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To Compare the Safety, Tolerability, and Pharmacokinetics of QBX258 in Patients With Asthma

Phase 1
Completed
Conditions
Asthma
Interventions
Drug: VAK694 placebo
Drug: QAX576 placebo
Registration Number
NCT01568762
Lead Sponsor
Novartis Pharmaceuticals
Brief Summary

This study is designed to compare the safety, tolerability, and pharmacokinetics of QBX258 (sequential administration of a fixed dose of VAK694 and single ascending doses of QAX576) in patients with well-controlled mild to moderate asthma.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
50
Inclusion Criteria
  • Male and female subjects age 18-60 years (inclusive)
  • Well controlled mild to moderate atopic asthma
  • Female subjects must be post-menopausal or surgically sterile
  • Male subjects must be using two methods of contraception
  • Subjects must have a positive skin prick test to one or more common airborne allergen
Exclusion Criteria
  • Participation in any clinical investigation or use of other investigational drugs at time of enrollment
  • A history of clinically significant ECG abnormalities
  • History of malignancy of any organ system
  • Smokers (use of tobacco products in the previous 3 months)
  • Use of prescription drugs other than those required for control and relief of asthma
  • Use of oral steroids within 12 weeks prior to dosing
  • FEVI < 80% predicted at screening or baseline
  • Use of albuterol more than twice a week for relief of asthma
  • Patients suffering from active hay fever at baseline or likely to require treatment during the study
  • History of chronic respiratory disease other than asthma or chronic allergic rhinitis
  • Emergency room visit within 6 weeks of screening due to asthma
  • Hospitalization for asthma in the last year
  • History of intubation/assisted ventilation for asthma in the last 5 years
  • Administration of live vaccines within the preceding month

Other protocol-defined inclusion/exclusion criteria may apply.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
VAK694 PlaceboVAK694 placeboVAK694 placebo was administered as a one hour intravenous infusion
QAX576QAX576QAX576 was administered intravenously as a 2 hour infusion
QAX576 placeboQAX576 placeboQAX576 placebo was administered as a 2 hour intravenous infusion
VAK694VAK694VAK694 was administered as a 1 hour intravenous infusion
Primary Outcome Measures
NameTimeMethod
Number of patients with adverse events100 days

Adverse events will be determined by evaluating clinical, laboratory evaluations, impact on vital signs and impacts on ECGs

Secondary Outcome Measures
NameTimeMethod
Concentration of serum anti-VAK694 antibodiesPre-dose, Day 71, 85 and 100

Blood will be collected to determine concentrations if anti-VAK964 antibodies

Concentration of serum anti-QAX576 antibodiesPre-dose, Day 71, 85 and 100

Blood will be collected to determine concentrations if anti-QAX576 antibodies

Area under the serum concentration curve for VAK694Pre-dose, 1, 2, 4, 11, 24, 48, 96 hours and Days 8, 15, 29, 43, 57, 71, 85, 100

Blood will be collected for the measurement of VAK694 serum concentrations

Area under the serum concentration curve for QAX576Pre-dose, 1, 2, 4, 11, 24, 48, 96 hours and Days 8, 15, 29, 43, 57, 71, 85, 100

Blood will be collected for the measurement of QAX576 concentrations

Change in interleukin concentrationsPre-dose, 1, 2, 4, 11, 24, 48, 96 hours and Days 8, 15, 29, 43, 57, 71, 85, 100

Blood samples will be collected to measure interleukin concetrations.

Trial Locations

Locations (1)

Novartis Investigative Site

🇺🇸

Raleigh, North Carolina, United States

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