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Multiple Dose Safety Study of NPT088 in Patients With Mild to Moderate Probable Alzheimer's Disease

Phase 1
Completed
Conditions
Alzheimer Disease
Interventions
Drug: Placebo
Registration Number
NCT03008161
Lead Sponsor
Proclara Biosciences, Inc.
Brief Summary

The purpose of the study is to evaluate the safety and tolerability of multiple doses of NPT088 in patients with mild to moderate probable Alzheimer's Disease. The study will also evaluate the pharmacokinetics, immunogenicity and exploratory pharmacodynamic characteristics of multiple doses of NPT088.

Detailed Description

This study is a multicenter Phase 1, randomized, double-blind, placebo-controlled, multiple-dose, dose-escalation safety and tolerability study of NPT088 or placebo in patients with Probable AD with a MMSE score of 16-27. Enrolled patients will receive an intravenous infusion of NPT088 or placebo once a month for six months during this study. Four dose cohorts are planned with the first two cohorts enrolling 9 patients each (6 NPT088: 3 placebo) and the final two cohorts enrolling 24 patients each (16 NPT088: 8 placebo) for a total of 66 patients (44 NPT088: 22 placebo).

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
83
Inclusion Criteria

For enrollment in the study, participants must

  • be between 50 and 85 years of age, inclusive
  • have a Mini Mental State Examination (MMSE) scores between 16-27 (inclusive)
  • have a Modified Hachinski Score of less than or equal to 4
  • have a diagnosis of Probable Alzheimer's Disease (AD) according to consensus criteria defined by the National Institute on Aging-Alzheimer's Association work group
  • have a Clinical Dementia Rating Scale (CDR) of 0.5 or 1.0, with the memory box score equal to or greater than 0.5
  • have a positive florbetapir positron emission tomography (PET) amyloid scan
  • consent to apolipoprotein E (ApoE) genotyping
  • be willing to undergo repeat Magnetic Resonance Imaging (MRI) and PET imaging
  • be on stable doses of allowed medications for at least 30 days prior to Screening. Concurrent treatment with cholinesterase inhibitors and/or memantine is allowed
  • be in good healthy apart from the clinical diagnosis of AD
  • have a dedicated Caregiver who provides care at least 4 hours a day for 4 days a week and will provide informed consent for their participation
Exclusion Criteria

For enrollment in the study, participants must NOT:

  • have a history of, or screening MRI indicative of any significant brain abnormality
  • have any major medical illness or unstable medical condition or in the opinion of the Investigator have any reason that may interfere with the participants ability to comply with the study procedures and abide by study restrictions or with the ability to interpret safety data
  • reside in a nursing home or need 24-hour care and supervision
  • take excluded medications
  • have exclusionary values on the Screening blood and urine sample
  • have been treated with immunomodulators to treat AD
  • have participated in an investigational drug or device study within 90 days
  • have a known allergy to study drug

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Cohort 3NPT088Participants will receive monthly IV infusions of either mid-high dose NPT088 (16 participants) or placebo (8 participants) for a total of 6 months
Cohort 4PlaceboParticipants will receive monthly IV infusions of either high dose NPT088 (16 participants) or placebo (8 participants) for a total of 6 months
Cohort 1PlaceboParticipants will receive monthly IV infusions of either low dose NPT088 (6 participants) or placebo (3 participants) for a total of 6 months
Cohort 2PlaceboParticipants will receive monthly IV infusions of either mid-low dose NPT088 (6 participants) or placebo (3 participants) for a total of 6 months
Cohort 3PlaceboParticipants will receive monthly IV infusions of either mid-high dose NPT088 (16 participants) or placebo (8 participants) for a total of 6 months
Cohort 4NPT088Participants will receive monthly IV infusions of either high dose NPT088 (16 participants) or placebo (8 participants) for a total of 6 months
Cohort 1NPT088Participants will receive monthly IV infusions of either low dose NPT088 (6 participants) or placebo (3 participants) for a total of 6 months
Cohort 2NPT088Participants will receive monthly IV infusions of either mid-low dose NPT088 (6 participants) or placebo (3 participants) for a total of 6 months
Primary Outcome Measures
NameTimeMethod
Number of patients with adverse eventsBaseline to Week 32
Secondary Outcome Measures
NameTimeMethod
Multiple dose PK CSF concentrations of NPT088Up to Week 32
Multiple dose pharmacokinetic (PK) serum concentrations of NPT088Up to Week 32
Multiple dose immunogenicity of NPT088Up to Week 32

Trial Locations

Locations (23)

Neurology Center of North Orange County

🇺🇸

Fullerton, California, United States

NeuroStudies LLC

🇺🇸

Decatur, Georgia, United States

Princeton Medical Institute

🇺🇸

Princeton, New Jersey, United States

Lehigh Center for Clinical Research

🇺🇸

Allentown, Pennsylvania, United States

Alzheimer's Research and Treatment Center

🇺🇸

Lake Worth, Florida, United States

Southern California Research

🇺🇸

Simi Valley, California, United States

Collaborative Neuroscience Network

🇺🇸

Long Beach, California, United States

Indago Research and Health Center

🇺🇸

Hialeah, Florida, United States

Miami Jewish Health Systems

🇺🇸

Miami, Florida, United States

Medical Research Group of Central Florida

🇺🇸

Orange City, Florida, United States

Associated Neurologists of Southern Connecticut

🇺🇸

Fairfield, Connecticut, United States

ATP Clinical Research, Inc.

🇺🇸

Costa Mesa, California, United States

JEM Research Institute

🇺🇸

Atlantis, Florida, United States

Compass-The Villages

🇺🇸

The Villages, Florida, United States

Progressive Medical Research

🇺🇸

Port Orange, Florida, United States

Medical Research and Health Education Foundation

🇺🇸

Columbus, Georgia, United States

Integrative Clinical Trials, Inc.

🇺🇸

Brooklyn, New York, United States

Alzheimer's Memory Center

🇺🇸

Charlotte, North Carolina, United States

Abington Neurological Associates, Ltd

🇺🇸

Willow Grove, Pennsylvania, United States

Neurology Clinic, PC

🇺🇸

Cordova, Tennessee, United States

Neurological Associates of Albany

🇺🇸

Albany, New York, United States

Compass Research

🇺🇸

Orlando, Florida, United States

Axiom Clinical Research

🇺🇸

Tampa, Florida, United States

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