MedPath

TEPEZZA® (Teprotumumab-trbw) Post-Marketing Requirement Study

Phase 4
Active, not recruiting
Conditions
Thyroid Eye Disease
Interventions
Drug: Placebo
Registration Number
NCT05002998
Lead Sponsor
Amgen
Brief Summary

This is a double-masked, randomized, parallel-assignment, multicenter trial examining the safety and tolerability of teprotumumab in the treatment of Thyroid Eye Disease (TED) in adult participants. This international, Phase 3b/4 trial is being conducted to fulfill an FDA post-marketing requirement for a descriptive trial to evaluate the safety, efficacy and need for re-treatment of 3 different teprotumumab treatment durations for TED. In addition, serum samples from participants with a Baseline Clinical Activity Score (CAS) ≥3 will be evaluated for biomarkers of disease.

Detailed Description

Participants will be screened for eligibility within 4 weeks prior to the Baseline (Day 1) Visit. Approximately 300 participants who meet the trial eligibility criteria will be randomized on Day 1 in a 1:1:1 ratio in a double-masked fashion (stratified by CAS(clinical activity score) \[≥3 (active) or \<3 (inactive)\] and disease severity \[severe disease, defined as both proptosis above normal for race and gender with binocular diplopia at Baseline vs. non-severe disease\]) to receive:

* 4 infusions of teprotumumab (10 mg/kg for the first infusion and 20 mg/kg for the remaining 3 infusions) (Cohort 1) followed by 4 infusions of:

* Placebo if a participants is a treatment responder at Week 12 or

* Teprotumumab 20 mg/kg if a participant is a treatment non-responder at Week 12

* 8 infusions of teprotumumab (10 mg/kg for the first infusion and 20 mg/kg for the remaining 7 infusions) (Cohort 2)

* 16 infusions of teprotumumab (10 mg/kg for the first infusion and 20 mg/kg for the remaining 15 infusions) (Cohort 3)

Three weeks following the final infusion of the Initial Treatment Period, there will be a comprehensive End-of-Initial Treatment Visit at Week 24 (Cohorts 1 and 2)/Week 48 (Cohort 3). At this visit, all participants will be assessed for treatment response.

Proptosis responders in all cohorts and non-responders in Cohorts 1 and 2 who choose not to receive a second treatment course, will enter a 52 week Initial Follow-up Period.

Proptosis non-responders in Cohorts 1 and 2 who choose to receive a second treatment course (8 infusions) of teprotumumab will receive an infusion q3W.

Proptosis non-responders in Cohort 3 are not eligible for a second treatment course following initial treatment.

Participants in any of the 3 cohorts who are proptosis responders following the Initial Treatment Period and who flare during the Initial Follow up Period will be eligible to receive re treatment.

Acquired from Horizon in 2024

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
All
Target Recruitment
313
Inclusion Criteria
  1. Written informed consent.
  2. Male or female between the ages of 18 and 80 years, inclusive, at Screening.
  3. Initial diagnosis of TED within 7 years prior to Screening.
  4. Proptosis ≥3 mm from baseline (prior to diagnosis of TED), as estimated by treating physician, and/or proptosis >3 mm above normal for race and gender.
  5. Participants must be euthyroid with the baseline disease under control or have mild hypo or hyperthyroidism (defined as free thyroxine and free triiodothyronine levels <50% above or below the normal limits) at Screening. Every effort should be made to correct the mild hypo- or hyperthyroidism promptly and to maintain the euthyroid state for the duration of the trial.
  6. Does not require immediate surgical ophthalmological intervention and is not planning corrective surgery/irradiation during the course of the trial.
  7. Diabetic participants must have HbA1c ≤8.0% at Screening.
  8. Participants with a history of IBD (ulcerative colitis or Crohn's disease)
Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Teprotumumab 4 InfusionsPlacebo• 4 infusions of teprotumumab (10 mg/kg for the first infusion and 20 mg/kg for the remaining 3 infusions) (Cohort 1) followed by 4 infusions of: * Placebo if a participant is a treatment responder at Week 12 or * Teprotumumab 20 mg/kg if a participant is a treatment non-responder at Week 12
Teprotumumab 4 InfusionsTeprotumumab• 4 infusions of teprotumumab (10 mg/kg for the first infusion and 20 mg/kg for the remaining 3 infusions) (Cohort 1) followed by 4 infusions of: * Placebo if a participant is a treatment responder at Week 12 or * Teprotumumab 20 mg/kg if a participant is a treatment non-responder at Week 12
Teprotumumab 8 InfusionsTeprotumumab8 infusions of teprotumumab (10 mg/kg for the first infusion and 20 mg/kg for the remaining 7 infusions) (Cohort 2)
Teprotumumab 16 InfusionsTeprotumumab16 infusions of teprotumumab (10 mg/kg for the first infusion and 20 mg/kg for the remaining 15 infusions) (Cohort 3)
Primary Outcome Measures
NameTimeMethod
Percentage of Participants who experience at least 1 treatment-emergent adverse event (TEAE) and the percentage of participants who experience at least 1 treatment emergent AESI during treatment with teprotumumabScreening to End of Study (last visit possible is Week 136)

