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Study to Evaluate the Efficacy and Safety of Oral Difelikefalin for Moderate to Severe Pruritus in Subjects With Notalgia Paresthetica

Phase 2
Terminated
Conditions
Pruritus
Notalgia Paresthetica
Interventions
Registration Number
NCT05978063
Lead Sponsor
Cara Therapeutics, Inc.
Brief Summary

This is a 2-part, multicenter, randomized, double-blind, placebo-controlled study to evaluate the efficacy and safety of twice-daily (BID) oral difelikefalin for moderate-to-severe pruritus in adult subjects with NP.

Detailed Description

Part A of this study will evaluate the benefit-risk of 3 doses of difelikefalin compared to placebo. The dose with the best benefit-risk profile will be further evaluated in Part B. Part A of this study comprises a 28-day Screening Period, a 7-day Run-in Period, an 8-week Double-blind Treatment Period, a 2-week Treatment Discontinuation Period, and a Safety Follow-up Visit (14 days after the last dose of study treatment).

Part B of this study will evaluate the efficacy, safety, and tolerability of oral difelikefalin. The dose of oral difelikefalin to be assessed in Part B will depend on the results of Part A. Part B of this study comprises a 28-day Screening Period, a 7-day Run-in Period, an 8-week Double-blind Treatment Period, up to a 52-week OLE Period, and a Safety Follow-up Visit.

Subjects who participated in Part A of the study may not participate in Part B.

All subjects will sign an informed consent form (ICF) and undergo screening for study eligibility.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
214
Inclusion Criteria

To be eligible for inclusion into the study, a patient must meet the following criteria:

  • Subject has clinically confirmed diagnosis of active Notalgia Paresthetica;
  • Subject has a history of chronic pruritus due to Notalgia Paresthetica;
  • Subject has moderate to severe pruritus;
  • Female subject is not pregnant or nursing during any period of the study.

Key

Exclusion Criteria

A patient will be excluded from the study if any of the following criteria are met:

  • Subject has pruritus attributed to a cause other than Notalgia Paresthetica;
  • Subject has any clinically significant medical condition or physical/laboratory/ECG/vital signs abnormality that would, in the opinion of the investigator, put the subject at undue risk or interfere with interpretation of study results.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Difelikefalin 2.0 mg tabletsdifelikefalin 2.0 mg tabletsOral difelikefalin 2.0 mg tablet administered twice daily
Difelikefalin 0.25 mg tabletsdifelikefalin 0.25 mg tabletsOral difelikefalin 0.25 mg tablet administered twice daily
Difelikefalin 1.0 mg tabletsdifelikefalin 1.0 mg tabletsOral difelikefalin 1.0 mg tablet administered twice daily
Placebo tabletsPlacebo tabletsOral placebo tablet administered twice daily
Primary Outcome Measures
NameTimeMethod
Proportion of subjects achieving ≥4-point improvement from baseline in the weekly mean of the daily 24-hour I-NRS scoreBaseline, Week 8
Secondary Outcome Measures
NameTimeMethod
Proportion of subjects achieving ≥4-point improvement from baseline in the weekly mean of the daily 24-hour I-NRS score at Week 4 in Part BBaseline, Week 4
Proportion of subjects achieving ≥4-point improvement from baseline in the weekly mean of the daily 24-hour I-NRS score at Week 2 in Part BBaseline, Week 2
Change from Baseline in the Numeric Rating Scale of Burning Sensation and Skin Tingling at Week 8 in Part BBaseline, Week 8
Proportion of Subjects with H-IGA of Clear or Almost Clear at Week 8 in Part BWeek 8
Proportion of ≥4-point Improvement in Daily I-NRS at Day 2 in Part BDay 2
Proportion of subjects achieving ≥4-point improvement from baseline in the weekly mean of the daily 24-hour I-NRS score at Week 1 in Part BBaseline, Week 1

Trial Locations

Locations (2)

Cara Therapeutics Study Site

🇪🇸

Madrid, Spain

Cara Therapeutics Study Site 2

🇵🇱

Katowice, Poland

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