oncology Group (ECOG) performance status ≤1 (Karnofsky ≥60%).
  • Life expectancy of greater than 4 months.
  • Patients must have normal organ and marrow function as defined below: leukocytes ≥3,000/mcL, absolute neutrophil count ≥1,500/mcL, platelets ≥100,000/mcL, total bilirubin within normal institutional limits, aspartate aminotransferase AST(SGOT)/ alanine aminotransferase ALT(SGPT) ≤2.5 X institutional upper limit of normal, creatinine within normal institutional limits OR creatinine clearance ≥60 mL/min/1.73 m^2 for patients with creatinine levels above institutional normal.
  • Patients with known brain metastases will only be eligible after their tumors have been treated with definitive resection and/or radiotherapy and they are neurologically stable for at least 1 month off steroids.
  • Male and female subjects of child producing potential must agree to use adequate forms of contraception or avoidance of pregnancy measures prior to study entry, while enrolled on study and for a minimum of one month after completion of the study.
  • Ability to understand and the willingness to sign a written informed consent document.
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Exclusion Criteria
  • Patients who have had chemotherapy for the treatment of metastatic breast cancer are not eligible. Patients who have had radiotherapy within 3 weeks prior to entering the study or those who have not recovered from adverse events due to agents administered more than 3 weeks earlier are not eligible.
  • Patients who are currently receiving any other investigational agents.
  • Patients with known active, untreated brain metastases should be excluded from this clinical trial. Those with previously treated inactive brain metastases with no evidence of active disease documented on brain MRI at least 4 weeks after radiation and off all steroids may be eligible.
  • History of allergic reactions attributed to compounds of similar chemical or biologic composition to docetaxel or tryptophan containing substances. This would include L-tryptophan or 5-hydroxy-tryptophan supplements. Also patients with a history of severe hypersensitivity reactions to docetaxel or to other drugs formulated with polysorbate 80 are excluded.
  • Uncontrolled intercurrent illness including, but not limited to, ongoing or active infection, symptomatic congestive heart failure, unstable angina pectoris, cardiac arrhythmia, or psychiatric illness/social situations that would limit compliance with study requirements.
  • Pregnant women are excluded from this study because indoximod is an immunoregulatory agent with the potential for abortifacient effects due to fetal rejection by the maternal immune system. Because there is an unknown but potential risk for adverse events in nursing infants secondary to treatment of the mother with indoximod, breastfeeding should be discontinued if the mother is treated with indoximod. Also, docetaxel and paclitaxel are category D cytotoxic agents and are not administered to pregnant females.
  • Known HIV-positive patients and those with other acquired/inherited immunodeficiencies are ineligible due to the possibility of affecting the response to indoximod and the higher risk of active opportunistic infections.
  • Patients with more than one active malignancy at the time of enrollment.
  • Patients who have received any prior experimental active immunotherapy consisting of targeted monoclonal antibodies (ipilimumab) or pharmaceutical compounds are excluded.
  • Patients with any active autoimmune disease (i.e. psoriasis, extensive atopic dermatitis, asthma, inflammatory bowel disease (IBD), multiple sclerosis (M.S.), uveitis, vasculitis), chronic inflammatory condition, or any condition requiring concurrent use of any systemic immunosuppressants or steroids for any reason would be excluded from the study. Any patient with an allo-transplant of any kind would be excluded as well. This would include those with a xenograft heart valve to avoid the potential risk of any immune reaction causing valvular degeneration. Mild-intermittent asthma requiring only occasional beta-agonist inhaler use or mild localized eczema will not be excluded.
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Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Arm 1A: Docetaxel + PlaceboPlaceboArm 1A: Docetaxel 75 mg/m\^2 IV given every 3 weeks (on day 8 of 21 day cycle), plus placebo PO BID (days 1-14 of 21 day cycle).
Arm 2A: Paclitaxel + PlaceboPlaceboArm 2A: Paclitaxel 80 mg/m\^2 IV given weekly x3 followed by a week of rest (28 day cycle), plus placebo PO BID (days 1-21 of 28 day cycle).
Arm 1A: Docetaxel + PlaceboDocetaxelArm 1A: Docetaxel 75 mg/m\^2 IV given every 3 weeks (on day 8 of 21 day cycle), plus placebo PO BID (days 1-14 of 21 day cycle).
Arm 1B: Docetaxel + IndoximodDocetaxelArm 1B: Docetaxel 75 mg/m\^2 IV given every 3 weeks (on day 8 of 21 day cycle), plus Indoximod 1200 mg PO BID (days 1-14 of 21 day cycle).
Arm 1B: Docetaxel + IndoximodIndoximodArm 1B: Docetaxel 75 mg/m\^2 IV given every 3 weeks (on day 8 of 21 day cycle), plus Indoximod 1200 mg PO BID (days 1-14 of 21 day cycle).
Arm 2A: Paclitaxel + PlaceboPaclitaxelArm 2A: Paclitaxel 80 mg/m\^2 IV given weekly x3 followed by a week of rest (28 day cycle), plus placebo PO BID (days 1-21 of 28 day cycle).
Arm 2B: Paclitaxel + IndoximodIndoximodArm 2B: Paclitaxel 80 mg/m\^2 IV given weekly x3 followed by a week of rest (28 day cycle), plus Indoximod 1200 mg PO BID (days 1-21 of 28 day cycle).
Arm 2B: Paclitaxel + IndoximodPaclitaxelArm 2B: Paclitaxel 80 mg/m\^2 IV given weekly x3 followed by a week of rest (28 day cycle), plus Indoximod 1200 mg PO BID (days 1-21 of 28 day cycle).
Primary Outcome Measures
NameTimeMethod
Progression Free Survival12 months

