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A Study to Evaluate the Effect of Injection Site on PK of Astegolimab in Healthy Subjects

Phase 1
Completed
Conditions
Healthy Volunteers
Interventions
Registration Number
NCT06462118
Lead Sponsor
Genentech, Inc.
Brief Summary

The main objective is to study how astegolimab may behave in the body when injected subcutaneously into the abdomen, thigh, or upper arm in healthy participants.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
78
Inclusion Criteria
  • Body weight of ≥50 kg to ≤110 kg with body mass index (BMI) range 18.0 to 30.0 kg/m2 (inclusive) at screening
Exclusion Criteria
  • History of significant hypersensitivity or severe allergic reaction, including anaphylaxis, to any drug compound, food, or other substance
  • Any immunization or vaccination 14 days prior to the Check-in (Day -1) or plans to obtain any immunization or vaccination within 30 days after the Check-in
  • Any surgical procedure (except for minor surgeries) within 28 days prior to initiation of study treatment, or anticipation of need for a major surgical procedure during the study
  • Donation of blood from 30 days prior to screening through study completion or end of trial, inclusive, or of plasma from 2 weeks prior to screening through study completion or end of trial, inclusive
  • History of immunodeficiency, including but not limited to, human immunodeficiency virus (HIV) infection
  • History of active or untreated latent tuberculosis
  • History of malignancy within 5 years prior to screening, except for appropriately treated carcinoma in situ of the cervix, non-melanoma skin carcinoma, or Stage I uterine cancer
  • Unstable cardiac disease, myocardial infarction, or New York Heart Association Class 3 or 4 heart failure within 12 months prior to screening
  • History or presence of clinically significant ECG abnormalities at screening or check-in (Day -1)
  • Positive for Hepatitis B or Hepatitis C (HCV)
  • Tattoo(s) or scarring at or near the site of injection (abdomen, front and middle thigh, or upper arm) or any other condition which may interfere with the injection site examination (as determined by the Investigator)

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Treatment AAstegolimabParticipants will receive one subcutaneous (SC) dose in the abdomen.
Treatment BAstegolimabParticipants will receive one subcutaneous (SC) dose in the thigh.
Treatment CAstegolimabParticipants will receive one subcutaneous (SC) dose in the upper arm.
Primary Outcome Measures
NameTimeMethod
Maximum serum concentration (Cmax) of astegolimabApproximately 85 days
Area under the curve from Hour 0 to the time of last measurable concentration (AUC0-t) of astegolimabApproximately 85 days
AUC extrapolated to infinity (AUC0-infinity) of astegolimabApproximately 85 days
Secondary Outcome Measures
NameTimeMethod
Incidence of anti-drug antibodies (ADAs)Approximately 85 days
Relative bioavailability (F%) for thigh injection of astegolimabApproximately 85 days
Apparent volume of distribution during the terminal elimination phase (Vz/F) of astegolimabApproximately 85 days
Time to maximum serum concentration (Tmax) of astegolimabApproximately 85 days
F% for upper arm injection of astegolimabApproximately 85 days
Half-life (T1/2) of astegolimabApproximately 85 days
Apparent systemic clearance (CL/F) of astegolimabApproximately 85 days

Trial Locations

Locations (3)

Covance Research Unit - Daytona

🇺🇸

Daytona Beach, Florida, United States

Covance Clinical Research Unit, Inc

🇺🇸

Madison, Wisconsin, United States

Covance Research Unit - Dallas

🇺🇸

Dallas, Texas, United States

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