Treatment emergent adverse events and treatment emergent adverse events of special interest will be evaluated from the beginning of the study until follow up.

Percentage of Participants who receive re-treatmentWeek 27 to Week 136

Participants who are not proptosis responders after initial treatment or participants who are proptosis responders after initial treatment but who have flared during follow-up (relapsed).

Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (29)

The Private Practice of Raymond Douglas, MD - Beverly Hills

🇺🇸

Beverly Hills, California, United States

University of Colorado - Eye Center - PPDS

🇺🇸

Aurora, Colorado, United States

Mayo Clinic - PPDS

🇺🇸

Rochester, Minnesota, United States

Washington University

🇺🇸

Saint Louis, Missouri, United States

Hospices Civils de Lyon - Hôpital Louis Pradel

🇫🇷

Bron, Rhône, France

Hôpital Claude Huriez-Lille-Rue Michel Polonovski

🇫🇷

Lille, France

ARNAS Garibaldi - PO Garibaldi-Centro

🇮🇹

Catania, Sicilia, Italy

Azienda Ospedaliero Universitaria Pisana - Stabilimento Santa Chiara

🇮🇹

Pisa, Toscana, Italy

Hospital Universitario Ramon y Cajal

🇪🇸

Madrid, Spain

Royal Victoria Infirmary

🇬🇧

Newcastle Upon Tyne, Tyne And Wear, United Kingdom

Southampton University Hospitals NHS Trust

🇬🇧

Southampton, United Kingdom

USC Roski Eye Institute - Los Angeles

🇺🇸

Los Angeles, California, United States

Stanford University

🇺🇸

Palo Alto, California, United States

Bascom Palmer Eye Institute

🇺🇸

Miami, Florida, United States

Casey Eye Institute - OHSU

🇺🇸

Portland, Oregon, United States

Hopital Jean Minjoz

🇫🇷

Besançon, Doubs, France

Centre Hospitalier National D'ophtalmologie Des Quinze Vingts

🇫🇷

Paris, France

Universitätsklinikum Tübingen

🇩🇪

Tübingen, Baden-Württemberg, Germany

University Medicine Göttingen Germany

🇩🇪

Göttingen, Niedersachsen, Germany

Universitätsmedizin der Johannes Gutenberg-Universität Mainz

🇩🇪

Mainz, Rheinland-Pfalz, Germany

Universitätsklinikum Essen

🇩🇪

Essen, Germany

Universitätsklinikum Münster

🇩🇪

Münster, Germany

Azienda Ospedaliera Universitaria Federico II

🇮🇹

Napoli, Campania, Italy

ASST dei Sette Laghi - Ospedale Di Circolo E Fondazione Macchi

🇮🇹

Varese, Lombardia, Italy

Hospital La Arruzafa

🇪🇸

Cordoba, Córdoba, Spain

Hospital Universitario Virgen Macarena

🇪🇸

Sevilla, Spain

Moorfields Eye Hospital

🇬🇧

London, London, City Of, United Kingdom

Imperial College Healthcare NHS Trust

🇬🇧

London, London, City Of, United Kingdom

University Hospital of Cardiff

🇬🇧

Cardiff, South Glamorgan, United Kingdom

© Copyright 2025. All Rights Reserved by MedPath