The primary objective of this phase 2 study is the progression free survival of docetaxel or paclitaxel in combination with indoximod compared to docetaxel or paclitaxel plus placebo in metastatic breast cancer.

Secondary Outcome Measures
NameTimeMethod
Correlation of clinical and pathologic variables and clinical benefit (progression free survival rate) from treatment12 months

A secondary objective of this phase 2 study is determining the correlation between clinical and pathologic variables and clinical benefit from docetaxel or paclitaxel and indoximod.

Objective Response Rate (Complete Response + Partial Response)12 Months

A secondary objective is to determine the objective response rate (CR+PR) as measured by Response Evaluation Criteria in Solid Tumors (RECIST 1.1) of docetaxel or paclitaxel + indoximod compared to docetaxel or paclitaxel plus placebo.

Median Overall Survival12 months

A secondary objective of this phase 2 study is to observe median overall survival of all patients.

Frequency and grade of adverse events of docetaxel and paclitaxel in combination with indoximod versus docetaxel alone12 months

A secondary objective of this phase 2 study is to determine the safety/toxicity (frequency and grade of adverse events) of docetaxel or paclitaxel in combination with indoximod versus docetaxel or paclitaxel plus placebo.

Trial Locations

Locations (31)

Research Site

🇵🇱

Warsaw, Poland

University of North Carolina

🇺🇸

Chapel Hill, North Carolina, United States

University of Virginia

🇺🇸

Charlottesville, Virginia, United States

University of Florida Health Cancer Center

🇺🇸

Gainesville, Florida, United States

University Cancer & Blood Center, LLC

🇺🇸

Athens, Georgia, United States

Illinois Cancer Specialists

🇺🇸

Arlington Heights, Illinois, United States

H. Lee Moffitt Cancer Center and Research Institute

🇺🇸

Tampa, Florida, United States

Wake Forest Baptist Hospital

🇺🇸

Winston-Salem, North Carolina, United States

Georgia Regents University

🇺🇸

Augusta, Georgia, United States

Indiana University Health Goshen Center for Cancer Care

🇺🇸

Goshen, Indiana, United States

University of Iowa Hospitals and Clinics

🇺🇸

Iowa City, Iowa, United States

Fairview Hospital

🇺🇸

Cleveland, Ohio, United States

Cleveland Clinic - Taussig Cancer Center

🇺🇸

Cleveland, Ohio, United States

Taussig Cancer Institute

🇺🇸

Mayfield Heights, Ohio, United States

Peninsula Cancer Center

🇺🇸

Newport News, Virginia, United States

Research SiteR

🇵🇱

Brzozow, Poland

Virginia Commonwealth University

🇺🇸

Richmond, Virginia, United States

Aurora Baycare

🇺🇸

Green Bay, Wisconsin, United States

Reserach Site

🇵🇱

Konin, Poland

Wheaton Franciscan Healthcare- Reiman Cancer Center

🇺🇸

Franklin, Wisconsin, United States

Space Coast Cancer Center

🇺🇸

Titusville, Florida, United States

Cleveland Clinic - Florida

🇺🇸

Weston, Florida, United States

Eastchester Center for Cancer Care

🇺🇸

Bronx, New York, United States

Pennsylvania State University Milton S. Hershey Medical Center

🇺🇸

Hershey, Pennsylvania, United States

Paoli Hospital

🇺🇸

Paoli, Pennsylvania, United States

MD Anderson Cancer Center

🇺🇸

Houston, Texas, United States

Lynchburg Hematology Oncology

🇺🇸

Lynchburg, Virginia, United States

Bryn Mawr Hospital

🇺🇸

Bryn Mawr, Pennsylvania, United States

University of Illinois Cancer Center

🇺🇸

Chicago, Illinois, United States

University of Tennessee Medical Center

🇺🇸

Knoxville, Tennessee, United States

Lankenau Medical Center

🇺🇸

Wynnewood, Pennsylvania, United States

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